Kopsimaline B

Details

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Internal ID 64c9b820-976e-4643-a458-e4ae318f8b6f
Taxonomy Alkaloids and derivatives > Aspidofractine alkaloids
IUPAC Name dimethyl (1R,2R,4S,9R,17S,18R,19R,22R)-14,18,19-trihydroxy-3-oxa-6,16-diazaheptacyclo[15.2.2.11,6.02,4.09,17.010,15.09,22]docosa-10(15),11,13-triene-16,18-dicarboxylate
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C23H26N2O8/c1-31-18(28)23(30)17(27)20-6-7-22(23)21(8-9-24(16(20)21)10-13-15(20)33-13)11-4-3-5-12(26)14(11)25(22)19(29)32-2/h3-5,13,15-17,26-27,30H,6-10H2,1-2H3/t13-,15-,16-,17+,20+,21+,22-,23+/m0/s1
InChI Key SNYWZYAYAZZSTH-XOVVLEAVSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C23H26N2O8
Molecular Weight 458.50 g/mol
Exact Mass 458.16891579 g/mol
Topological Polar Surface Area (TPSA) 132.00 Ų
XlogP 0.20

Synonyms

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dimethyl (1R,2R,4S,9R,17S,18R,19R,22R)-14,18,19-trihydroxy-3-oxa-6,16-diazaheptacyclo(15.2.2.11,6.02,4.09,17.010,15.09,22)docosa-10(15),11,13-triene-16,18-dicarboxylate
dimethyl (1R,2R,4S,9R,17S,18R,19R,22R)-14,18,19-trihydroxy-3-oxa-6,16-diazaheptacyclo[15.2.2.11,6.02,4.09,17.010,15.09,22]docosa-10(15),11,13-triene-16,18-dicarboxylate
RefChem:151409
1005004-47-6
CHEMBL255673

2D Structure

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2D Structure of Kopsimaline B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.77% 96.09%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.89% 91.11%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 93.40% 95.56%
CHEMBL2581 P07339 Cathepsin D 93.28% 98.95%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 91.77% 85.14%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 91.70% 94.45%
CHEMBL5028 O14672 ADAM10 90.11% 97.50%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 89.95% 99.23%
CHEMBL4208 P20618 Proteasome component C5 87.68% 90.00%
CHEMBL5608 Q16288 NT-3 growth factor receptor 87.23% 95.89%
CHEMBL1293249 Q13887 Kruppel-like factor 5 84.74% 86.33%
CHEMBL4227 P25090 Lipoxin A4 receptor 82.72% 100.00%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 82.47% 97.14%
CHEMBL340 P08684 Cytochrome P450 3A4 82.02% 91.19%
CHEMBL3137262 O60341 LSD1/CoREST complex 81.92% 97.09%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 81.08% 93.03%
CHEMBL1821 P08173 Muscarinic acetylcholine receptor M4 80.77% 94.08%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Kopsia singapurensis

Cross-Links

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PubChem 24770293
LOTUS LTS0130282
wikiData Q105256769