Maltacine B1a

Details

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Internal ID 620074fb-aa86-4d8d-b66e-03211d61424a
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name 3-[27-[[2-[[5-amino-5-oxo-2-(pyrrolidine-2-carbonylamino)pentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-12-(3-aminopropyl)-3-butan-2-yl-9-(4-hydroxybutyl)-18-(1-hydroxyethyl)-6,15-bis[(4-hydroxyphenyl)methyl]-24-methyl-2,5,8,11,14,17,20,23,26-nonaoxo-1-oxa-4,7,10,13,16,19,22,25-octazacyclohentriacont-21-yl]propanoic acid
SMILES (Canonical) CCC(C)C1C(=O)OCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N1)CC2=CC=C(C=C2)O)CCCCO)CCCN)CC3=CC=C(C=C3)O)C(C)O)CCC(=O)O)C)NC(=O)C(CC4=CC=C(C=C4)O)NC(=O)C(CCC(=O)N)NC(=O)C5CCCN5
SMILES (Isomeric) CCC(C)C1C(=O)OCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N1)CC2=CC=C(C=C2)O)CCCCO)CCCN)CC3=CC=C(C=C3)O)C(C)O)CCC(=O)O)C)NC(=O)C(CC4=CC=C(C=C4)O)NC(=O)C(CCC(=O)N)NC(=O)C5CCCN5
InChI InChI=1S/C72H104N14O21/c1-5-39(2)59-72(106)107-35-9-7-13-49(79-68(102)54(36-42-16-22-45(89)23-17-42)82-66(100)52(28-30-57(74)92)81-62(96)48-15-11-33-75-48)63(97)76-40(3)61(95)77-53(29-31-58(93)94)67(101)86-60(41(4)88)71(105)84-55(37-43-18-24-46(90)25-19-43)69(103)80-51(14-10-32-73)64(98)78-50(12-6-8-34-87)65(99)83-56(70(104)85-59)38-44-20-26-47(91)27-21-44/h16-27,39-41,48-56,59-60,75,87-91H,5-15,28-38,73H2,1-4H3,(H2,74,92)(H,76,97)(H,77,95)(H,78,98)(H,79,102)(H,80,103)(H,81,96)(H,82,100)(H,83,99)(H,84,105)(H,85,104)(H,86,101)(H,93,94)
InChI Key VRVZMVNJCUIYQB-UHFFFAOYSA-N
Popularity 0 references in papers

Physical and Chemical Properties

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Molecular Formula C72H104N14O21
Molecular Weight 1501.70 g/mol
Exact Mass 1500.75004638 g/mol
Topological Polar Surface Area (TPSA) 566.00 Ų
XlogP -1.60

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Maltacine B1a

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 99.90% 93.10%
CHEMBL3837 P07711 Cathepsin L 99.86% 96.61%
CHEMBL2581 P07339 Cathepsin D 99.80% 98.95%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 99.20% 94.45%
CHEMBL4040 P28482 MAP kinase ERK2 99.07% 83.82%
CHEMBL3137262 O60341 LSD1/CoREST complex 99.06% 97.09%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.52% 96.09%
CHEMBL1255126 O15151 Protein Mdm4 98.05% 90.20%
CHEMBL3060 Q9Y345 Glycine transporter 2 97.70% 99.17%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 97.62% 95.00%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 97.58% 97.23%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.33% 91.11%
CHEMBL5103 Q969S8 Histone deacetylase 10 96.60% 90.08%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 96.43% 97.64%
CHEMBL236 P41143 Delta opioid receptor 95.22% 99.35%
CHEMBL2514 O95665 Neurotensin receptor 2 95.16% 100.00%
CHEMBL1293287 P14735 Insulin-degrading enzyme 95.09% 88.10%
CHEMBL3359 P21462 Formyl peptide receptor 1 95.07% 93.56%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 94.41% 92.88%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 93.59% 97.14%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 93.20% 96.47%
CHEMBL4777 P25929 Neuropeptide Y receptor type 1 93.17% 96.67%
CHEMBL259 P32245 Melanocortin receptor 4 92.74% 95.38%
CHEMBL2094135 Q96BI3 Gamma-secretase 92.72% 98.05%
CHEMBL5608 Q16288 NT-3 growth factor receptor 92.70% 95.89%
CHEMBL3880 P07900 Heat shock protein HSP 90-alpha 92.36% 96.21%
CHEMBL2288 Q13526 Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 92.20% 91.71%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 91.93% 93.00%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 90.88% 88.42%
CHEMBL4227 P25090 Lipoxin A4 receptor 90.78% 100.00%
CHEMBL242 Q92731 Estrogen receptor beta 90.35% 98.35%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 90.31% 90.71%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 89.96% 95.50%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 89.85% 95.56%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 89.69% 95.50%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 89.46% 96.11%
CHEMBL233 P35372 Mu opioid receptor 89.06% 97.93%
CHEMBL4198 P98170 Inhibitor of apoptosis protein 3 88.84% 97.79%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 88.27% 100.00%
CHEMBL340 P08684 Cytochrome P450 3A4 88.02% 91.19%
CHEMBL3310 Q96DB2 Histone deacetylase 11 87.85% 88.56%
CHEMBL206 P03372 Estrogen receptor alpha 87.44% 97.64%
CHEMBL4018 P49146 Neuropeptide Y receptor type 2 87.33% 98.94%
CHEMBL2208 P49137 MAP kinase-activated protein kinase 2 86.68% 95.20%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 86.46% 85.14%
CHEMBL2001 Q9H244 Purinergic receptor P2Y12 86.36% 96.00%
CHEMBL2413 P32246 C-C chemokine receptor type 1 86.28% 89.50%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 86.17% 96.90%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 85.82% 97.33%
CHEMBL1801 P00747 Plasminogen 85.65% 92.44%
CHEMBL1907589 P17787 Neuronal acetylcholine receptor; alpha4/beta2 85.59% 94.55%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 84.77% 96.00%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 84.69% 95.89%
CHEMBL226 P30542 Adenosine A1 receptor 84.38% 95.93%
CHEMBL1075317 P61964 WD repeat-containing protein 5 84.34% 96.33%
CHEMBL2327 P21452 Neurokinin 2 receptor 84.30% 98.89%
CHEMBL4123 P30989 Neurotensin receptor 1 84.11% 96.67%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 84.05% 82.69%
CHEMBL1907591 P30926 Neuronal acetylcholine receptor; alpha4/beta4 83.49% 100.00%
CHEMBL3232685 O00257 E3 SUMO-protein ligase CBX4 83.42% 93.00%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 83.37% 98.33%
CHEMBL253 P34972 Cannabinoid CB2 receptor 83.00% 97.25%
CHEMBL1937 Q92769 Histone deacetylase 2 82.77% 94.75%
CHEMBL249 P25103 Neurokinin 1 receptor 81.94% 99.17%
CHEMBL2072 P35499 Sodium channel protein type IV alpha subunit 81.89% 92.32%
CHEMBL4633 P22001 Voltage-gated potassium channel subunit Kv1.3 81.26% 100.00%
CHEMBL5261 Q7L7X3 Serine/threonine-protein kinase TAO1 81.05% 89.33%
CHEMBL3476 O15111 Inhibitor of nuclear factor kappa B kinase alpha subunit 80.56% 95.83%
CHEMBL4581 P52732 Kinesin-like protein 1 80.55% 93.18%
CHEMBL4330 Q9NS75 Cysteinyl leukotriene receptor 2 80.41% 98.00%
CHEMBL5852 Q96P65 Pyroglutamylated RFamide peptide receptor 80.11% 85.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139583720
LOTUS LTS0023057
wikiData Q75066676