Lobatamide A

Details

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Internal ID 38047e2a-bc79-4bd8-8bf7-f52ed01c98de
Taxonomy Phenylpropanoids and polyketides > Macrolides and analogues
IUPAC Name (Z,4Z)-N-[(E)-3-[(9E,12Z)-11,19-dihydroxy-8,12-dimethyl-2,6-dioxo-3,7-dioxabicyclo[13.4.0]nonadeca-1(15),9,12,16,18-pentaen-4-yl]prop-1-enyl]-4-methoxyiminobut-2-enamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C27H32N2O8/c1-18-11-13-20-7-4-9-23(31)26(20)27(34)37-21(17-25(33)36-19(2)12-14-22(18)30)8-5-15-28-24(32)10-6-16-29-35-3/h4-7,9-12,14-16,19,21-22,30-31H,8,13,17H2,1-3H3,(H,28,32)/b10-6-,14-12+,15-5+,18-11-,29-16-
InChI Key JYHIHHYYXXKTTJ-JSFHDESQSA-N
Popularity 5 references in papers

Physical and Chemical Properties

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Molecular Formula C27H32N2O8
Molecular Weight 512.60 g/mol
Exact Mass 512.21586598 g/mol
Topological Polar Surface Area (TPSA) 144.00 Ų
XlogP 3.00

Synonyms

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(Z,4Z)-N-[(E)-3-[(9E,12Z)-11,19-dihydroxy-8,12-dimethyl-2,6-dioxo-3,7-dioxabicyclo[13.4.0]nonadeca-1(15),9,12,16,18-pentaen-4-yl]prop-1-enyl]-4-methoxyiminobut-2-enamide
(Z,4Z)-N-((E)-3-((9E,12Z)-11,19-dihydroxy-8,12-dimethyl-2,6-dioxo-3,7-dioxabicyclo(13.4.0)nonadeca-1(15),9,12,16,18-pentaen-4-yl)prop-1-enyl)-4-methoxyiminobut-2-enamide
RefChem:924863
200563-47-9
YM-75518
SCHEMBL81777
CHEBI:216143

2D Structure

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2D Structure of Lobatamide A

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 98.34% 98.95%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.81% 91.11%
CHEMBL3401 O75469 Pregnane X receptor 95.82% 94.73%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.72% 95.56%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 91.28% 99.23%
CHEMBL3060 Q9Y345 Glycine transporter 2 90.65% 99.17%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 89.87% 94.45%
CHEMBL1806 P11388 DNA topoisomerase II alpha 89.60% 89.00%
CHEMBL1293249 Q13887 Kruppel-like factor 5 87.80% 86.33%
CHEMBL5608 Q16288 NT-3 growth factor receptor 87.05% 95.89%
CHEMBL3137262 O60341 LSD1/CoREST complex 86.09% 97.09%
CHEMBL2996 Q05655 Protein kinase C delta 85.24% 97.79%
CHEMBL3359 P21462 Formyl peptide receptor 1 85.08% 93.56%
CHEMBL4793 Q86TI2 Dipeptidyl peptidase IX 84.84% 96.95%
CHEMBL3192 Q9BY41 Histone deacetylase 8 84.46% 93.99%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 81.86% 93.03%
CHEMBL5697 Q9GZT9 Egl nine homolog 1 80.99% 93.40%
CHEMBL5028 O14672 ADAM10 80.73% 97.50%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 10505925
LOTUS LTS0070747
wikiData Q77499050