Spiroindimicin B

Details

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Internal ID b1274f7f-7cc1-4839-a013-ba2acb982a1b
Taxonomy Organoheterocyclic compounds > Indoles and derivatives > Indoles
IUPAC Name methyl (3R)-4',5-dichloro-1-methylspiro[2H-indole-3,10'-8,13-diazatetracyclo[7.6.0.02,7.011,15]pentadeca-1(9),2(7),3,5,11,14-hexaene]-12'-carboxylate
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C23H17Cl2N3O2/c1-28-10-23(15-8-12(25)4-6-17(15)28)19-14(9-26-20(19)22(29)30-2)18-13-7-11(24)3-5-16(13)27-21(18)23/h3-9,26-27H,10H2,1-2H3/t23-/m1/s1
InChI Key FEZAUMRIJDPBGI-HSZRJFAPSA-N
Popularity 6 references in papers

Physical and Chemical Properties

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Molecular Formula C23H17Cl2N3O2
Molecular Weight 438.30 g/mol
Exact Mass 437.0697822 g/mol
Topological Polar Surface Area (TPSA) 61.10 Ų
XlogP 5.30

Synonyms

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methyl (3R)-4',5-dichloro-1-methylspiro[2H-indole-3,10'-8,13-diazatetracyclo[7.6.0.02,7.011,15]pentadeca-1(9),2(7),3,5,11,14-hexaene]-12'-carboxylate
Methyl (3R)-4',5-dichloro-1-methyl-1,2-dihydro-8',13'-diazaspiro(indole-3,10'-tetracyclo(7.6.0.0,.0,)pentadecane)-1'(9'),2'(7'),3',5',11',14'-hexaene-12'-carboxylic acid
Methyl (3R)-4',5-dichloro-1-methyl-1,2-dihydro-8',13'-diazaspiro[indole-3,10'-tetracyclo[7.6.0.0,.0,]pentadecane]-1'(9'),2'(7'),3',5',11',14'-hexaene-12'-carboxylic acid
methyl (3R)-4',5-dichloro-1-methylspiro(2H-indole-3,10'-8,13-diazatetracyclo(7.6.0.02,7.011,15)pentadeca-1(9),2(7),3,5,11,14-hexaene)-12'-carboxylate
RefChem:184871
CHEMBL5410584
CHEBI:209034
1380717-82-7

2D Structure

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2D Structure of Spiroindimicin B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 98.95% 94.45%
CHEMBL335 P18031 Protein-tyrosine phosphatase 1B 98.65% 95.17%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.97% 96.09%
CHEMBL4016 P42262 Glutamate receptor ionotropic, AMPA 2 95.21% 86.92%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 94.56% 91.11%
CHEMBL4208 P20618 Proteasome component C5 94.27% 90.00%
CHEMBL2581 P07339 Cathepsin D 93.41% 98.95%
CHEMBL2094127 P06493 Cyclin-dependent kinase 1/cyclin B 92.98% 96.00%
CHEMBL3492 P49721 Proteasome Macropain subunit 92.98% 90.24%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 91.99% 93.03%
CHEMBL2535 P11166 Glucose transporter 91.37% 98.75%
CHEMBL240 Q12809 HERG 91.02% 89.76%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 88.29% 94.00%
CHEMBL2095172 P14867 GABA-A receptor; alpha-1/beta-2/gamma-2 87.49% 92.67%
CHEMBL4303 P08238 Heat shock protein HSP 90-beta 87.15% 96.77%
CHEMBL213 P08588 Beta-1 adrenergic receptor 87.02% 95.56%
CHEMBL5852 Q96P65 Pyroglutamylated RFamide peptide receptor 86.64% 85.00%
CHEMBL3430907 Q96GD4 Aurora kinase B/Inner centromere protein 86.27% 97.50%
CHEMBL5608 Q16288 NT-3 growth factor receptor 85.80% 95.89%
CHEMBL340 P08684 Cytochrome P450 3A4 85.32% 91.19%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 84.61% 95.56%
CHEMBL2146302 O94925 Glutaminase kidney isoform, mitochondrial 83.98% 100.00%
CHEMBL4040 P28482 MAP kinase ERK2 83.86% 83.82%
CHEMBL1293289 P25440 Bromodomain-containing protein 2 83.66% 86.19%
CHEMBL217 P14416 Dopamine D2 receptor 83.32% 95.62%
CHEMBL3085 P43003 Excitatory amino acid transporter 1 81.78% 94.67%
CHEMBL3475 P05121 Plasminogen activator inhibitor-1 81.22% 83.00%
CHEMBL5028 O14672 ADAM10 81.02% 97.50%
CHEMBL1293249 Q13887 Kruppel-like factor 5 80.45% 86.33%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 80.29% 100.00%
CHEMBL2378 P30307 Dual specificity phosphatase Cdc25C 80.16% 96.67%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 60166298
LOTUS LTS0122352
wikiData Q104994279