Pompanopeptin A

Details

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Internal ID 6def4851-1499-4c6c-a61a-bea413563931
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name (2S)-N-[(2S,5S,8S,11R,12S,15S,18S,21R)-5-[(3-bromo-4-methoxyphenyl)methyl]-2-[(2S)-butan-2-yl]-15-[3-(diaminomethylideneamino)propyl]-21-hydroxy-4,11-dimethyl-3,6,9,13,16,22-hexaoxo-8-propan-2-yl-10-oxa-1,4,7,14,17-pentazabicyclo[16.3.1]docosan-12-yl]-2-(butanoylamino)-4-methylsulfinylbutanamide
SMILES (Canonical) CCCC(=O)NC(CCS(=O)C)C(=O)NC1C(OC(=O)C(NC(=O)C(N(C(=O)C(N2C(CCC(C2=O)NC(=O)C(NC1=O)CCCN=C(N)N)O)C(C)CC)C)CC3=CC(=C(C=C3)OC)Br)C(C)C)C
SMILES (Isomeric) CCCC(=O)N[C@@H](CCS(=O)C)C(=O)N[C@H]1[C@H](OC(=O)[C@@H](NC(=O)[C@@H](N(C(=O)[C@@H](N2[C@@H](CC[C@@H](C2=O)NC(=O)[C@@H](NC1=O)CCCN=C(N)N)O)[C@@H](C)CC)C)CC3=CC(=C(C=C3)OC)Br)C(C)C)C
InChI InChI=1S/C46H73BrN10O12S/c1-10-13-34(58)51-30(19-21-70(9)67)40(61)55-37-26(6)69-45(66)36(24(3)4)54-41(62)32(23-27-15-17-33(68-8)28(47)22-27)56(7)44(65)38(25(5)11-2)57-35(59)18-16-31(43(57)64)53-39(60)29(52-42(37)63)14-12-20-50-46(48)49/h15,17,22,24-26,29-32,35-38,59H,10-14,16,18-21,23H2,1-9H3,(H,51,58)(H,52,63)(H,53,60)(H,54,62)(H,55,61)(H4,48,49,50)/t25-,26+,29-,30-,31-,32-,35+,36-,37-,38-,70?/m0/s1
InChI Key KHHPHRPDQUMGBB-LLNFQSNNSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C46H73BrN10O12S
Molecular Weight 1070.10 g/mol
Exact Mass 1068.43135 g/mol
Topological Polar Surface Area (TPSA) 343.00 Ų
XlogP 1.40

Synonyms

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DTXSID901046220

2D Structure

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2D Structure of Pompanopeptin A

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.75% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.38% 96.09%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 99.25% 94.45%
CHEMBL3060 Q9Y345 Glycine transporter 2 98.59% 99.17%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.20% 91.11%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 96.21% 93.00%
CHEMBL4040 P28482 MAP kinase ERK2 96.10% 83.82%
CHEMBL5608 Q16288 NT-3 growth factor receptor 95.72% 95.89%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 95.19% 92.88%
CHEMBL4588 P22894 Matrix metalloproteinase 8 94.99% 94.66%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 94.31% 95.56%
CHEMBL3137262 O60341 LSD1/CoREST complex 93.62% 97.09%
CHEMBL3837 P07711 Cathepsin L 93.39% 96.61%
CHEMBL261 P00915 Carbonic anhydrase I 93.05% 96.76%
CHEMBL2413 P32246 C-C chemokine receptor type 1 91.93% 89.50%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 91.68% 90.71%
CHEMBL5103 Q969S8 Histone deacetylase 10 91.56% 90.08%
CHEMBL255 P29275 Adenosine A2b receptor 90.98% 98.59%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 90.62% 97.14%
CHEMBL1949 P62937 Cyclophilin A 90.46% 98.57%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 90.13% 96.38%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 89.81% 96.00%
CHEMBL4072 P07858 Cathepsin B 89.52% 93.67%
CHEMBL2096618 P11274 Bcr/Abl fusion protein 89.43% 85.83%
CHEMBL2535 P11166 Glucose transporter 88.98% 98.75%
CHEMBL1806 P11388 DNA topoisomerase II alpha 88.50% 89.00%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 87.39% 96.90%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 86.78% 82.38%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 86.76% 93.03%
CHEMBL333 P08253 Matrix metalloproteinase-2 86.72% 96.31%
CHEMBL259 P32245 Melanocortin receptor 4 86.54% 95.38%
CHEMBL1255126 O15151 Protein Mdm4 86.34% 90.20%
CHEMBL1293249 Q13887 Kruppel-like factor 5 86.07% 86.33%
CHEMBL4644 P41968 Melanocortin receptor 3 86.07% 99.52%
CHEMBL2094135 Q96BI3 Gamma-secretase 85.01% 98.05%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 84.99% 100.00%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 84.77% 95.89%
CHEMBL253 P34972 Cannabinoid CB2 receptor 83.82% 97.25%
CHEMBL340 P08684 Cytochrome P450 3A4 83.61% 91.19%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 82.92% 97.64%
CHEMBL3359 P21462 Formyl peptide receptor 1 82.86% 93.56%
CHEMBL283 P08254 Matrix metalloproteinase 3 82.52% 97.29%
CHEMBL4227 P25090 Lipoxin A4 receptor 82.44% 100.00%
CHEMBL2000 P03952 Plasma kallikrein 81.97% 93.92%
CHEMBL225 P28335 Serotonin 2c (5-HT2c) receptor 81.65% 89.62%
CHEMBL2443 P49862 Kallikrein 7 81.53% 94.00%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 81.51% 97.23%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 81.22% 94.00%
CHEMBL4769 O95749 Geranylgeranyl pyrophosphate synthetase 80.22% 92.08%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 24862182
LOTUS LTS0213521
wikiData Q104203225