Phakellistatin 3

Details

Top
Internal ID bb14d073-d2b6-47b4-9ba2-88e7d1b75e06
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Oligopeptides
IUPAC Name (1S,7S,10S,19S,22S,25S,28R,36S)-10-benzyl-36-hydroxy-22-[(1R)-1-hydroxyethyl]-25-(2-methylpropyl)-3,9,12,15,21,24,27,29-octazahexacyclo[25.10.0.03,7.015,19.028,36.030,35]heptatriaconta-30,32,34-triene-2,8,11,14,20,23,26-heptone
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C42H54N8O9/c1-23(2)19-29-39(57)50-32(21-42(59)26-13-7-8-14-27(26)46-41(42)50)40(58)49-18-10-16-31(49)36(54)44-28(20-25-11-5-4-6-12-25)35(53)43-22-33(52)48-17-9-15-30(48)37(55)47-34(24(3)51)38(56)45-29/h4-8,11-14,23-24,28-32,34,41,46,51,59H,9-10,15-22H2,1-3H3,(H,43,53)(H,44,54)(H,45,56)(H,47,55)/t24-,28+,29+,30+,31+,32+,34+,41-,42+/m1/s1
InChI Key KFCKDHAGPVEUCT-RPELCPBOSA-N
Popularity 4 references in papers

Physical and Chemical Properties

Top
Molecular Formula C42H54N8O9
Molecular Weight 814.90 g/mol
Exact Mass 814.40137533 g/mol
Topological Polar Surface Area (TPSA) 230.00 Ų
XlogP 1.80

Synonyms

Top
(1S,7S,10S,19S,22S,25S,28R,36S)-10-Benzyl-36-hydroxy-22-[(1R)-1-hydroxyethyl]-25-(2-methylpropyl)-3,9,12,15,21,24,27,29-octazahexacyclo[25.10.0.03,7.015,19.028,36.030,35]heptatriaconta-30,32,34-triene-2,8,11,14,20,23,26-heptone

2D Structure

Top
2D Structure of Phakellistatin 3

3D Structure

Top

ADMET Properties (via admetSAR 2)

Top
Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

Top

Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.78% 98.95%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 99.55% 85.14%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.75% 96.09%
CHEMBL3524 P56524 Histone deacetylase 4 98.58% 92.97%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 95.36% 97.64%
CHEMBL333 P08253 Matrix metalloproteinase-2 95.19% 96.31%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 94.99% 91.11%
CHEMBL5103 Q969S8 Histone deacetylase 10 94.48% 90.08%
CHEMBL1902 P62942 FK506-binding protein 1A 94.07% 97.05%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 92.24% 93.00%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 91.94% 95.56%
CHEMBL5608 Q16288 NT-3 growth factor receptor 91.78% 95.89%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 91.22% 82.38%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 89.76% 94.45%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 88.66% 97.14%
CHEMBL1293249 Q13887 Kruppel-like factor 5 88.51% 86.33%
CHEMBL221 P23219 Cyclooxygenase-1 88.49% 90.17%
CHEMBL4208 P20618 Proteasome component C5 88.34% 90.00%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 88.11% 93.03%
CHEMBL1937 Q92769 Histone deacetylase 2 87.74% 94.75%
CHEMBL3137262 O60341 LSD1/CoREST complex 87.25% 97.09%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 87.08% 90.93%
CHEMBL4588 P22894 Matrix metalloproteinase 8 86.85% 94.66%
CHEMBL4071 P08311 Cathepsin G 86.09% 94.64%
CHEMBL321 P14780 Matrix metalloproteinase 9 85.96% 92.12%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 85.74% 95.89%
CHEMBL3310 Q96DB2 Histone deacetylase 11 85.26% 88.56%
CHEMBL228 P31645 Serotonin transporter 85.04% 95.51%
CHEMBL5203 P33316 dUTP pyrophosphatase 83.12% 99.18%
CHEMBL4447 Q9Y337 Kallikrein 5 82.24% 87.50%
CHEMBL253 P34972 Cannabinoid CB2 receptor 80.12% 97.25%

Plants that contains it

Top
Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

Top
PubChem 10485551
LOTUS LTS0095699
wikiData Q105140306