Microviridin C

Details

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Internal ID 2f7a1b91-c16a-41ce-a3c5-029a0f906cc3
Taxonomy Organic Polymers > Polypeptides
IUPAC Name (2S)-2-[[(1S,4S,7S,10S,19S,22S,28S,31S,37R,38S,41S)-38-[[(2S,3R)-2-[[2-[[(2S)-2-acetamido-3-phenylpropanoyl]amino]acetyl]amino]-3-hydroxybutanoyl]amino]-31-(hydroxymethyl)-22-[(4-hydroxyphenyl)methyl]-4-(1H-indol-2-ylmethyl)-7-(3-methoxy-3-oxopropyl)-37-methyl-41-(2-methylpropyl)-2,5,8,13,20,23,29,32,35,39,42-undecaoxo-36-oxa-3,6,9,14,21,24,30,33,40,43-decazatricyclo[17.14.10.024,28]tritetracontane-10-carbonyl]amino]-3-(4-hydroxyphenyl)propanoic acid
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C85H110N16O25/c1-44(2)35-59-77(115)90-56-19-12-13-33-86-67(107)31-29-57(76(114)97-64(85(123)124)38-50-23-27-54(106)28-24-50)91-75(113)58(30-32-69(109)125-6)92-78(116)61(40-52-39-51-17-10-11-18-55(51)89-52)93-79(117)62(94-80(118)65(43-102)98-81(119)66-20-14-34-101(66)84(122)63(96-74(56)112)37-49-21-25-53(105)26-22-49)41-70(110)126-46(4)72(83(121)95-59)100-82(120)71(45(3)103)99-68(108)42-87-73(111)60(88-47(5)104)36-48-15-8-7-9-16-48/h7-11,15-18,21-28,39,44-46,56-66,71-72,89,102-103,105-106H,12-14,19-20,29-38,40-43H2,1-6H3,(H,86,107)(H,87,111)(H,88,104)(H,90,115)(H,91,113)(H,92,116)(H,93,117)(H,94,118)(H,95,121)(H,96,112)(H,97,114)(H,98,119)(H,99,108)(H,100,120)(H,123,124)/t45-,46-,56+,57+,58+,59+,60+,61+,62+,63+,64+,65+,66+,71+,72+/m1/s1
InChI Key WMSHUAZOBJFDIH-MJWXGQQYSA-N
Popularity 4 references in papers

Physical and Chemical Properties

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Molecular Formula C85H110N16O25
Molecular Weight 1755.90 g/mol
Exact Mass 1754.78280306 g/mol
Topological Polar Surface Area (TPSA) 614.00 Ų
XlogP 1.50
Atomic LogP (AlogP) -3.33
H-Bond Acceptor 24
H-Bond Donor 20
Rotatable Bonds 25

Synonyms

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RefChem:158814
((3S,6S,9S,12S,15S,24S,27S,32aS,35S,38S,39R)-9-((1H-indol-2-yl)methyl)-38-((2S,3R)-2-(2-((S)-2-acetamido-3-phenylpropanamido)acetamido)-3-hydroxybutanamido)-27-(4-hydroxybenzyl)-3-(hydroxymethyl)-35-isobutyl-12-(3-methoxy-3-oxopropyl)-39-methyl-1,4,7,10,13,18,25,28,34,37,41-undecaoxodotriacontahydro-24,6-(epiminoethanoiminopropanooxyethano)pyrrolo(1,2-d)(1,4,7,10,13,16,19,24)octaazacyclotriacontine-15-carbonyl)-L-tyrosine
((3S,6S,9S,12S,15S,24S,27S,32aS,35S,38S,39R)-9-((1H-indol-2-yl)methyl)-38-((2S,3R)-2-(2-((S)-2-acetamido-3-phenylpropanamido)acetamido)-3-hydroxybutanamido)-27-(4-hydroxybenzyl)-3-(hydroxymethyl)-35-isobutyl-12-(3-methoxy-3-oxopropyl)-39-methyl-1,4,7,10,13,18,25,28,34,37,41-undecaoxodotriacontahydro-24,6-(epiminoethanoiminopropanooxyethano)pyrrolo[1,2-d][1,4,7,10,13,16,19,24]octaazacyclotriacontine-15-carbonyl)-L-tyrosine
(2S)-2-((((1S,4S,7S,10S,19S,22S,28S,31S,37R,38S,41S)-38-(((2S,3R)-1,3-dihydroxy-2-((1-hydroxy-2-(((2S)-1-hydroxy-2-(1-hydroxyethylideneamino)-3-phenylpropylidene)amino)ethylidene)amino)butylidene)amino)-2,5,8,13,20,29,32,39,42-nonahydroxy-31-(hydroxymethyl)-22-((4-hydroxyphenyl)methyl)-4-(1H-indol-2-ylmethyl)-7-(3-methoxy-3-oxopropyl)-37-methyl-41-(2-methylpropyl)-23,35-dioxo-36-oxa-3,6,9,14,21,24,30,33,40,43-decazatricyclo(17.14.10.024,28)tritetraconta-2,5,8,13,20,29,32,39,42-nonaen-10-yl)-hydroxymethylidene)amino)-3-(4-hydroxyphenyl)propanoic acid
(2S)-2-(((1S,4S,7S,10S,19S,22S,28S,31S,37R,38S,41S)-38-(((2S,3R)-2-((2-(((2S)-2-acetamido-3-phenylpropanoyl)amino)acetyl)amino)-3-hydroxybutanoyl)amino)-31-(hydroxymethyl)-22-((4-hydroxyphenyl)methyl)-4-(1H-indol-2-ylmethyl)-7-(3-methoxy-3-oxopropyl)-37-methyl-41-(2-methylpropyl)-2,5,8,13,20,23,29,32,35,39,42-undecaoxo-36-oxa-3,6,9,14,21,24,30,33,40,43-decazatricyclo(17.14.10.024,28)tritetracontane-10-carbonyl)amino)-3-(4-hydroxyphenyl)propanoic acid
(2S)-2-[[(1S,4S,7S,10S,19S,22S,28S,31S,37R,38S,41S)-38-[[(2S,3R)-2-[[2-[[(2S)-2-acetamido-3-phenylpropanoyl]amino]acetyl]amino]-3-hydroxybutanoyl]amino]-31-(hydroxymethyl)-22-[(4-hydroxyphenyl)methyl]-4-(1H-indol-2-ylmethyl)-7-(3-methoxy-3-oxopropyl)-37-methyl-41-(2-methylpropyl)-2,5,8,13,20,23,29,32,35,39,42-undecaoxo-36-oxa-3,6,9,14,21,24,30,33,40,43-decazatricyclo[17.14.10.024,28]tritetracontane-10-carbonyl]amino]-3-(4-hydroxyphenyl)propanoic acid
(2S)-2-[[[(1S,4S,7S,10S,19S,22S,28S,31S,37R,38S,41S)-38-[[(2S,3R)-1,3-dihydroxy-2-[[1-hydroxy-2-[[(2S)-1-hydroxy-2-(1-hydroxyethylideneamino)-3-phenylpropylidene]amino]ethylidene]amino]butylidene]amino]-2,5,8,13,20,29,32,39,42-nonahydroxy-31-(hydroxymethyl)-22-[(4-hydroxyphenyl)methyl]-4-(1H-indol-2-ylmethyl)-7-(3-methoxy-3-oxopropyl)-37-methyl-41-(2-methylpropyl)-23,35-dioxo-36-oxa-3,6,9,14,21,24,30,33,40,43-decazatricyclo[17.14.10.024,28]tritetraconta-2,5,8,13,20,29,32,39,42-nonaen-10-yl]-hydroxymethylidene]amino]-3-(4-hydroxyphenyl)propanoic acid
CHEBI:207756
DTXSID801334791

2D Structure

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2D Structure of Microviridin C

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
Human Intestinal Absorption + 0.7601 76.01%
Caco-2 - 0.8633 86.33%
Blood Brain Barrier - 1.0000 100.00%
Human oral bioavailability - 0.7286 72.86%
Subcellular localzation Lysosomes 0.3423 34.23%
OATP2B1 inhibitior - 1.0000 100.00%
OATP1B1 inhibitior + 0.7987 79.87%
OATP1B3 inhibitior + 0.9207 92.07%
MATE1 inhibitior - 0.7409 74.09%
OCT2 inhibitior - 0.9000 90.00%
BSEP inhibitior + 0.9691 96.91%
P-glycoprotein inhibitior + 0.7419 74.19%
P-glycoprotein substrate + 0.8687 86.87%
CYP3A4 substrate + 0.7613 76.13%
CYP2C9 substrate - 0.6112 61.12%
CYP2D6 substrate - 0.8448 84.48%
CYP3A4 inhibition - 0.5736 57.36%
CYP2C9 inhibition - 0.8190 81.90%
CYP2C19 inhibition - 0.8328 83.28%
CYP2D6 inhibition - 0.8579 85.79%
CYP1A2 inhibition - 0.9428 94.28%
CYP2C8 inhibition + 0.8592 85.92%
CYP inhibitory promiscuity - 0.6138 61.38%
UGT catelyzed + 0.7000 70.00%
Carcinogenicity (binary) - 0.8700 87.00%
Carcinogenicity (trinary) Non-required 0.6152 61.52%
Eye corrosion - 0.9889 98.89%
Eye irritation - 0.8954 89.54%
Skin irritation - 0.7866 78.66%
Skin corrosion - 0.9372 93.72%
Ames mutagenesis - 0.5919 59.19%
Human Ether-a-go-go-Related Gene inhibition + 0.7326 73.26%
Micronuclear + 0.8200 82.00%
Hepatotoxicity + 0.5040 50.40%
skin sensitisation - 0.8939 89.39%
Respiratory toxicity + 0.7556 75.56%
Reproductive toxicity + 0.9667 96.67%
Mitochondrial toxicity + 0.9250 92.50%
Nephrotoxicity + 0.6218 62.18%
Acute Oral Toxicity (c) III 0.5897 58.97%
Estrogen receptor binding - 0.4753 47.53%
Androgen receptor binding + 0.7322 73.22%
Thyroid receptor binding + 0.7773 77.73%
Glucocorticoid receptor binding + 0.8322 83.22%
Aromatase binding + 0.7983 79.83%
PPAR gamma + 0.7794 77.94%
Honey bee toxicity - 0.6169 61.69%
Biodegradation - 0.8250 82.50%
Crustacea aquatic toxicity - 0.5100 51.00%
Fish aquatic toxicity + 0.9236 92.36%

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 100.00% 98.95%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 99.45% 85.14%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.37% 91.11%
CHEMBL3524 P56524 Histone deacetylase 4 98.88% 92.97%
CHEMBL2288 Q13526 Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 98.53% 91.71%
CHEMBL1255126 O15151 Protein Mdm4 98.50% 90.20%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 98.21% 97.14%
CHEMBL3060 Q9Y345 Glycine transporter 2 97.67% 99.17%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 97.64% 97.64%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.52% 96.09%
CHEMBL3837 P07711 Cathepsin L 97.39% 96.61%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 97.36% 82.38%
CHEMBL5103 Q969S8 Histone deacetylase 10 96.63% 90.08%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 96.09% 99.23%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 94.37% 94.45%
CHEMBL3137262 O60341 LSD1/CoREST complex 94.10% 97.09%
CHEMBL3476 O15111 Inhibitor of nuclear factor kappa B kinase alpha subunit 93.90% 95.83%
CHEMBL259 P32245 Melanocortin receptor 4 93.70% 95.38%
CHEMBL2535 P11166 Glucose transporter 93.50% 98.75%
CHEMBL3359 P21462 Formyl peptide receptor 1 91.52% 93.56%
CHEMBL3310 Q96DB2 Histone deacetylase 11 91.19% 88.56%
CHEMBL2413 P32246 C-C chemokine receptor type 1 91.06% 89.50%
CHEMBL2563 Q9UQL6 Histone deacetylase 5 90.93% 89.67%
CHEMBL4777 P25929 Neuropeptide Y receptor type 1 90.79% 96.67%
CHEMBL2095172 P14867 GABA-A receptor; alpha-1/beta-2/gamma-2 90.56% 92.67%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 90.03% 95.50%
CHEMBL340 P08684 Cytochrome P450 3A4 89.59% 91.19%
CHEMBL4801 P29466 Caspase-1 89.36% 96.85%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 89.26% 93.00%
CHEMBL1801 P00747 Plasminogen 89.24% 92.44%
CHEMBL4608 P33032 Melanocortin receptor 5 89.13% 97.00%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 88.63% 90.71%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 88.31% 93.10%
CHEMBL1806 P11388 DNA topoisomerase II alpha 87.99% 89.00%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 87.17% 95.56%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 86.52% 95.00%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 86.21% 96.90%
CHEMBL4227 P25090 Lipoxin A4 receptor 84.79% 100.00%
CHEMBL1293249 Q13887 Kruppel-like factor 5 84.24% 86.33%
CHEMBL4394 Q9NYA1 Sphingosine kinase 1 84.13% 96.03%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 83.67% 95.89%
CHEMBL3105 P09874 Poly [ADP-ribose] polymerase-1 83.67% 93.90%
CHEMBL5852 Q96P65 Pyroglutamylated RFamide peptide receptor 83.05% 85.00%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 82.71% 93.03%
CHEMBL221 P23219 Cyclooxygenase-1 82.69% 90.17%
CHEMBL4644 P41968 Melanocortin receptor 3 82.61% 99.52%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 82.52% 99.15%
CHEMBL230 P35354 Cyclooxygenase-2 82.36% 89.63%
CHEMBL1937 Q92769 Histone deacetylase 2 81.82% 94.75%
CHEMBL1744525 P43490 Nicotinamide phosphoribosyltransferase 81.66% 96.25%
CHEMBL2803 P43403 Tyrosine-protein kinase ZAP-70 81.63% 82.50%
CHEMBL5608 Q16288 NT-3 growth factor receptor 81.22% 95.89%
CHEMBL2000 P03952 Plasma kallikrein 80.81% 93.92%
CHEMBL256 P0DMS8 Adenosine A3 receptor 80.72% 95.93%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 80.37% 98.33%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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Cross-Links

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PubChem 16142910
LOTUS LTS0144800
wikiData Q104203121