Syringomycin

Details

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Internal ID 076b45e1-f365-47f8-ba1d-529547381948
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name (2S)-2-[(3S,6S,9Z,12S,15S,18S,21R,24R,27S)-18,21-bis(2-aminoethyl)-12-benzyl-3-[(1S)-2-chloro-1-hydroxyethyl]-15-[3-(diaminomethylideneamino)propyl]-9-ethylidene-27-[[(3S)-3-hydroxydodecanoyl]amino]-24-(hydroxymethyl)-2,5,8,11,14,17,20,23,26-nonaoxo-1-oxa-4,7,10,13,16,19,22,25-octazacyclooctacos-6-yl]-2-hydroxyacetic acid
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C53H85ClN14O17/c1-3-5-6-7-8-9-13-17-30(70)25-39(72)60-37-28-85-52(84)40(38(71)26-54)67-50(81)41(42(73)51(82)83)68-43(74)31(4-2)61-47(78)35(24-29-15-11-10-12-16-29)65-44(75)32(18-14-23-59-53(57)58)62-45(76)33(19-21-55)63-46(77)34(20-22-56)64-48(79)36(27-69)66-49(37)80/h4,10-12,15-16,30,32-38,40-42,69-71,73H,3,5-9,13-14,17-28,55-56H2,1-2H3,(H,60,72)(H,61,78)(H,62,76)(H,63,77)(H,64,79)(H,65,75)(H,66,80)(H,67,81)(H,68,74)(H,82,83)(H4,57,58,59)/b31-4-/t30-,32-,33-,34+,35-,36+,37-,38+,40-,41-,42-/m0/s1
InChI Key ZQVJBRJGDVZANE-MXDMHAPNSA-N
Popularity 62 references in papers

Physical and Chemical Properties

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Molecular Formula C53H85ClN14O17
Molecular Weight 1225.80 g/mol
Exact Mass 1224.5905650 g/mol
Topological Polar Surface Area (TPSA) 523.00 Ų
XlogP -2.90

Synonyms

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(2S)-2-[(3S,6S,9Z,12S,15S,18S,21R,24R,27S)-18,21-bis(2-aminoethyl)-12-benzyl-3-[(1S)-2-chloro-1-hydroxyethyl]-15-[3-(diaminomethylideneamino)propyl]-9-ethylidene-27-[[(3S)-3-hydroxydodecanoyl]amino]-24-(hydroxymethyl)-2,5,8,11,14,17,20,23,26-nonaoxo-1-oxa-4,7,10,13,16,19,22,25-octazacyclooctacos-6-yl]-2-hydroxyacetic acid

2D Structure

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2D Structure of Syringomycin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.71% 91.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 99.70% 94.45%
CHEMBL2581 P07339 Cathepsin D 99.07% 98.95%
CHEMBL4040 P28482 MAP kinase ERK2 98.79% 83.82%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.70% 96.09%
CHEMBL3060 Q9Y345 Glycine transporter 2 96.64% 99.17%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 94.75% 92.88%
CHEMBL230 P35354 Cyclooxygenase-2 93.56% 89.63%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 93.04% 95.56%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 92.89% 97.64%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 92.42% 96.47%
CHEMBL3137262 O60341 LSD1/CoREST complex 92.27% 97.09%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 92.06% 95.00%
CHEMBL3892 Q99500 Sphingosine 1-phosphate receptor Edg-3 91.09% 97.29%
CHEMBL218 P21554 Cannabinoid CB1 receptor 89.93% 96.61%
CHEMBL2327 P21452 Neurokinin 2 receptor 89.25% 98.89%
CHEMBL221 P23219 Cyclooxygenase-1 88.87% 90.17%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 87.49% 95.50%
CHEMBL3401 O75469 Pregnane X receptor 87.44% 94.73%
CHEMBL299 P17252 Protein kinase C alpha 87.30% 98.03%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 86.73% 96.11%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 86.65% 90.71%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 85.97% 100.00%
CHEMBL4769 O95749 Geranylgeranyl pyrophosphate synthetase 85.93% 92.08%
CHEMBL1255126 O15151 Protein Mdm4 83.59% 90.20%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 83.44% 97.14%
CHEMBL3475 P05121 Plasminogen activator inhibitor-1 83.37% 83.00%
CHEMBL1293267 Q9HC97 G-protein coupled receptor 35 83.31% 89.34%
CHEMBL2072 P35499 Sodium channel protein type IV alpha subunit 82.64% 92.32%
CHEMBL5103 Q969S8 Histone deacetylase 10 82.31% 90.08%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 82.23% 96.90%
CHEMBL4581 P52732 Kinesin-like protein 1 82.18% 93.18%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 82.15% 82.69%
CHEMBL1293249 Q13887 Kruppel-like factor 5 81.69% 86.33%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 80.71% 93.00%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 80.32% 88.42%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 11966095
LOTUS LTS0123401
wikiData Q105381778