Varamine A

Details

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Internal ID 7dc017f6-b78b-4f6c-a910-aa40908a383c
Taxonomy Organoheterocyclic compounds > Quinolines and derivatives > Benzoquinolines > Pyridoacridines > Pyrido[2,3,4-kl]acridines
IUPAC Name N-[2-(12-methoxy-11-methylsulfanyl-8,14-diazatetracyclo[7.7.1.02,7.013,17]heptadeca-1(17),2,4,6,9,11,13,15-octaen-10-yl)ethyl]propanamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C22H23N3O2S/c1-4-17(26)23-11-10-15-19-18-14(13-7-5-6-8-16(13)25-19)9-12-24-20(18)21(27-2)22(15)28-3/h5-9,12,25H,4,10-11H2,1-3H3,(H,23,26)
InChI Key ATGZYGBQIFBZRA-UHFFFAOYSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C22H23N3O2S
Molecular Weight 393.50 g/mol
Exact Mass 393.15109816 g/mol
Topological Polar Surface Area (TPSA) 88.60 Ų
XlogP 4.00

Synonyms

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122093-14-5
DTXSID10153495
Propanamide, N-(2-(4-methoxy-5-(methylthio)-7H-pyrido(2,3,4-kl)acridin-6-yl)ethyl)-

2D Structure

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2D Structure of Varamine A

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL240 Q12809 HERG 98.56% 89.76%
CHEMBL255 P29275 Adenosine A2b receptor 98.38% 98.59%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.35% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.21% 96.09%
CHEMBL4040 P28482 MAP kinase ERK2 95.74% 83.82%
CHEMBL1806 P11388 DNA topoisomerase II alpha 95.19% 89.00%
CHEMBL2535 P11166 Glucose transporter 95.18% 98.75%
CHEMBL2581 P07339 Cathepsin D 95.00% 98.95%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 94.34% 94.45%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 93.64% 99.23%
CHEMBL3060 Q9Y345 Glycine transporter 2 90.18% 99.17%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 89.89% 85.14%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 89.41% 94.00%
CHEMBL1914 P06276 Butyrylcholinesterase 88.88% 95.00%
CHEMBL1781 P11387 DNA topoisomerase I 88.10% 97.00%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 85.28% 96.00%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 84.73% 95.56%
CHEMBL1937 Q92769 Histone deacetylase 2 83.54% 94.75%
CHEMBL230 P35354 Cyclooxygenase-2 83.24% 89.63%
CHEMBL1868 P17948 Vascular endothelial growth factor receptor 1 82.32% 96.47%
CHEMBL4208 P20618 Proteasome component C5 82.10% 90.00%
CHEMBL1287628 Q9Y5S8 NADPH oxidase 1 81.94% 95.48%
CHEMBL3401 O75469 Pregnane X receptor 81.57% 94.73%
CHEMBL2094127 P06493 Cyclin-dependent kinase 1/cyclin B 81.31% 96.00%
CHEMBL2378 P30307 Dual specificity phosphatase Cdc25C 80.02% 96.67%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

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PubChem 180091
LOTUS LTS0082024
wikiData Q83020383