Unk-D-Ser(1)-D-Pip-Gly-Sar-N(Me)Val-(2).Unk-Ser(2)-D-Pip-Gly-Sar-D-N(Me)Val-(1)

Details

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Internal ID 011ff8ec-9cb6-4860-8b21-25963b339d1c
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name 3-hydroxy-N-[(3S,7S,16R,23R,27R,36R)-23-[(3-hydroxyquinoline-2-carbonyl)amino]-8,11,28,31-tetramethyl-2,6,9,12,15,22,26,29,32,35-decaoxo-7,27-di(propan-2-yl)-5,25-dioxa-1,8,11,14,21,28,31,34-octazatricyclo[34.4.0.016,21]tetracontan-3-yl]quinoline-2-carboxamide
SMILES (Canonical) CC(C)C1C(=O)OCC(C(=O)N2CCCCC2C(=O)NCC(=O)N(CC(=O)N(C(C(=O)OCC(C(=O)N3CCCCC3C(=O)NCC(=O)N(CC(=O)N1C)C)NC(=O)C4=NC5=CC=CC=C5C=C4O)C(C)C)C)C)NC(=O)C6=NC7=CC=CC=C7C=C6O
SMILES (Isomeric) CC(C)[C@H]1C(=O)OC[C@@H](C(=O)N2CCCC[C@@H]2C(=O)NCC(=O)N(CC(=O)N([C@@H](C(=O)OC[C@H](C(=O)N3CCCC[C@@H]3C(=O)NCC(=O)N(CC(=O)N1C)C)NC(=O)C4=NC5=CC=CC=C5C=C4O)C(C)C)C)C)NC(=O)C6=NC7=CC=CC=C7C=C6O
InChI InChI=1S/C60H76N12O16/c1-33(2)51-59(85)87-31-39(65-55(81)49-43(73)25-35-17-9-11-19-37(35)63-49)57(83)71-23-15-13-21-41(71)53(79)62-28-46(76)68(6)30-48(78)70(8)52(34(3)4)60(86)88-32-40(66-56(82)50-44(74)26-36-18-10-12-20-38(36)64-50)58(84)72-24-16-14-22-42(72)54(80)61-27-45(75)67(5)29-47(77)69(51)7/h9-12,17-20,25-26,33-34,39-42,51-52,73-74H,13-16,21-24,27-32H2,1-8H3,(H,61,80)(H,62,79)(H,65,81)(H,66,82)/t39-,40+,41-,42-,51-,52+/m1/s1
InChI Key WXIVYIYCEBUEHL-HLBGSBEJSA-N
Popularity 9 references in papers

Physical and Chemical Properties

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Molecular Formula C60H76N12O16
Molecular Weight 1221.30 g/mol
Exact Mass 1220.55022438 g/mol
Topological Polar Surface Area (TPSA) 357.00 Ų
XlogP 3.80

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Unk-D-Ser(1)-D-Pip-Gly-Sar-N(Me)Val-(2).Unk-Ser(2)-D-Pip-Gly-Sar-D-N(Me)Val-(1)

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 98.86% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.61% 96.09%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 98.37% 85.14%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 95.49% 93.03%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 94.92% 91.11%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 93.47% 99.23%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 91.17% 90.71%
CHEMBL1806 P11388 DNA topoisomerase II alpha 90.70% 89.00%
CHEMBL3524 P56524 Histone deacetylase 4 90.08% 92.97%
CHEMBL2535 P11166 Glucose transporter 88.97% 98.75%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 88.77% 95.56%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 88.68% 100.00%
CHEMBL1907598 P05106 Integrin alpha-V/beta-3 88.51% 95.71%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 87.08% 94.00%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 86.50% 88.42%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 85.50% 99.15%
CHEMBL3401 O75469 Pregnane X receptor 85.04% 94.73%
CHEMBL2378 P30307 Dual specificity phosphatase Cdc25C 84.85% 96.67%
CHEMBL3038469 P24941 CDK2/Cyclin A 84.39% 91.38%
CHEMBL204 P00734 Thrombin 84.28% 96.01%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 84.14% 97.64%
CHEMBL253 P34972 Cannabinoid CB2 receptor 82.59% 97.25%
CHEMBL2553 Q15418 Ribosomal protein S6 kinase alpha 1 82.59% 85.11%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 82.55% 98.33%
CHEMBL4531 P17931 Galectin-3 82.42% 96.90%
CHEMBL2095172 P14867 GABA-A receptor; alpha-1/beta-2/gamma-2 81.87% 92.67%
CHEMBL5028 O14672 ADAM10 81.14% 97.50%
CHEMBL4073 P09237 Matrix metalloproteinase 7 80.99% 97.56%
CHEMBL4208 P20618 Proteasome component C5 80.86% 90.00%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 80.34% 93.10%
CHEMBL5409 Q8TDU6 G-protein coupled bile acid receptor 1 80.03% 93.65%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139588936
LOTUS LTS0132731
wikiData Q105314666