Angustifodilactone B

Details

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Internal ID 1c6b43ba-4e6f-4515-bfdb-855ef8fd0b75
Taxonomy Lipids and lipid-like molecules > Prenol lipids > Triterpenoids
IUPAC Name (1R,3S,9S,10S,12S,13S,16S,17R,18S)-10,18-dihydroxy-16-[(1R)-1-hydroxy-1-[(2R)-5-methyl-6-oxo-2,3-dihydropyran-2-yl]ethyl]-8,8,13,17-tetramethyl-7-oxapentacyclo[10.7.0.01,3.03,9.013,17]nonadec-4-en-6-one
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C30H42O7/c1-16-7-8-21(36-24(16)34)28(6,35)18-9-11-26(4)19-13-17(31)23-25(2,3)37-22(33)10-12-29(23)15-30(19,29)14-20(32)27(18,26)5/h7,10,12,17-21,23,31-32,35H,8-9,11,13-15H2,1-6H3/t17-,18-,19-,20-,21+,23-,26-,27-,28+,29+,30-/m0/s1
InChI Key QCYCYOUXODNCMX-LDUYZNKBSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C30H42O7
Molecular Weight 514.60 g/mol
Exact Mass 514.29305367 g/mol
Topological Polar Surface Area (TPSA) 113.00 Ų
XlogP 3.80

Synonyms

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(1R,3S,9S,10S,12S,13S,16S,17R,18S)-10,18-dihydroxy-16-((1R)-1-hydroxy-1-((2R)-5-methyl-6-oxo-2,3-dihydropyran-2-yl)ethyl)-8,8,13,17-tetramethyl-7-oxapentacyclo(10.7.0.01,3.03,9.013,17)nonadec-4-en-6-one
(1R,3S,9S,10S,12S,13S,16S,17R,18S)-10,18-dihydroxy-16-[(1R)-1-hydroxy-1-[(2R)-5-methyl-6-oxo-2,3-dihydropyran-2-yl]ethyl]-8,8,13,17-tetramethyl-7-oxapentacyclo[10.7.0.01,3.03,9.013,17]nonadec-4-en-6-one
RefChem:112748
CHEMBL1669431
DTXSID001336050
(1S,3aS,3bS,5S,5aS,10aS,11aR,13S,13aR)-5,13-Dihydroxy-1-{(1R)-1-hydroxy-1-[(2R)-5-methyl-6-oxo-3,6-dihydro-2H-pyran-2-yl]ethyl}-3a,6,6,13a-tetramethyl-1,2,3,3a,3b,4,5,5a,6,12,13,13a-dodecahydro-8H-cyclopenta[5,6]cyclopropa[1,8a]naphtho[2,1-c]oxepin-8-one
dihydroxy-[(1R)-1-hydroxy-1-[(2R)-5-methyl-6-oxo-2,3-dihydropyran-2-yl]ethyl]-tetramethyl-[?]one

2D Structure

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2D Structure of Angustifodilactone B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.14% 91.11%
CHEMBL253 P34972 Cannabinoid CB2 receptor 96.46% 97.25%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 94.53% 95.56%
CHEMBL1937 Q92769 Histone deacetylase 2 91.48% 94.75%
CHEMBL1871 P10275 Androgen Receptor 90.38% 96.43%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 89.36% 99.23%
CHEMBL1806 P11388 DNA topoisomerase II alpha 88.79% 89.00%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 87.88% 97.14%
CHEMBL1994 P08235 Mineralocorticoid receptor 87.64% 100.00%
CHEMBL3137262 O60341 LSD1/CoREST complex 84.91% 97.09%
CHEMBL5608 Q16288 NT-3 growth factor receptor 83.90% 95.89%
CHEMBL3359 P21462 Formyl peptide receptor 1 83.87% 93.56%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 83.28% 93.03%
CHEMBL2007 P16234 Platelet-derived growth factor receptor alpha 82.63% 91.07%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 82.23% 82.69%
CHEMBL4303 P08238 Heat shock protein HSP 90-beta 81.52% 96.77%
CHEMBL1293249 Q13887 Kruppel-like factor 5 80.43% 86.33%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Kadsura angustifolia

Cross-Links

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PubChem 51003491
LOTUS LTS0200763
wikiData Q105218657