Unguisin A

Details

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Internal ID 7c53f368-d24b-4fff-aca9-8657097b73ad
Taxonomy Organic acids and derivatives > Peptidomimetics > Hybrid peptides
IUPAC Name (3R,6R,9R,12S,15R,18R)-12-benzyl-3-(1H-indol-3-ylmethyl)-6,18-dimethyl-9,15-di(propan-2-yl)-1,4,7,10,13,16,19-heptazacyclotricosane-2,5,8,11,14,17,20-heptone
SMILES (Canonical) CC1C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NCCCC(=O)N1)CC2=CNC3=CC=CC=C32)C)C(C)C)CC4=CC=CC=C4)C(C)C
SMILES (Isomeric) C[C@@H]1C(=O)N[C@@H](C(=O)N[C@H](C(=O)N[C@@H](C(=O)N[C@@H](C(=O)N[C@@H](C(=O)NCCCC(=O)N1)CC2=CNC3=CC=CC=C32)C)C(C)C)CC4=CC=CC=C4)C(C)C
InChI InChI=1S/C40H54N8O7/c1-22(2)33-39(54)44-25(6)35(50)45-31(20-27-21-42-29-16-11-10-15-28(27)29)37(52)41-18-12-17-32(49)43-24(5)36(51)47-34(23(3)4)40(55)46-30(38(53)48-33)19-26-13-8-7-9-14-26/h7-11,13-16,21-25,30-31,33-34,42H,12,17-20H2,1-6H3,(H,41,52)(H,43,49)(H,44,54)(H,45,50)(H,46,55)(H,47,51)(H,48,53)/t24-,25-,30+,31-,33-,34-/m1/s1
InChI Key JLLVQPKAQVOYFS-KVOZXUITSA-N
Popularity 6 references in papers

Physical and Chemical Properties

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Molecular Formula C40H54N8O7
Molecular Weight 758.90 g/mol
Exact Mass 758.41154609 g/mol
Topological Polar Surface Area (TPSA) 220.00 Ų
XlogP 3.30

Synonyms

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226956-06-5
(3R,6R,9R,12S,15R,18R)-12-Benzyl-3-(1H-indol-3-ylmethyl)-6,18-dimethyl-9,15-di(propan-2-yl)-1,4,7,10,13,16,19-heptazacyclotricosane-2,5,8,11,14,17,20-heptone
RefChem:193128
cyclo(D-alanyl-D-tryptophyl-4-aminobutanoyl-D-alanyl-D-valyl-L-phenylalanyl-D-valyl)
orb1943865
CHEBI:203737
C40H54N8O7
DA-78781
HY-133801
CS-0133187
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

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2D Structure of Unguisin A

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.49% 98.95%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.46% 91.11%
CHEMBL4040 P28482 MAP kinase ERK2 98.36% 83.82%
CHEMBL5103 Q969S8 Histone deacetylase 10 97.41% 90.08%
CHEMBL3310 Q96DB2 Histone deacetylase 11 96.33% 88.56%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 96.17% 97.64%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.19% 95.56%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 94.51% 96.09%
CHEMBL1937 Q92769 Histone deacetylase 2 93.85% 94.75%
CHEMBL1949 P62937 Cyclophilin A 93.69% 98.57%
CHEMBL3192 Q9BY41 Histone deacetylase 8 93.33% 93.99%
CHEMBL3137262 O60341 LSD1/CoREST complex 92.94% 97.09%
CHEMBL1914 P06276 Butyrylcholinesterase 90.85% 95.00%
CHEMBL3155 P34969 Serotonin 7 (5-HT7) receptor 90.65% 90.71%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 89.70% 85.14%
CHEMBL2288 Q13526 Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 89.57% 91.71%
CHEMBL2095172 P14867 GABA-A receptor; alpha-1/beta-2/gamma-2 87.74% 92.67%
CHEMBL2996 Q05655 Protein kinase C delta 87.23% 97.79%
CHEMBL2373 P21730 C5a anaphylatoxin chemotactic receptor 85.91% 92.62%
CHEMBL1951 P21397 Monoamine oxidase A 85.52% 91.49%
CHEMBL255 P29275 Adenosine A2b receptor 85.47% 98.59%
CHEMBL213 P08588 Beta-1 adrenergic receptor 85.05% 95.56%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 83.92% 95.50%
CHEMBL253 P34972 Cannabinoid CB2 receptor 82.84% 97.25%
CHEMBL4644 P41968 Melanocortin receptor 3 82.06% 99.52%
CHEMBL5608 Q16288 NT-3 growth factor receptor 81.78% 95.89%
CHEMBL5896 O75164 Lysine-specific demethylase 4A 81.21% 99.09%
CHEMBL4608 P33032 Melanocortin receptor 5 81.12% 97.00%
CHEMBL5805 Q9NR97 Toll-like receptor 8 80.84% 96.25%
CHEMBL2535 P11166 Glucose transporter 80.60% 98.75%
CHEMBL1293287 P14735 Insulin-degrading enzyme 80.54% 88.10%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 10652700
LOTUS LTS0071830
wikiData Q77380564