Subterisin

Details

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Internal ID ce792154-599d-4b94-b495-02e496caef8c
Taxonomy Organic acids and derivatives > Peptidomimetics > Hybrid peptides
IUPAC Name 2-[(3S,14S,17S,20S,23S,29S)-14-[[(2S)-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-1-[(2S)-2-(carboxymethylcarbamoyl)pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]carbamoyl]-17-[(2S)-butan-2-yl]-20-[3-(diaminomethylideneamino)propyl]-2,8,11,16,19,22,25,28-octaoxo-1,7,10,15,18,21,24,27-octazatricyclo[27.3.0.03,7]dotriacontan-23-yl]acetic acid
SMILES (Canonical) CCC(C)C1C(=O)NC(CCC(=O)NCC(=O)N2CCCC2C(=O)N3CCCC3C(=O)NCC(=O)NC(C(=O)NC(C(=O)N1)CCCN=C(N)N)CC(=O)O)C(=O)NC(CC4=CC=CC=C4)C(=O)NCC(=O)NC(C(C)C)C(=O)NC(CC(C)C)C(=O)NC(C)C(=O)NC(CCC(=O)N)C(=O)NC(CC(C)C)C(=O)N5CCCC5C(=O)NCC(=O)O
SMILES (Isomeric) CC[C@H](C)[C@H]1C(=O)N[C@@H](CCC(=O)NCC(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N1)CCCN=C(N)N)CC(=O)O)C(=O)N[C@@H](CC4=CC=CC=C4)C(=O)NCC(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(=O)N)C(=O)N[C@@H](CC(C)C)C(=O)N5CCC[C@H]5C(=O)NCC(=O)O
InChI InChI=1S/C78H121N21O22/c1-10-43(8)64-75(119)91-48(25-27-57(101)83-38-60(104)97-29-17-23-55(97)77(121)99-31-16-22-54(99)72(116)85-36-58(102)88-51(35-61(105)106)71(115)90-46(69(113)96-64)20-14-28-82-78(80)81)67(111)92-50(34-45-18-12-11-13-19-45)66(110)84-37-59(103)95-63(42(6)7)74(118)93-49(32-40(2)3)70(114)87-44(9)65(109)89-47(24-26-56(79)100)68(112)94-52(33-41(4)5)76(120)98-30-15-21-53(98)73(117)86-39-62(107)108/h11-13,18-19,40-44,46-55,63-64H,10,14-17,20-39H2,1-9H3,(H2,79,100)(H,83,101)(H,84,110)(H,85,116)(H,86,117)(H,87,114)(H,88,102)(H,89,109)(H,90,115)(H,91,119)(H,92,111)(H,93,118)(H,94,112)(H,95,103)(H,96,113)(H,105,106)(H,107,108)(H4,80,81,82)/t43-,44-,46-,47-,48-,49-,50-,51-,52-,53-,54-,55-,63-,64-/m0/s1
InChI Key FUHIJKMLJFMUPU-HYFOAOAQSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C78H121N21O22
Molecular Weight 1704.90 g/mol
Exact Mass 1703.89950457 g/mol
Topological Polar Surface Area (TPSA) 650.00 Ų
XlogP -2.20

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Subterisin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 100.00% 98.95%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 99.62% 97.64%
CHEMBL3837 P07711 Cathepsin L 99.56% 96.61%
CHEMBL221 P23219 Cyclooxygenase-1 99.44% 90.17%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.26% 96.09%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 99.03% 98.33%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 98.97% 82.38%
CHEMBL4588 P22894 Matrix metalloproteinase 8 98.96% 94.66%
CHEMBL236 P41143 Delta opioid receptor 98.92% 99.35%
CHEMBL220 P22303 Acetylcholinesterase 98.88% 94.45%
CHEMBL1801 P00747 Plasminogen 98.78% 92.44%
CHEMBL4777 P25929 Neuropeptide Y receptor type 1 98.64% 96.67%
CHEMBL4018 P49146 Neuropeptide Y receptor type 2 97.83% 98.94%
CHEMBL230 P35354 Cyclooxygenase-2 97.71% 89.63%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 97.49% 82.69%
CHEMBL4979 P13866 Sodium/glucose cotransporter 1 97.12% 98.24%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 96.72% 97.14%
CHEMBL2514 O95665 Neurotensin receptor 2 96.64% 100.00%
CHEMBL3137262 O60341 LSD1/CoREST complex 96.46% 97.09%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 96.24% 91.11%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 96.04% 88.42%
CHEMBL1907591 P30926 Neuronal acetylcholine receptor; alpha4/beta4 95.93% 100.00%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 95.75% 94.45%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 95.70% 97.23%
CHEMBL4361 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 95.42% 95.52%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 95.32% 93.00%
CHEMBL5103 Q969S8 Histone deacetylase 10 95.06% 90.08%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 94.75% 96.47%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 94.45% 90.71%
CHEMBL333 P08253 Matrix metalloproteinase-2 93.82% 96.31%
CHEMBL4071 P08311 Cathepsin G 93.79% 94.64%
CHEMBL259 P32245 Melanocortin receptor 4 92.33% 95.38%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 92.33% 95.56%
CHEMBL3024 P53350 Serine/threonine-protein kinase PLK1 92.26% 97.43%
CHEMBL3060 Q9Y345 Glycine transporter 2 92.06% 99.17%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 91.86% 95.00%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 91.30% 93.03%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 90.45% 91.81%
CHEMBL3359 P21462 Formyl peptide receptor 1 90.43% 93.56%
CHEMBL5608 Q16288 NT-3 growth factor receptor 90.18% 95.89%
CHEMBL5701 Q9H2K8 Serine/threonine-protein kinase TAO3 90.05% 96.67%
CHEMBL2073 P07947 Tyrosine-protein kinase YES 90.00% 83.14%
CHEMBL4801 P29466 Caspase-1 89.47% 96.85%
CHEMBL255 P29275 Adenosine A2b receptor 88.60% 98.59%
CHEMBL204 P00734 Thrombin 88.40% 96.01%
CHEMBL1914 P06276 Butyrylcholinesterase 88.19% 95.00%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 87.74% 96.11%
CHEMBL4394 Q9NYA1 Sphingosine kinase 1 87.36% 96.03%
CHEMBL4227 P25090 Lipoxin A4 receptor 87.21% 100.00%
CHEMBL2535 P11166 Glucose transporter 86.57% 98.75%
CHEMBL2094135 Q96BI3 Gamma-secretase 86.49% 98.05%
CHEMBL5028 O14672 ADAM10 86.37% 97.50%
CHEMBL237 P41145 Kappa opioid receptor 86.26% 98.10%
CHEMBL5261 Q7L7X3 Serine/threonine-protein kinase TAO1 86.07% 89.33%
CHEMBL1255126 O15151 Protein Mdm4 85.94% 90.20%
CHEMBL2803 P43403 Tyrosine-protein kinase ZAP-70 85.92% 82.50%
CHEMBL3202 P48147 Prolyl endopeptidase 85.86% 90.65%
CHEMBL3310 Q96DB2 Histone deacetylase 11 85.53% 88.56%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 85.38% 96.90%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 84.51% 96.00%
CHEMBL217 P14416 Dopamine D2 receptor 84.23% 95.62%
CHEMBL4123 P30989 Neurotensin receptor 1 83.75% 96.67%
CHEMBL2095172 P14867 GABA-A receptor; alpha-1/beta-2/gamma-2 83.35% 92.67%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 83.30% 95.50%
CHEMBL1744525 P43490 Nicotinamide phosphoribosyltransferase 83.27% 96.25%
CHEMBL321 P14780 Matrix metalloproteinase 9 82.73% 92.12%
CHEMBL2443 P49862 Kallikrein 7 82.33% 94.00%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 81.10% 99.23%
CHEMBL3729 P22748 Carbonic anhydrase IV 80.81% 99.23%
CHEMBL5939 Q9NZ08 Endoplasmic reticulum aminopeptidase 1 80.07% 100.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139591211
LOTUS LTS0133051
wikiData Q105001709