Pneumocandin B2

Details

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Internal ID 88538d2d-b78a-419e-a14a-1a9cb2723fb9
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Cyclic peptides
IUPAC Name (10R,12S)-N-[(3S,6S,9S,11R,15S,18R,24S,25S)-3-[(1R)-3-amino-1-hydroxy-3-oxopropyl]-6-[(1S,2S)-1,2-dihydroxy-2-(4-hydroxyphenyl)ethyl]-11,25-dihydroxy-15-[(1R)-1-hydroxyethyl]-2,5,8,14,17,23-hexaoxo-1,4,7,13,16,22-hexazatricyclo[22.3.0.09,13]heptacosan-18-yl]-10,12-dimethyltetradecanamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C50H80N8O15/c1-5-27(2)23-28(3)13-10-8-6-7-9-11-15-38(65)53-33-14-12-21-52-48(71)42-35(62)20-22-57(42)50(73)40(36(63)25-37(51)64)55-47(70)41(44(67)43(66)30-16-18-31(60)19-17-30)56-46(69)34-24-32(61)26-58(34)49(72)39(29(4)59)54-45(33)68/h16-19,27-29,32-36,39-44,59-63,66-67H,5-15,20-26H2,1-4H3,(H2,51,64)(H,52,71)(H,53,65)(H,54,68)(H,55,70)(H,56,69)/t27-,28+,29+,32+,33+,34-,35-,36+,39-,40-,41-,42-,43-,44-/m0/s1
InChI Key CAUDURDUCQQHDE-GHMALVTLSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C50H80N8O15
Molecular Weight 1033.20 g/mol
Exact Mass 1032.57431387 g/mol
Topological Polar Surface Area (TPSA) 371.00 Ų
XlogP 2.00

Synonyms

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(10R,12S)-N-[(3S,6S,9S,11R,15S,18R,24S,25S)-3-[(1R)-3-amino-1-hydroxy-3-oxopropyl]-6-[(1S,2S)-1,2-dihydroxy-2-(4-hydroxyphenyl)ethyl]-11,25-dihydroxy-15-[(1R)-1-hydroxyethyl]-2,5,8,14,17,23-hexaoxo-1,4,7,13,16,22-hexazatricyclo[22.3.0.09,13]heptacosan-18-yl]-10,12-dimethyltetradecanamide
(10R,12S)-N-((3S,6S,9S,11R,15S,18R,24S,25S)-3-((1R)-3-amino-1-hydroxy-3-oxopropyl)-6-((1S,2S)-1,2-dihydroxy-2-(4-hydroxyphenyl)ethyl)-11,25-dihydroxy-15-((1R)-1-hydroxyethyl)-2,5,8,14,17,23-hexaoxo-1,4,7,13,16,22-hexazatricyclo(22.3.0.09,13)heptacosan-18-yl)-10,12-dimethyltetradecanamide
(10R,12S)-N-((3S,6S,9S,11R,15S,18R,24S,25S)-6-((1S,2S)-1,2-Dihydroxy-2-(4-hydroxyphenyl)ethyl)-5,8,11,17,23,25-hexahydroxy-3-((1R)-1-hydroxy-2-(C-hydroxycarbonimidoyl)ethyl)-15-((1R)-1-hydroxyethyl)-2,14-dioxo-1,4,7,13,16,22-hexaazatricyclo(22.3.0.0,)heptacosa-4,7,16,22-tetraen-18-yl)-10,12-dimethyltetradecanimidate
(10R,12S)-N-[(3S,6S,9S,11R,15S,18R,24S,25S)-6-[(1S,2S)-1,2-Dihydroxy-2-(4-hydroxyphenyl)ethyl]-5,8,11,17,23,25-hexahydroxy-3-[(1R)-1-hydroxy-2-(C-hydroxycarbonimidoyl)ethyl]-15-[(1R)-1-hydroxyethyl]-2,14-dioxo-1,4,7,13,16,22-hexaazatricyclo[22.3.0.0,]heptacosa-4,7,16,22-tetraen-18-yl]-10,12-dimethyltetradecanimidate
RefChem:174961
CHEBI:224602

2D Structure

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2D Structure of Pneumocandin B2

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.73% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.55% 96.09%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.95% 91.11%
CHEMBL3137262 O60341 LSD1/CoREST complex 97.84% 97.09%
CHEMBL2996 Q05655 Protein kinase C delta 97.59% 97.79%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 96.99% 94.45%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 96.00% 90.71%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 94.84% 95.00%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 94.43% 85.14%
CHEMBL5103 Q969S8 Histone deacetylase 10 94.41% 90.08%
CHEMBL3060 Q9Y345 Glycine transporter 2 93.11% 99.17%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 92.38% 100.00%
CHEMBL226 P30542 Adenosine A1 receptor 90.68% 95.93%
CHEMBL3359 P21462 Formyl peptide receptor 1 89.69% 93.56%
CHEMBL225 P28335 Serotonin 2c (5-HT2c) receptor 89.22% 89.62%
CHEMBL255 P29275 Adenosine A2b receptor 88.48% 98.59%
CHEMBL4588 P22894 Matrix metalloproteinase 8 87.71% 94.66%
CHEMBL268 P43235 Cathepsin K 87.08% 96.85%
CHEMBL5608 Q16288 NT-3 growth factor receptor 87.07% 95.89%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 86.34% 91.81%
CHEMBL1806 P11388 DNA topoisomerase II alpha 85.99% 89.00%
CHEMBL5469 Q14289 Protein tyrosine kinase 2 beta 85.29% 91.03%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 84.07% 96.11%
CHEMBL2514 O95665 Neurotensin receptor 2 84.05% 100.00%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 84.04% 82.69%
CHEMBL299 P17252 Protein kinase C alpha 83.86% 98.03%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 83.73% 99.23%
CHEMBL2781 P19634 Sodium/hydrogen exchanger 1 83.47% 90.24%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 83.29% 97.64%
CHEMBL3830 Q2M2I8 Adaptor-associated kinase 83.26% 83.10%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 83.20% 94.33%
CHEMBL204 P00734 Thrombin 83.17% 96.01%
CHEMBL218 P21554 Cannabinoid CB1 receptor 82.35% 96.61%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 81.66% 95.56%
CHEMBL5255 O00206 Toll-like receptor 4 81.61% 92.50%
CHEMBL1907591 P30926 Neuronal acetylcholine receptor; alpha4/beta4 81.33% 100.00%
CHEMBL1744525 P43490 Nicotinamide phosphoribosyltransferase 81.29% 96.25%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 81.27% 93.00%
CHEMBL4227 P25090 Lipoxin A4 receptor 80.48% 100.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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Cross-Links

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PubChem 139586570
LOTUS LTS0131869
wikiData Q77509208