Palosine, 17-demethoxy-

Details

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Internal ID 45e66c86-b35f-4cb9-add5-bae7275f1fdd
Taxonomy Alkaloids and derivatives > Aspidospermatan-type alkaloids
IUPAC Name 1-(12-ethyl-8,16-diazapentacyclo[10.6.1.01,9.02,7.016,19]nonadeca-2,4,6-trien-8-yl)propan-1-one
SMILES (Canonical) CCC(=O)N1C2CCC3(CCCN4C3C2(CC4)C5=CC=CC=C51)CC
SMILES (Isomeric) CCC(=O)N1C2CCC3(CCCN4C3C2(CC4)C5=CC=CC=C51)CC
InChI InChI=1S/C22H30N2O/c1-3-19(25)24-17-9-6-5-8-16(17)22-13-15-23-14-7-11-21(4-2,20(22)23)12-10-18(22)24/h5-6,8-9,18,20H,3-4,7,10-15H2,1-2H3
InChI Key ZVJUOTFDVKNXIK-UHFFFAOYSA-N
Popularity 0 references in papers

Physical and Chemical Properties

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Molecular Formula C22H30N2O
Molecular Weight 338.50 g/mol
Exact Mass 338.235813585 g/mol
Topological Polar Surface Area (TPSA) 23.60 Ų
XlogP 3.90

Synonyms

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1-Propionylaspidospermidine #
ZVJUOTFDVKNXIK-UHFFFAOYSA-N
Aspidospermidine, 1-(1-oxopropyl)-

2D Structure

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2D Structure of Palosine, 17-demethoxy-

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.55% 96.09%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 91.94% 95.56%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 90.83% 91.11%
CHEMBL221 P23219 Cyclooxygenase-1 87.78% 90.17%
CHEMBL3137262 O60341 LSD1/CoREST complex 86.24% 97.09%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 85.98% 82.69%
CHEMBL1293249 Q13887 Kruppel-like factor 5 85.44% 86.33%
CHEMBL2581 P07339 Cathepsin D 85.21% 98.95%
CHEMBL2781 P19634 Sodium/hydrogen exchanger 1 84.44% 90.24%
CHEMBL5028 O14672 ADAM10 84.26% 97.50%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 84.21% 93.03%
CHEMBL4208 P20618 Proteasome component C5 83.56% 90.00%
CHEMBL5608 Q16288 NT-3 growth factor receptor 80.80% 95.89%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 80.77% 90.71%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 80.35% 94.45%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Aspidosperma discolor

Cross-Links

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PubChem 579957
LOTUS LTS0111986
wikiData Q105384345