Roquefortine D

Details

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Internal ID 7f99e791-6f2b-4581-ba72-fff31c73201c
Taxonomy Organoheterocyclic compounds > Indoles and derivatives > Pyrroloindoles
IUPAC Name 4-(1H-imidazol-5-ylmethyl)-9-(2-methylbut-3-en-2-yl)-2,5,16-triazatetracyclo[7.7.0.02,7.010,15]hexadeca-10,12,14-triene-3,6-dione
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C22H25N5O2/c1-4-21(2,3)22-10-17-18(28)25-16(9-13-11-23-12-24-13)19(29)27(17)20(22)26-15-8-6-5-7-14(15)22/h4-8,11-12,16-17,20,26H,1,9-10H2,2-3H3,(H,23,24)(H,25,28)
InChI Key IQVNREJWRXOHEO-UHFFFAOYSA-N
Popularity 7 references in papers

Physical and Chemical Properties

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Molecular Formula C22H25N5O2
Molecular Weight 391.50 g/mol
Exact Mass 391.20082506 g/mol
Topological Polar Surface Area (TPSA) 90.10 Ų
XlogP 2.90

Synonyms

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MEGxm0_000337
ACon1_001592
DTXSID40894026
NCGC00180346-02
C22163
BRD-A75055874-001-01-2
(3S,5aS,10bR,11aS)-3-(1H-Imidazol-5-ylmethyl)-10b-(2-methyl-3-buten-2-yl)-6,10b,11,11a-tetrahydro-2H-pyrazino[1',2':1,5]pyrrolo[2,3-b]indole-1,4(3H,5aH)-dione

2D Structure

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2D Structure of Roquefortine D

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.12% 96.09%
CHEMBL1937 Q92769 Histone deacetylase 2 96.35% 94.75%
CHEMBL3524 P56524 Histone deacetylase 4 95.55% 92.97%
CHEMBL2581 P07339 Cathepsin D 94.09% 98.95%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 92.50% 97.64%
CHEMBL5697 Q9GZT9 Egl nine homolog 1 92.02% 93.40%
CHEMBL253 P34972 Cannabinoid CB2 receptor 91.68% 97.25%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 90.54% 85.14%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 90.53% 95.56%
CHEMBL3310 Q96DB2 Histone deacetylase 11 90.46% 88.56%
CHEMBL1293249 Q13887 Kruppel-like factor 5 90.19% 86.33%
CHEMBL5103 Q969S8 Histone deacetylase 10 89.61% 90.08%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 89.50% 91.11%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 89.49% 93.03%
CHEMBL2095226 P05556 Integrin alpha-5/beta-1 88.46% 96.39%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 84.13% 99.23%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 84.07% 94.45%
CHEMBL3038469 P24941 CDK2/Cyclin A 83.88% 91.38%
CHEMBL1902 P62942 FK506-binding protein 1A 83.86% 97.05%
CHEMBL255 P29275 Adenosine A2b receptor 82.90% 98.59%
CHEMBL2035 P08912 Muscarinic acetylcholine receptor M5 81.90% 94.62%
CHEMBL3137262 O60341 LSD1/CoREST complex 81.01% 97.09%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 80.30% 97.33%
CHEMBL3869 P50281 Matrix metalloproteinase 14 80.25% 93.10%
CHEMBL5028 O14672 ADAM10 80.08% 97.50%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 15386782
LOTUS LTS0133401
wikiData Q77493973