Lyngbyabellin E

Details

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Internal ID a8952338-aec2-4507-9e0b-ea7a9e27fd2b
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name [(5R,12S,13S,16S)-12-(4,4-dichloropentyl)-16-(2-hydroxypropan-2-yl)-13-methyl-2,10,14-trioxo-3,11,15-trioxa-7,18-dithia-20,21-diazatricyclo[15.2.1.16,9]henicosa-1(19),6(21),8,17(20)-tetraen-5-yl] (3R,4S)-3-acetyloxy-4-(butanoylamino)-6-methylheptanoate
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C37H51Cl2N3O12S2/c1-9-11-28(44)40-22(14-19(2)3)26(51-21(5)43)15-29(45)52-27-16-50-34(47)23-17-56-32(42-23)30(36(6,7)49)54-33(46)20(4)25(12-10-13-37(8,38)39)53-35(48)24-18-55-31(27)41-24/h17-20,22,25-27,30,49H,9-16H2,1-8H3,(H,40,44)/t20-,22-,25-,26+,27+,30+/m0/s1
InChI Key UQKCUAHEIXPDOS-GCKMHMQYSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C37H51Cl2N3O12S2
Molecular Weight 864.90 g/mol
Exact Mass 863.2291218 g/mol
Topological Polar Surface Area (TPSA) 263.00 Ų
XlogP 6.20

Synonyms

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DTXSID001334761

2D Structure

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2D Structure of Lyngbyabellin E

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.79% 98.95%
CHEMBL4040 P28482 MAP kinase ERK2 98.99% 83.82%
CHEMBL230 P35354 Cyclooxygenase-2 98.94% 89.63%
CHEMBL253 P34972 Cannabinoid CB2 receptor 97.39% 97.25%
CHEMBL2996 Q05655 Protein kinase C delta 95.27% 97.79%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 94.95% 91.11%
CHEMBL3060 Q9Y345 Glycine transporter 2 94.70% 99.17%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 94.60% 99.23%
CHEMBL3401 O75469 Pregnane X receptor 93.03% 94.73%
CHEMBL3359 P21462 Formyl peptide receptor 1 91.95% 93.56%
CHEMBL4657 Q6V1X1 Dipeptidyl peptidase VIII 91.66% 97.21%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 90.79% 85.14%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 90.74% 94.45%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 90.67% 96.90%
CHEMBL3976 Q9UHL4 Dipeptidyl peptidase II 89.84% 92.29%
CHEMBL2243 O00519 Anandamide amidohydrolase 89.62% 97.53%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 88.49% 98.33%
CHEMBL3891 P07384 Calpain 1 88.20% 93.04%
CHEMBL1293249 Q13887 Kruppel-like factor 5 88.03% 86.33%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 87.01% 96.09%
CHEMBL3691 Q13822 Autotaxin 86.91% 96.39%
CHEMBL2265 P23141 Acyl coenzyme A:cholesterol acyltransferase 86.18% 85.94%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 85.75% 100.00%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 84.92% 97.14%
CHEMBL340 P08684 Cytochrome P450 3A4 84.39% 91.19%
CHEMBL5103 Q969S8 Histone deacetylase 10 84.31% 90.08%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 84.19% 96.00%
CHEMBL1806 P11388 DNA topoisomerase II alpha 82.30% 89.00%
CHEMBL5028 O14672 ADAM10 81.77% 97.50%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 81.00% 93.03%
CHEMBL5255 O00206 Toll-like receptor 4 80.88% 92.50%
CHEMBL2373 P21730 C5a anaphylatoxin chemotactic receptor 80.66% 92.62%
CHEMBL299 P17252 Protein kinase C alpha 80.49% 98.03%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 11622047
LOTUS LTS0070930
wikiData Q77424901