Tubulysin C

Details

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Internal ID 42a3742f-c584-45d8-a9c6-2587aa2b3df3
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Dipeptides
IUPAC Name (2S,4R)-4-[[2-[(1R,3R)-1-acetyloxy-4-methyl-3-[[(2S,3S)-3-methyl-2-[[(2R)-1-methylpiperidine-2-carbonyl]amino]pentanoyl]-(propanoyloxymethyl)amino]pentyl]-1,3-thiazole-4-carbonyl]amino]-5-(4-hydroxyphenyl)-2-methylpentanoic acid
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C41H61N5O10S/c1-9-25(5)36(44-38(51)32-13-11-12-18-45(32)8)40(52)46(23-55-35(49)10-2)33(24(3)4)21-34(56-27(7)47)39-43-31(22-57-39)37(50)42-29(19-26(6)41(53)54)20-28-14-16-30(48)17-15-28/h14-17,22,24-26,29,32-34,36,48H,9-13,18-21,23H2,1-8H3,(H,42,50)(H,44,51)(H,53,54)/t25-,26-,29+,32+,33+,34+,36-/m0/s1
InChI Key NZCNGJHOIKMMCG-UZRVFEFTSA-N
Popularity 0 references in papers

Physical and Chemical Properties

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Molecular Formula C41H61N5O10S
Molecular Weight 816.00 g/mol
Exact Mass 815.41391433 g/mol
Topological Polar Surface Area (TPSA) 233.00 Ų
XlogP 3.90

Synonyms

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205304-88-7
072P54KU0L
UNII-072P54KU0L
(2S,4R)-4-[[2-[(1R,3R)-1-acetyloxy-4-methyl-3-[[(2S,3S)-3-methyl-2-[[(2R)-1-methylpiperidine-2-carbonyl]amino]pentanoyl]-(propanoyloxymethyl)amino]pentyl]-1,3-thiazole-4-carbonyl]amino]-5-(4-hydroxyphenyl)-2-methylpentanoic acid
Benzenepentanoic acid, gamma-(((2-((1R,3R)-1-(acetyloxy)-4-methyl-3-(((2S,3S)-3-methyl-2-((((2R)-1-methyl-2-piperidinyl)carbonyl)amino)-1-oxopentyl)((1-oxopropoxy)methyl)amino)pentyl)-4-thiazolyl)carbonyl)amino)-4-hydroxy-alpha-methyl-, (alphaS,.ga
SCHEMBL24218753
EX-A5466C
HY-N2347
AKOS040740942
CS-0021784
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

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2D Structure of Tubulysin C

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.80% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.87% 96.09%
CHEMBL4072 P07858 Cathepsin B 98.78% 93.67%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 97.77% 93.10%
CHEMBL253 P34972 Cannabinoid CB2 receptor 95.85% 97.25%
CHEMBL215 P09917 Arachidonate 5-lipoxygenase 94.79% 92.68%
CHEMBL335 P18031 Protein-tyrosine phosphatase 1B 94.40% 95.17%
CHEMBL340 P08684 Cytochrome P450 3A4 93.48% 91.19%
CHEMBL221 P23219 Cyclooxygenase-1 93.45% 90.17%
CHEMBL3359 P21462 Formyl peptide receptor 1 93.03% 93.56%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 91.02% 93.00%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 89.13% 90.71%
CHEMBL240 Q12809 HERG 88.73% 89.76%
CHEMBL3060 Q9Y345 Glycine transporter 2 88.70% 99.17%
CHEMBL2514 O95665 Neurotensin receptor 2 88.23% 100.00%
CHEMBL4835 P00338 L-lactate dehydrogenase A chain 87.95% 95.34%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 87.44% 85.14%
CHEMBL3837 P07711 Cathepsin L 87.14% 96.61%
CHEMBL5608 Q16288 NT-3 growth factor receptor 86.03% 95.89%
CHEMBL226 P30542 Adenosine A1 receptor 85.78% 95.93%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 85.23% 96.90%
CHEMBL4227 P25090 Lipoxin A4 receptor 84.57% 100.00%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 83.53% 97.64%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 83.49% 99.15%
CHEMBL4208 P20618 Proteasome component C5 83.40% 90.00%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 83.40% 95.56%
CHEMBL3430907 Q96GD4 Aurora kinase B/Inner centromere protein 82.79% 97.50%
CHEMBL268 P43235 Cathepsin K 82.36% 96.85%
CHEMBL2535 P11166 Glucose transporter 82.09% 98.75%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 81.47% 95.89%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 81.46% 98.33%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 81.14% 94.45%
CHEMBL2073 P07947 Tyrosine-protein kinase YES 80.15% 83.14%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 11262920
LOTUS LTS0121563
wikiData Q77491093