Marikarin

Details

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Internal ID c2117c67-f021-4c9d-a317-533499f9a750
Taxonomy Phenylpropanoids and polyketides > Stilbenes
IUPAC Name (2S,10R,11R)-2,4-dihydroxy-6-methoxy-10-(4-methoxyphenyl)-11-phenyl-9-oxa-14,19-diazapentacyclo[10.7.0.02,10.03,8.014,18]nonadeca-1(12),3,5,7,18-pentaen-13-one
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C30H26N2O6/c1-36-19-12-10-18(11-13-19)30-25(17-7-4-3-5-8-17)24-27(31-23-9-6-14-32(23)28(24)34)29(30,35)26-21(33)15-20(37-2)16-22(26)38-30/h3-5,7-8,10-13,15-16,25,33,35H,6,9,14H2,1-2H3/t25-,29+,30+/m1/s1
InChI Key KTFBOLLZQNMGNM-CPESWEKQSA-N
Popularity 0 references in papers

Physical and Chemical Properties

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Molecular Formula C30H26N2O6
Molecular Weight 510.50 g/mol
Exact Mass 510.17908655 g/mol
Topological Polar Surface Area (TPSA) 101.00 Ų
XlogP 2.30

Synonyms

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(-)-(6R,6aR,11bS)-11,11b-Dihydroxy-9-methoxy-6a-(4-methoxyphenyl)-6-phenyl-2,3,5,6,6a,11b-hexahydro-1H-benzo[4",5"]furo[2",3":4",5"]cyclopenta[1',2'-d]pyrrolo[1,2-a]pyrimidin-5-one
7H-benzofuro[2',3':4,5]cyclopenta[1,2-d]pyrrolo[1,2-a]pyrimidin-7-one, 5a,6,9,10,11,12b-hexahydro-1,12b-dihydroxy-3-methoxy-5a-(4-methoxyphenyl)-6-phenyl-, (5aR,6R,12bS)-
InChI=1/C30H26N2O6/c1-36-19-12-10-18(11-13-19)30-25(17-7-4-3-5-8-17)24-27(31-23-9-6-14-32(23)28(24)34)29(30,35)26-21(33)15-20(37-2)16-22(26)38-30/h3-5,7-8,10-13,15-16,25,33,35H,6,9,14H2,1-2H3/t25-,29+,30+/m1/s
rel-(5aR,6R,12bS)-1,12b-dihydroxy-3-methoxy-5a-(4-methoxyphenyl)-6-phenyl-5a,6,9,10,11,12b-hexahydro-7H-[1]benzofuro[2',3':4,5]cyclopenta[1,2-d]pyrrolo[1,2-a]pyrimidin-7-one

2D Structure

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2D Structure of Marikarin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.19% 91.11%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 97.98% 95.56%
CHEMBL2581 P07339 Cathepsin D 97.60% 98.95%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 97.59% 85.14%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 97.06% 99.15%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 96.86% 99.23%
CHEMBL1293249 Q13887 Kruppel-like factor 5 95.22% 86.33%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 95.21% 96.09%
CHEMBL5697 Q9GZT9 Egl nine homolog 1 95.03% 93.40%
CHEMBL3192 Q9BY41 Histone deacetylase 8 94.94% 93.99%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 93.18% 94.00%
CHEMBL3137262 O60341 LSD1/CoREST complex 88.56% 97.09%
CHEMBL4208 P20618 Proteasome component C5 87.79% 90.00%
CHEMBL5203 P33316 dUTP pyrophosphatase 85.65% 99.18%
CHEMBL5608 Q16288 NT-3 growth factor receptor 84.97% 95.89%
CHEMBL2146302 O94925 Glutaminase kidney isoform, mitochondrial 83.01% 100.00%
CHEMBL2095226 P05556 Integrin alpha-5/beta-1 82.11% 96.39%
CHEMBL1821 P08173 Muscarinic acetylcholine receptor M4 81.37% 94.08%
CHEMBL2535 P11166 Glucose transporter 80.94% 98.75%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 80.69% 95.50%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Aglaia gracilis

Cross-Links

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PubChem 636971
LOTUS LTS0226348
wikiData Q105145760