Pumiliotoxin A

Details

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Internal ID 98482b33-ca0e-436c-9b14-e4ccf52eb6da
Taxonomy Alkaloids and derivatives > Pumiliotoxins, homopumiliotoxins, and allopumiliotoxins
IUPAC Name (6Z,8S,8aS)-6-[(E,2R,6S)-6-hydroxy-2,5-dimethyloct-4-enylidene]-8-methyl-1,2,3,5,7,8a-hexahydroindolizin-8-ol
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C19H33NO2/c1-5-17(21)15(3)9-8-14(2)11-16-12-19(4,22)18-7-6-10-20(18)13-16/h9,11,14,17-18,21-22H,5-8,10,12-13H2,1-4H3/b15-9+,16-11-/t14-,17+,18+,19+/m1/s1
InChI Key CUBVJLHFQCEJGM-SZIIBLSRSA-N
Popularity 15 references in papers

Physical and Chemical Properties

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Molecular Formula C19H33NO2
Molecular Weight 307.50 g/mol
Exact Mass 307.251129295 g/mol
Topological Polar Surface Area (TPSA) 43.70 Ų
XlogP 2.80

Synonyms

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CHEMBL145948
SCHEMBL10726788
DTXSID80897238
C20033
(6Z,8S,8aS)-6-[(E,2R,6S)-6-hydroxy-2,5-dimethyloct-4-enylidene]-8-methyl-1,2,3,5,7,8a-hexahydroindolizin-8-ol

2D Structure

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2D Structure of Pumiliotoxin A

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL240 Q12809 HERG 99.26% 89.76%
CHEMBL253 P34972 Cannabinoid CB2 receptor 98.68% 97.25%
CHEMBL2581 P07339 Cathepsin D 96.61% 98.95%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 95.99% 94.45%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 95.50% 96.09%
CHEMBL5608 Q16288 NT-3 growth factor receptor 92.06% 95.89%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 90.77% 91.11%
CHEMBL5469 Q14289 Protein tyrosine kinase 2 beta 86.64% 91.03%
CHEMBL4208 P20618 Proteasome component C5 84.54% 90.00%
CHEMBL3359 P21462 Formyl peptide receptor 1 83.63% 93.56%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 83.58% 95.56%
CHEMBL4227 P25090 Lipoxin A4 receptor 82.94% 100.00%
CHEMBL4005 P42336 PI3-kinase p110-alpha subunit 82.49% 97.47%
CHEMBL5203 P33316 dUTP pyrophosphatase 82.42% 99.18%
CHEMBL3430907 Q96GD4 Aurora kinase B/Inner centromere protein 82.33% 97.50%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 82.25% 98.33%
CHEMBL3476 O15111 Inhibitor of nuclear factor kappa B kinase alpha subunit 81.30% 95.83%
CHEMBL3137262 O60341 LSD1/CoREST complex 80.98% 97.09%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 80.62% 100.00%
CHEMBL1994 P08235 Mineralocorticoid receptor 80.17% 100.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

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PubChem 10979740
LOTUS LTS0216590
wikiData Q104396334