Topsentin

Details

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Internal ID 7b38a97b-eff2-4ac9-b778-303b379847f6
Taxonomy Organoheterocyclic compounds > Indoles and derivatives > Indolecarboxylic acids and derivatives
IUPAC Name (6-hydroxy-1H-indol-3-yl)-[5-(1H-indol-3-yl)-1H-imidazol-2-yl]methanone
SMILES (Canonical) C1=CC=C2C(=C1)C(=CN2)C3=CN=C(N3)C(=O)C4=CNC5=C4C=CC(=C5)O
SMILES (Isomeric) C1=CC=C2C(=C1)C(=CN2)C3=CN=C(N3)C(=O)C4=CNC5=C4C=CC(=C5)O
InChI InChI=1S/C20H14N4O2/c25-11-5-6-13-15(9-22-17(13)7-11)19(26)20-23-10-18(24-20)14-8-21-16-4-2-1-3-12(14)16/h1-10,21-22,25H,(H,23,24)
InChI Key TVPNFKRGOFJQOO-UHFFFAOYSA-N
Popularity 21 references in papers

Physical and Chemical Properties

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Molecular Formula C20H14N4O2
Molecular Weight 342.30 g/mol
Exact Mass 342.11167570 g/mol
Topological Polar Surface Area (TPSA) 97.60 Ų
XlogP 3.30

Synonyms

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112515-43-2
Topsentin B1
CHEMBL303282
Methanone,(6-hydroxy-1H-indol-3-yl)[5-(1H-indol-3-yl)-1H-imidazol-2-yl]-
Topsentine B 1
SCHEMBL19235593
DTXSID30150087
TVPNFKRGOFJQOO-UHFFFAOYSA-N
BDBM50287721
(6-hydroxy-1H-indol-3-yl)-[5-(1H-indol-3-yl)-1H-imidazol-2-yl]methanone
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

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2D Structure of Topsentin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2535 P11166 Glucose transporter 97.42% 98.75%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 96.13% 91.11%
CHEMBL2035 P08912 Muscarinic acetylcholine receptor M5 95.01% 94.62%
CHEMBL2095172 P14867 GABA-A receptor; alpha-1/beta-2/gamma-2 94.17% 92.67%
CHEMBL213 P08588 Beta-1 adrenergic receptor 91.61% 95.56%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 90.55% 95.56%
CHEMBL2716 Q8WUI4 Histone deacetylase 7 90.32% 89.44%
CHEMBL1951 P21397 Monoamine oxidase A 90.30% 91.49%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 89.79% 94.00%
CHEMBL4145 Q9UKV0 Histone deacetylase 9 88.17% 85.49%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 87.77% 99.23%
CHEMBL3310 Q96DB2 Histone deacetylase 11 87.71% 88.56%
CHEMBL2708 Q16584 Mitogen-activated protein kinase kinase kinase 11 87.66% 81.14%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 87.27% 96.09%
CHEMBL1806 P11388 DNA topoisomerase II alpha 86.89% 89.00%
CHEMBL2581 P07339 Cathepsin D 85.21% 98.95%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 84.52% 93.10%
CHEMBL2292 Q13627 Dual-specificity tyrosine-phosphorylation regulated kinase 1A 84.36% 93.24%
CHEMBL1781 P11387 DNA topoisomerase I 84.15% 97.00%
CHEMBL2563 Q9UQL6 Histone deacetylase 5 83.46% 89.67%
CHEMBL3060 Q9Y345 Glycine transporter 2 82.16% 99.17%
CHEMBL1868 P17948 Vascular endothelial growth factor receptor 1 81.44% 96.47%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 81.29% 99.15%
CHEMBL4101 P17612 cAMP-dependent protein kinase alpha-catalytic subunit 80.49% 82.86%
CHEMBL4208 P20618 Proteasome component C5 80.09% 90.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 72457
LOTUS LTS0084541
wikiData Q83016025