Tsushimycin

Details

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Internal ID bb87bd63-2d32-4822-a687-deabb0f0e373
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Oligopeptides
IUPAC Name (3S)-4-[[(3S,7S,13S,16R,22S,28S,31S,34R)-16-(1-aminoethyl)-31-(1-carboxyethyl)-22,28-bis(carboxymethyl)-4-methyl-2,6,12,15,18,21,24,27,30,33-decaoxo-13-propan-2-yl-1,5,11,14,17,20,23,26,29,32-decazatricyclo[32.4.0.07,11]octatriacontan-3-yl]amino]-3-[[(Z)-12-methyltridec-3-enoyl]amino]-4-oxobutanoic acid
SMILES (Canonical) CC1C(C(=O)N2CCCCC2C(=O)NC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)N3CCCC3C(=O)N1)C(C)C)C(C)N)CC(=O)O)CC(=O)O)C(C)C(=O)O)NC(=O)C(CC(=O)O)NC(=O)CC=CCCCCCCCC(C)C
SMILES (Isomeric) CC1[C@@H](C(=O)N2CCCC[C@@H]2C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)NCC(=O)N[C@@H](C(=O)N[C@H](C(=O)N3CCC[C@H]3C(=O)N1)C(C)C)C(C)N)CC(=O)O)CC(=O)O)C(C)C(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)C/C=C\CCCCCCCC(C)C
InChI InChI=1S/C59H93N13O20/c1-30(2)19-14-12-10-8-9-11-13-15-22-40(73)64-37(27-45(80)81)52(84)70-49-34(7)63-53(85)39-21-18-24-72(39)57(89)46(31(3)4)68-56(88)48(33(6)60)67-42(75)29-62-50(82)35(25-43(76)77)65-41(74)28-61-51(83)36(26-44(78)79)66-55(87)47(32(5)59(91)92)69-54(86)38-20-16-17-23-71(38)58(49)90/h13,15,30-39,46-49H,8-12,14,16-29,60H2,1-7H3,(H,61,83)(H,62,82)(H,63,85)(H,64,73)(H,65,74)(H,66,87)(H,67,75)(H,68,88)(H,69,86)(H,70,84)(H,76,77)(H,78,79)(H,80,81)(H,91,92)/b15-13-/t32?,33?,34?,35-,36-,37-,38+,39-,46-,47-,48+,49-/m0/s1
InChI Key BYWOWQCRVFUOLF-AQZAFBPESA-N
Popularity 6 references in papers

Physical and Chemical Properties

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Molecular Formula C59H93N13O20
Molecular Weight 1304.40 g/mol
Exact Mass 1303.66598241 g/mol
Topological Polar Surface Area (TPSA) 507.00 Ų
XlogP -2.30

Synonyms

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11054-63-0

2D Structure

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2D Structure of Tsushimycin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.75% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.41% 96.09%
CHEMBL236 P41143 Delta opioid receptor 98.95% 99.35%
CHEMBL4801 P29466 Caspase-1 98.94% 96.85%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.53% 91.11%
CHEMBL226 P30542 Adenosine A1 receptor 97.83% 95.93%
CHEMBL5469 Q14289 Protein tyrosine kinase 2 beta 97.14% 91.03%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 96.34% 93.00%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 95.55% 96.11%
CHEMBL3524 P56524 Histone deacetylase 4 95.35% 92.97%
CHEMBL3060 Q9Y345 Glycine transporter 2 95.31% 99.17%
CHEMBL5103 Q969S8 Histone deacetylase 10 94.97% 90.08%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 93.89% 90.71%
CHEMBL1902 P62942 FK506-binding protein 1A 93.69% 97.05%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 93.55% 82.38%
CHEMBL221 P23219 Cyclooxygenase-1 93.47% 90.17%
CHEMBL4071 P08311 Cathepsin G 93.16% 94.64%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 92.67% 95.50%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 92.02% 98.33%
CHEMBL5203 P33316 dUTP pyrophosphatase 90.89% 99.18%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 90.53% 96.90%
CHEMBL4588 P22894 Matrix metalloproteinase 8 89.85% 94.66%
CHEMBL5608 Q16288 NT-3 growth factor receptor 89.41% 95.89%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 89.39% 94.45%
CHEMBL4979 P13866 Sodium/glucose cotransporter 1 89.13% 98.24%
CHEMBL3359 P21462 Formyl peptide receptor 1 87.88% 93.56%
CHEMBL2413 P32246 C-C chemokine receptor type 1 87.19% 89.50%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 86.94% 93.03%
CHEMBL2781 P19634 Sodium/hydrogen exchanger 1 86.86% 90.24%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 86.84% 90.93%
CHEMBL3468 P55210 Caspase-7 86.66% 95.68%
CHEMBL2443 P49862 Kallikrein 7 85.56% 94.00%
CHEMBL3137262 O60341 LSD1/CoREST complex 85.54% 97.09%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 85.41% 96.38%
CHEMBL1806 P11388 DNA topoisomerase II alpha 84.71% 89.00%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 84.56% 97.64%
CHEMBL4394 Q9NYA1 Sphingosine kinase 1 84.41% 96.03%
CHEMBL333 P08253 Matrix metalloproteinase-2 83.75% 96.31%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 83.62% 96.47%
CHEMBL2514 O95665 Neurotensin receptor 2 83.57% 100.00%
CHEMBL2094135 Q96BI3 Gamma-secretase 83.46% 98.05%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 83.42% 95.56%
CHEMBL4462 Q8IXJ6 NAD-dependent deacetylase sirtuin 2 83.04% 90.24%
CHEMBL1907598 P05106 Integrin alpha-V/beta-3 82.96% 95.71%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 82.17% 94.33%
CHEMBL2001 Q9H244 Purinergic receptor P2Y12 81.53% 96.00%
CHEMBL340 P08684 Cytochrome P450 3A4 81.35% 91.19%
CHEMBL4618 P09960 Leukotriene A4 hydrolase 81.30% 97.86%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 80.87% 88.42%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 72201064
LOTUS LTS0080215
wikiData Q104950025