Nikkomycin Lx

Details

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Internal ID f0b50f78-fbc5-4b3f-b220-ff08c92dcf05
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides
IUPAC Name 2-[5-(5-acetyl-2-oxo-1H-imidazol-3-yl)-3,4-dihydroxyoxolan-2-yl]-2-[(2-amino-4-hydroxy-3-methyl-4-pyridin-2-ylbutanoyl)amino]acetic acid
SMILES (Canonical) CC(C(C1=CC=CC=N1)O)C(C(=O)NC(C2C(C(C(O2)N3C=C(NC3=O)C(=O)C)O)O)C(=O)O)N
SMILES (Isomeric) CC(C(C1=CC=CC=N1)O)C(C(=O)NC(C2C(C(C(O2)N3C=C(NC3=O)C(=O)C)O)O)C(=O)O)N
InChI InChI=1S/C21H27N5O9/c1-8(14(28)10-5-3-4-6-23-10)12(22)18(31)25-13(20(32)33)17-15(29)16(30)19(35-17)26-7-11(9(2)27)24-21(26)34/h3-8,12-17,19,28-30H,22H2,1-2H3,(H,24,34)(H,25,31)(H,32,33)
InChI Key ICXJRQHWJJTKQI-UHFFFAOYSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C21H27N5O9
Molecular Weight 493.50 g/mol
Exact Mass 493.18087746 g/mol
Topological Polar Surface Area (TPSA) 225.00 Ų
XlogP -5.20

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Nikkomycin Lx

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL4040 P28482 MAP kinase ERK2 99.30% 83.82%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.20% 96.09%
CHEMBL2581 P07339 Cathepsin D 98.42% 98.95%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 97.57% 85.14%
CHEMBL3401 O75469 Pregnane X receptor 91.93% 94.73%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 90.57% 95.56%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 90.03% 99.23%
CHEMBL1806 P11388 DNA topoisomerase II alpha 89.82% 89.00%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 89.01% 93.10%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 88.09% 100.00%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 86.78% 91.11%
CHEMBL5028 O14672 ADAM10 83.76% 97.50%
CHEMBL1821 P08173 Muscarinic acetylcholine receptor M4 82.92% 94.08%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 82.85% 90.71%
CHEMBL255 P29275 Adenosine A2b receptor 82.58% 98.59%
CHEMBL3359 P21462 Formyl peptide receptor 1 82.23% 93.56%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139588843
LOTUS LTS0029576
wikiData Q104168658