Oscillapeptin J

Details

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Internal ID 77222f6a-6d32-4daa-9776-9db446175a14
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name [(2R)-3-[[(2S)-1-[[(2S,5S,8S,11R,12S,15S,18S,21R)-8-[(2R)-butan-2-yl]-15-[3-(diaminomethylideneamino)propyl]-21-hydroxy-2-[(1R)-1-hydroxyethyl]-5-[(4-hydroxyphenyl)methyl]-4,11-dimethyl-3,6,9,13,16,22-hexaoxo-10-oxa-1,4,7,14,17-pentazabicyclo[16.3.1]docosan-12-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-2-hydroxy-3-oxopropyl] hydrogen sulfate
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C47H68N10O18S/c1-6-23(2)36-46(70)75-25(4)37(55-40(64)32(20-26-9-13-28(59)14-10-26)53-42(66)34(61)22-74-76(71,72)73)43(67)51-30(8-7-19-50-47(48)49)39(63)52-31-17-18-35(62)57(44(31)68)38(24(3)58)45(69)56(5)33(41(65)54-36)21-27-11-15-29(60)16-12-27/h9-16,23-25,30-38,58-62H,6-8,17-22H2,1-5H3,(H,51,67)(H,52,63)(H,53,66)(H,54,65)(H,55,64)(H4,48,49,50)(H,71,72,73)/t23-,24-,25-,30+,31+,32+,33+,34-,35-,36+,37+,38+/m1/s1
InChI Key TYSLVBJOPFOBFU-KHIPEBSYSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C47H68N10O18S
Molecular Weight 1093.20 g/mol
Exact Mass 1092.44337653 g/mol
Topological Polar Surface Area (TPSA) 450.00 Ų
XlogP -1.00

Synonyms

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SCHEMBL16431289

2D Structure

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2D Structure of Oscillapeptin J

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.91% 98.95%
CHEMBL3837 P07711 Cathepsin L 99.81% 96.61%
CHEMBL4040 P28482 MAP kinase ERK2 99.72% 83.82%
CHEMBL4072 P07858 Cathepsin B 99.67% 93.67%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.29% 96.09%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 99.15% 96.38%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 98.58% 94.45%
CHEMBL226 P30542 Adenosine A1 receptor 97.24% 95.93%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.62% 95.56%
CHEMBL3137262 O60341 LSD1/CoREST complex 94.85% 97.09%
CHEMBL255 P29275 Adenosine A2b receptor 94.33% 98.59%
CHEMBL4588 P22894 Matrix metalloproteinase 8 94.31% 94.66%
CHEMBL2094135 Q96BI3 Gamma-secretase 94.29% 98.05%
CHEMBL3060 Q9Y345 Glycine transporter 2 94.17% 99.17%
CHEMBL5103 Q969S8 Histone deacetylase 10 94.05% 90.08%
CHEMBL4198 P98170 Inhibitor of apoptosis protein 3 94.01% 97.79%
CHEMBL5608 Q16288 NT-3 growth factor receptor 93.91% 95.89%
CHEMBL333 P08253 Matrix metalloproteinase-2 93.61% 96.31%
CHEMBL3359 P21462 Formyl peptide receptor 1 92.63% 93.56%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 92.30% 95.89%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 92.28% 97.14%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 91.46% 92.88%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 89.78% 90.71%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 89.66% 93.03%
CHEMBL259 P32245 Melanocortin receptor 4 89.65% 95.38%
CHEMBL1806 P11388 DNA topoisomerase II alpha 89.26% 89.00%
CHEMBL2514 O95665 Neurotensin receptor 2 88.91% 100.00%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 88.82% 97.64%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 88.53% 96.90%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 88.39% 91.11%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 87.93% 93.10%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 86.37% 100.00%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 86.34% 93.00%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 85.51% 97.23%
CHEMBL4835 P00338 L-lactate dehydrogenase A chain 85.46% 95.34%
CHEMBL1801 P00747 Plasminogen 84.52% 92.44%
CHEMBL4227 P25090 Lipoxin A4 receptor 83.79% 100.00%
CHEMBL4461 Q9NTG7 NAD-dependent deacetylase sirtuin 3 83.52% 94.36%
CHEMBL1949 P62937 Cyclophilin A 82.83% 98.57%
CHEMBL2000 P03952 Plasma kallikrein 81.92% 93.92%
CHEMBL2413 P32246 C-C chemokine receptor type 1 81.84% 89.50%
CHEMBL261 P00915 Carbonic anhydrase I 81.61% 96.76%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 81.51% 95.50%
CHEMBL4777 P25929 Neuropeptide Y receptor type 1 81.49% 96.67%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 81.20% 99.23%
CHEMBL301 P24941 Cyclin-dependent kinase 2 80.90% 91.23%
CHEMBL4506 Q96EB6 NAD-dependent deacetylase sirtuin 1 80.71% 88.33%
CHEMBL2179 P04062 Beta-glucocerebrosidase 80.65% 85.31%
CHEMBL2072 P35499 Sodium channel protein type IV alpha subunit 80.23% 92.32%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 80.05% 94.33%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 11768341
LOTUS LTS0065696
wikiData Q77386058