L-Tryptophan, L-cysteinyl-L-leucylglycyl-L-isoleucylglycyl-L-seryl-L-cysteinyl-L-asparaginyl-L-alpha-aspartyl-L-phenylalanyl-L-alanylglycyl-L-cysteinylglycyl-L-tyrosyl-L-alanyl-L-isoleucyl-L-valyl-L-cysteinyl-L-phenylalanyl-, cyclic (9-1)-peptide, cyclic (1-13),(7-19)-bis(disulfide

Details

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Internal ID f1af7452-8a49-4473-9874-15e38b0080db
Taxonomy Organic Polymers > Polypeptides
IUPAC Name (2S)-2-[[(2S)-2-[[(1S,4S,7S,13R,19S,22S,25S,28S,31R,36R,39S,45S,51S,54R,60S)-60-(2-amino-2-oxoethyl)-4-benzyl-25,45-bis[(2S)-butan-2-yl]-39-(hydroxymethyl)-19-[(4-hydroxyphenyl)methyl]-7,22-dimethyl-51-(2-methylpropyl)-2,5,8,11,14,17,20,23,26,29,38,41,44,47,50,53,56,59,62-nonadecaoxo-28-propan-2-yl-33,34,64,65-tetrathia-3,6,9,12,15,18,21,24,27,30,37,40,43,46,49,52,55,58,61-nonadecazatricyclo[34.21.5.413,54]hexahexacontane-31-carbonyl]amino]-3-phenylpropanoyl]amino]-3-(1H-indol-3-yl)propanoic acid
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C98H133N23O26S4/c1-11-50(7)80-95(143)104-41-76(127)108-68(43-122)91(139)117-71-46-150-151-47-72(94(142)113-64(33-55-23-17-14-18-24-55)88(136)116-67(98(146)147)35-57-38-100-60-26-20-19-25-59(57)60)118-96(144)79(49(5)6)120-97(145)81(51(8)12-2)121-83(131)53(10)106-86(134)62(34-56-27-29-58(123)30-28-56)107-75(126)40-103-85(133)69-44-148-149-45-70(92(140)111-61(31-48(3)4)84(132)102-42-78(129)119-80)109-74(125)37-66(115-89(137)65(36-73(99)124)114-93(71)141)90(138)112-63(32-54-21-15-13-16-22-54)87(135)105-52(9)82(130)101-39-77(128)110-69/h13-30,38,48-53,61-72,79-81,100,122-123H,11-12,31-37,39-47H2,1-10H3,(H2,99,124)(H,101,130)(H,102,132)(H,103,133)(H,104,143)(H,105,135)(H,106,134)(H,107,126)(H,108,127)(H,109,125)(H,110,128)(H,111,140)(H,112,138)(H,113,142)(H,114,141)(H,115,137)(H,116,136)(H,117,139)(H,118,144)(H,119,129)(H,120,145)(H,121,131)(H,146,147)/t50-,51-,52-,53-,61-,62-,63-,64-,65-,66-,67-,68-,69-,70-,71-,72-,79-,80-,81-/m0/s1
InChI Key HQDWMGCEUREUTK-FYOZFPLDSA-N
Popularity 6 references in papers

Physical and Chemical Properties

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Molecular Formula C98H133N23O26S4
Molecular Weight 2177.50 g/mol
Exact Mass 2176.8708510 g/mol
Topological Polar Surface Area (TPSA) 849.00 Ų
XlogP 0.70

Synonyms

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BMY 29303
164802-69-1
L-Tryptophan, L-cysteinyl-L-leucylglycyl-L-isoleucylglycyl-L-seryl-L-cysteinyl-L-asparaginyl-L-alpha-aspartyl-L-phenylalanyl-L-alanylglycyl-L-cysteinylglycyl-L-tyrosyl-L-alanyl-L-isoleucyl-L-valyl-L-cysteinyl-L-phenylalanyl-, cyclic (9-1)-peptide, cyclic (1-13),(7-19)-bis(disulfide
WFCVIAYGCGAFDNCSGIGLC
BMY-29303
(2S)-2-[[(2S)-2-[[(2-amino-2-oxo-ethyl)-benzyl-(hydroxymethyl)-[(4-hydroxyphenyl)methyl]-isobutyl-isopropyl-dimethyl-bis[(1S)-1-methylpropyl]-nonadecaoxo-[?]carbonyl]amino]-3-phenyl-propanoyl]amino]-3-(1H-indol-3-yl)propanoic acid

2D Structure

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2D Structure of L-Tryptophan, L-cysteinyl-L-leucylglycyl-L-isoleucylglycyl-L-seryl-L-cysteinyl-L-asparaginyl-L-alpha-aspartyl-L-phenylalanyl-L-alanylglycyl-L-cysteinylglycyl-L-tyrosyl-L-alanyl-L-isoleucyl-L-valyl-L-cysteinyl-L-phenylalanyl-, cyclic (9-1)-peptide, cyclic (1-13),(7-19)-bis(disulfide

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.97% 98.95%
CHEMBL2288 Q13526 Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 99.70% 91.71%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.66% 91.11%
CHEMBL4040 P28482 MAP kinase ERK2 99.53% 83.82%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 99.41% 93.10%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 99.31% 97.64%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 98.70% 97.23%
CHEMBL3837 P07711 Cathepsin L 98.56% 96.61%
CHEMBL1255126 O15151 Protein Mdm4 98.29% 90.20%
CHEMBL5103 Q969S8 Histone deacetylase 10 98.20% 90.08%
CHEMBL3310 Q96DB2 Histone deacetylase 11 98.20% 88.56%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.18% 96.09%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 97.21% 95.56%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 97.10% 97.14%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 95.56% 95.50%
CHEMBL5896 O75164 Lysine-specific demethylase 4A 95.37% 99.09%
CHEMBL6175 Q9H3R0 Lysine-specific demethylase 4C 95.36% 96.69%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 95.19% 94.45%
CHEMBL2535 P11166 Glucose transporter 94.76% 98.75%
CHEMBL220 P22303 Acetylcholinesterase 94.67% 94.45%
CHEMBL4071 P08311 Cathepsin G 94.35% 94.64%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 93.95% 91.81%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 93.88% 96.90%
CHEMBL3830 Q2M2I8 Adaptor-associated kinase 92.65% 83.10%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 92.54% 96.11%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 91.54% 95.00%
CHEMBL4462 Q8IXJ6 NAD-dependent deacetylase sirtuin 2 91.30% 90.24%
CHEMBL2072 P35499 Sodium channel protein type IV alpha subunit 90.60% 92.32%
CHEMBL3137262 O60341 LSD1/CoREST complex 89.99% 97.09%
CHEMBL3060 Q9Y345 Glycine transporter 2 88.73% 99.17%
CHEMBL236 P41143 Delta opioid receptor 88.63% 99.35%
CHEMBL5608 Q16288 NT-3 growth factor receptor 88.39% 95.89%
CHEMBL2094135 Q96BI3 Gamma-secretase 88.25% 98.05%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 88.11% 88.42%
CHEMBL2821 P00748 Coagulation factor XII 88.10% 96.21%
CHEMBL226 P30542 Adenosine A1 receptor 86.73% 95.93%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 86.00% 95.50%
CHEMBL1806 P11388 DNA topoisomerase II alpha 85.79% 89.00%
CHEMBL1801 P00747 Plasminogen 85.28% 92.44%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 85.24% 99.15%
CHEMBL5939 Q9NZ08 Endoplasmic reticulum aminopeptidase 1 84.84% 100.00%
CHEMBL3476 O15111 Inhibitor of nuclear factor kappa B kinase alpha subunit 84.44% 95.83%
CHEMBL1937 Q92769 Histone deacetylase 2 84.34% 94.75%
CHEMBL221 P23219 Cyclooxygenase-1 83.65% 90.17%
CHEMBL1293287 P14735 Insulin-degrading enzyme 83.28% 88.10%
CHEMBL3359 P21462 Formyl peptide receptor 1 83.24% 93.56%
CHEMBL2035 P08912 Muscarinic acetylcholine receptor M5 83.13% 94.62%
CHEMBL340 P08684 Cytochrome P450 3A4 82.83% 91.19%
CHEMBL1907591 P30926 Neuronal acetylcholine receptor; alpha4/beta4 82.28% 100.00%
CHEMBL1949 P62937 Cyclophilin A 82.17% 98.57%
CHEMBL2095172 P14867 GABA-A receptor; alpha-1/beta-2/gamma-2 82.07% 92.67%
CHEMBL2514 O95665 Neurotensin receptor 2 81.82% 100.00%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 81.76% 99.23%
CHEMBL2563 Q9UQL6 Histone deacetylase 5 81.35% 89.67%
CHEMBL4227 P25090 Lipoxin A4 receptor 81.19% 100.00%
CHEMBL4101 P17612 cAMP-dependent protein kinase alpha-catalytic subunit 80.98% 82.86%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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Cross-Links

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PubChem 16130326
LOTUS LTS0135470
wikiData Q105032206