Ngercheumicin F

Details

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Internal ID f4790705-12ef-48ea-984e-c512e66526c7
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name (Z)-3-hydroxy-N-[1-[[(9S,12R,15S,16S)-9-[(1S)-1-hydroxyethyl]-12-(hydroxymethyl)-16-methyl-3,6-bis(2-methylpropyl)-2,5,8,11,14-pentaoxo-1-oxa-4,7,10,13-tetrazacyclohexadec-15-yl]amino]-4-methyl-1-oxopentan-2-yl]tetradec-7-enamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C43H76N6O11/c1-10-11-12-13-14-15-16-17-18-19-30(52)23-35(53)44-31(20-25(2)3)39(55)49-37-29(9)60-43(59)33(22-27(6)7)46-38(54)32(21-26(4)5)45-41(57)36(28(8)51)48-40(56)34(24-50)47-42(37)58/h15-16,25-34,36-37,50-52H,10-14,17-24H2,1-9H3,(H,44,53)(H,45,57)(H,46,54)(H,47,58)(H,48,56)(H,49,55)/b16-15-/t28-,29-,30?,31?,32?,33?,34+,36-,37-/m0/s1
InChI Key RHJAHLYWTDULNL-HJTHNFCZSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C43H76N6O11
Molecular Weight 853.10 g/mol
Exact Mass 852.55720726 g/mol
Topological Polar Surface Area (TPSA) 262.00 Ų
XlogP 5.80

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Ngercheumicin F

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.74% 98.95%
CHEMBL3837 P07711 Cathepsin L 99.68% 96.61%
CHEMBL3060 Q9Y345 Glycine transporter 2 98.96% 99.17%
CHEMBL3359 P21462 Formyl peptide receptor 1 97.62% 93.56%
CHEMBL4769 O95749 Geranylgeranyl pyrophosphate synthetase 97.25% 92.08%
CHEMBL230 P35354 Cyclooxygenase-2 96.06% 89.63%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 95.82% 96.47%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 95.80% 91.11%
CHEMBL2094135 Q96BI3 Gamma-secretase 94.53% 98.05%
CHEMBL4072 P07858 Cathepsin B 94.03% 93.67%
CHEMBL3892 Q99500 Sphingosine 1-phosphate receptor Edg-3 93.60% 97.29%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 93.30% 91.81%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 93.11% 96.90%
CHEMBL5103 Q969S8 Histone deacetylase 10 90.41% 90.08%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 89.88% 92.88%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 89.66% 96.11%
CHEMBL2413 P32246 C-C chemokine receptor type 1 89.62% 89.50%
CHEMBL1806 P11388 DNA topoisomerase II alpha 89.10% 89.00%
CHEMBL4227 P25090 Lipoxin A4 receptor 88.75% 100.00%
CHEMBL4588 P22894 Matrix metalloproteinase 8 88.52% 94.66%
CHEMBL236 P41143 Delta opioid receptor 88.14% 99.35%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 88.05% 97.14%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 88.01% 95.00%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 87.64% 90.71%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 87.60% 96.09%
CHEMBL4462 Q8IXJ6 NAD-dependent deacetylase sirtuin 2 87.51% 90.24%
CHEMBL4481 P35228 Nitric oxide synthase, inducible 86.83% 94.80%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 86.71% 90.93%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 85.65% 95.56%
CHEMBL1949 P62937 Cyclophilin A 83.69% 98.57%
CHEMBL3401 O75469 Pregnane X receptor 83.67% 94.73%
CHEMBL340 P08684 Cytochrome P450 3A4 83.60% 91.19%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 83.53% 97.64%
CHEMBL2955 O95136 Sphingosine 1-phosphate receptor Edg-5 83.33% 92.86%
CHEMBL4801 P29466 Caspase-1 83.02% 96.85%
CHEMBL1801 P00747 Plasminogen 82.96% 92.44%
CHEMBL2001 Q9H244 Purinergic receptor P2Y12 82.72% 96.00%
CHEMBL221 P23219 Cyclooxygenase-1 82.55% 90.17%
CHEMBL1255126 O15151 Protein Mdm4 82.32% 90.20%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 81.44% 100.00%
CHEMBL299 P17252 Protein kinase C alpha 80.71% 98.03%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 80.33% 99.23%
CHEMBL5255 O00206 Toll-like receptor 4 80.21% 92.50%
CHEMBL2514 O95665 Neurotensin receptor 2 80.14% 100.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Echinocereus triglochidiatus

Cross-Links

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PubChem 139583843
LOTUS LTS0076093
wikiData Q105288008