Nikkomycin X

Details

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Internal ID 213d0bc9-28d0-47d1-a104-15f2dcdf073e
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Dipeptides
IUPAC Name 2-[[2-amino-4-hydroxy-4-(5-hydroxypyridin-2-yl)-3-methylbutanoyl]amino]-2-[5-(5-formyl-2-oxo-1H-imidazol-3-yl)-3,4-dihydroxyoxolan-2-yl]acetic acid
SMILES (Canonical) CC(C(C1=NC=C(C=C1)O)O)C(C(=O)NC(C2C(C(C(O2)N3C=C(NC3=O)C=O)O)O)C(=O)O)N
SMILES (Isomeric) CC(C(C1=NC=C(C=C1)O)O)C(C(=O)NC(C2C(C(C(O2)N3C=C(NC3=O)C=O)O)O)C(=O)O)N
InChI InChI=1S/C20H25N5O10/c1-7(13(28)10-3-2-9(27)4-22-10)11(21)17(31)24-12(19(32)33)16-14(29)15(30)18(35-16)25-5-8(6-26)23-20(25)34/h2-7,11-16,18,27-30H,21H2,1H3,(H,23,34)(H,24,31)(H,32,33)
InChI Key AYXHZRVSIUJLAE-UHFFFAOYSA-N
Popularity 10 references in papers

Physical and Chemical Properties

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Molecular Formula C20H25N5O10
Molecular Weight 495.40 g/mol
Exact Mass 495.16014201 g/mol
Topological Polar Surface Area (TPSA) 245.00 Ų
XlogP -5.80

Synonyms

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Nikkomycin X
2-[[2-amino-4-hydroxy-4-(5-hydroxypyridin-2-yl)-3-methylbutanoyl]amino]-2-[5-(5-formyl-2-oxo-1H-imidazol-3-yl)-3,4-dihydroxyoxolan-2-yl]acetic acid
BRN 0873576
DTXSID10993651
beta-D-Allofuranuronic acid, 5-((2-amino-4-hydroxy-4-(5-hydroxy-2-pyridinyl)-3-methyl-1-oxobutyl)amino)-1,5-dideoxy-1-(4-formyl-2,3-dihydro-2-oxo-1H-imidazol-1-yl)-, (2S-(2R*,3R*,4R*))-
1-(5-{[2-Amino-1,4-dihydroxy-4-(5-hydroxypyridin-2-yl)-3-methylbutylidene]amino}-5-deoxyhexofuranuronosyl)-2-hydroxy-1H-imidazole-4-carbaldehyde
75044-69-8

2D Structure

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2D Structure of Nikkomycin X

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.48% 96.09%
CHEMBL2581 P07339 Cathepsin D 96.69% 98.95%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 95.78% 85.14%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.27% 95.56%
CHEMBL4040 P28482 MAP kinase ERK2 94.81% 83.82%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 90.43% 94.45%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 90.16% 93.10%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 89.45% 90.71%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 89.28% 99.23%
CHEMBL3401 O75469 Pregnane X receptor 89.14% 94.73%
CHEMBL1806 P11388 DNA topoisomerase II alpha 88.01% 89.00%
CHEMBL3060 Q9Y345 Glycine transporter 2 88.01% 99.17%
CHEMBL5608 Q16288 NT-3 growth factor receptor 87.97% 95.89%
CHEMBL3976 Q9UHL4 Dipeptidyl peptidase II 87.49% 92.29%
CHEMBL2345 P51812 Ribosomal protein S6 kinase alpha 3 86.74% 95.64%
CHEMBL4208 P20618 Proteasome component C5 84.92% 90.00%
CHEMBL220 P22303 Acetylcholinesterase 83.98% 94.45%
CHEMBL3359 P21462 Formyl peptide receptor 1 82.81% 93.56%
CHEMBL5103 Q969S8 Histone deacetylase 10 82.58% 90.08%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 81.99% 91.11%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 81.87% 99.15%
CHEMBL2535 P11166 Glucose transporter 81.78% 98.75%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 81.34% 100.00%
CHEMBL5678 P34947 G protein-coupled receptor kinase 5 80.15% 88.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 194647
LOTUS LTS0071463
wikiData Q82984368