Thalassospiramide B2

Details

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Internal ID b4b4fe84-9730-413a-a91b-76debc85f3e8
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name (Z)-N-[(2S,3S)-5-[[(2S)-1-[[(2S,3S)-1,3-dihydroxy-5-[[(2S)-1-[[(3S,6S,11R)-3-[(4-hydroxyphenyl)methyl]-4-methyl-2,5,8-trioxo-6-propan-2-yl-1-oxa-4,7-diazacyclododec-9-en-11-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-5-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1,3-dihydroxy-5-oxopentan-2-yl]dec-3-enamide
SMILES (Canonical) CCCCCCC=CCC(=O)NC(CO)C(CC(=O)NC(C(C)C)C(=O)NC(CO)C(CC(=O)NC(C(C)C)C(=O)NC1COC(=O)C(N(C(=O)C(NC(=O)C=C1)C(C)C)C)CC2=CC=C(C=C2)O)O)O
SMILES (Isomeric) CCCCCC/C=C\CC(=O)N[C@@H](CO)[C@H](CC(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CO)[C@H](CC(=O)N[C@@H](C(C)C)C(=O)N[C@H]1COC(=O)[C@@H](N(C(=O)[C@@H](NC(=O)C=C1)C(C)C)C)CC2=CC=C(C=C2)O)O)O
InChI InChI=1S/C50H79N7O14/c1-9-10-11-12-13-14-15-16-40(63)52-35(26-58)38(61)24-42(65)56-45(30(4)5)48(68)53-36(27-59)39(62)25-43(66)55-44(29(2)3)47(67)51-33-19-22-41(64)54-46(31(6)7)49(69)57(8)37(50(70)71-28-33)23-32-17-20-34(60)21-18-32/h14-15,17-22,29-31,33,35-39,44-46,58-62H,9-13,16,23-28H2,1-8H3,(H,51,67)(H,52,63)(H,53,68)(H,54,64)(H,55,66)(H,56,65)/b15-14-,22-19?/t33-,35+,36+,37+,38+,39+,44+,45+,46+/m1/s1
InChI Key GCLLLWFQLSIGIH-FFIMJHRBSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C50H79N7O14
Molecular Weight 1002.20 g/mol
Exact Mass 1001.56850022 g/mol
Topological Polar Surface Area (TPSA) 322.00 Ų
XlogP 2.50

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Thalassospiramide B2

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.98% 98.95%
CHEMBL5103 Q969S8 Histone deacetylase 10 98.94% 90.08%
CHEMBL3060 Q9Y345 Glycine transporter 2 98.68% 99.17%
CHEMBL3891 P07384 Calpain 1 97.76% 93.04%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.16% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.00% 96.09%
CHEMBL4588 P22894 Matrix metalloproteinase 8 96.03% 94.66%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 94.80% 94.45%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 93.95% 93.00%
CHEMBL4072 P07858 Cathepsin B 93.74% 93.67%
CHEMBL3892 Q99500 Sphingosine 1-phosphate receptor Edg-3 93.47% 97.29%
CHEMBL2563 Q9UQL6 Histone deacetylase 5 92.48% 89.67%
CHEMBL2955 O95136 Sphingosine 1-phosphate receptor Edg-5 92.24% 92.86%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 91.57% 90.71%
CHEMBL1806 P11388 DNA topoisomerase II alpha 90.72% 89.00%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 89.64% 95.89%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 89.33% 93.10%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 88.32% 96.90%
CHEMBL4769 O95749 Geranylgeranyl pyrophosphate synthetase 87.22% 92.08%
CHEMBL3359 P21462 Formyl peptide receptor 1 86.79% 93.56%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 86.54% 100.00%
CHEMBL3776 Q14790 Caspase-8 86.00% 97.06%
CHEMBL3310 Q96DB2 Histone deacetylase 11 85.82% 88.56%
CHEMBL5852 Q96P65 Pyroglutamylated RFamide peptide receptor 85.69% 85.00%
CHEMBL253 P34972 Cannabinoid CB2 receptor 85.10% 97.25%
CHEMBL2514 O95665 Neurotensin receptor 2 84.80% 100.00%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 84.61% 95.50%
CHEMBL1781 P11387 DNA topoisomerase I 84.45% 97.00%
CHEMBL220 P22303 Acetylcholinesterase 83.83% 94.45%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 83.74% 95.56%
CHEMBL3137262 O60341 LSD1/CoREST complex 82.73% 97.09%
CHEMBL4208 P20618 Proteasome component C5 81.79% 90.00%
CHEMBL3004 P33527 Multidrug resistance-associated protein 1 81.64% 96.37%
CHEMBL5261 Q7L7X3 Serine/threonine-protein kinase TAO1 81.36% 89.33%
CHEMBL4227 P25090 Lipoxin A4 receptor 80.99% 100.00%
CHEMBL268 P43235 Cathepsin K 80.48% 96.85%
CHEMBL3430907 Q96GD4 Aurora kinase B/Inner centromere protein 80.31% 97.50%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139587980
LOTUS LTS0125897
wikiData Q105006338