keramamide A

Details

Top
Internal ID 9cb91b61-3a9e-41c6-b9d4-67214334b6e8
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Oligopeptides
IUPAC Name 2-[[3-benzyl-6-[(6-chloro-5-hydroxy-1H-indol-3-yl)methyl]-7-methyl-9,12-bis(2-methylpropyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazacyclononadec-15-yl]carbamoylamino]-3-phenylpropanoic acid
SMILES (Canonical) CC(C)CC1C(=O)NC(C(=O)N(C(C(=O)NC(C(=O)NCCCCC(C(=O)N1)NC(=O)NC(CC2=CC=CC=C2)C(=O)O)CC3=CC=CC=C3)CC4=CNC5=CC(=C(C=C54)O)Cl)C)CC(C)C
SMILES (Isomeric) CC(C)CC1C(=O)NC(C(=O)N(C(C(=O)NC(C(=O)NCCCCC(C(=O)N1)NC(=O)NC(CC2=CC=CC=C2)C(=O)O)CC3=CC=CC=C3)CC4=CNC5=CC(=C(C=C54)O)Cl)C)CC(C)C
InChI InChI=1S/C49H63ClN8O9/c1-28(2)20-37-45(62)55-39(21-29(3)4)47(64)58(5)41(24-32-27-52-36-26-34(50)42(59)25-33(32)36)46(63)54-38(22-30-14-8-6-9-15-30)43(60)51-19-13-12-18-35(44(61)53-37)56-49(67)57-40(48(65)66)23-31-16-10-7-11-17-31/h6-11,14-17,25-29,35,37-41,52,59H,12-13,18-24H2,1-5H3,(H,51,60)(H,53,61)(H,54,63)(H,55,62)(H,65,66)(H2,56,57,67)
InChI Key OCMXOQFOMBDMCH-UHFFFAOYSA-N
Popularity 0 references in papers

Physical and Chemical Properties

Top
Molecular Formula C49H63ClN8O9
Molecular Weight 943.50 g/mol
Exact Mass 942.4406533 g/mol
Topological Polar Surface Area (TPSA) 251.00 Ų
XlogP 6.60

Synonyms

Top
There are no found synonyms.

2D Structure

Top
2D Structure of keramamide A

3D Structure

Top

ADMET Properties (via admetSAR 2)

Top
Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

Top

Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.95% 98.95%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.37% 91.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 97.98% 94.45%
CHEMBL221 P23219 Cyclooxygenase-1 96.09% 90.17%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 95.79% 96.09%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 95.15% 97.64%
CHEMBL4040 P28482 MAP kinase ERK2 94.58% 83.82%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 94.42% 98.33%
CHEMBL2373 P21730 C5a anaphylatoxin chemotactic receptor 94.03% 92.62%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 93.12% 88.42%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 92.53% 99.15%
CHEMBL5103 Q969S8 Histone deacetylase 10 92.52% 90.08%
CHEMBL3155 P34969 Serotonin 7 (5-HT7) receptor 91.70% 90.71%
CHEMBL4072 P07858 Cathepsin B 90.92% 93.67%
CHEMBL4835 P00338 L-lactate dehydrogenase A chain 90.39% 95.34%
CHEMBL3202 P48147 Prolyl endopeptidase 89.98% 90.65%
CHEMBL3837 P07711 Cathepsin L 89.81% 96.61%
CHEMBL225 P28335 Serotonin 2c (5-HT2c) receptor 89.50% 89.62%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 88.49% 95.00%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 87.53% 93.03%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 87.15% 95.56%
CHEMBL1741221 Q9Y4P1 Cysteine protease ATG4B 86.06% 87.50%
CHEMBL2083 P15090 Fatty acid binding protein adipocyte 85.72% 95.71%
CHEMBL4208 P20618 Proteasome component C5 85.15% 90.00%
CHEMBL4644 P41968 Melanocortin receptor 3 85.09% 99.52%
CHEMBL226 P30542 Adenosine A1 receptor 84.94% 95.93%
CHEMBL2327 P21452 Neurokinin 2 receptor 84.59% 98.89%
CHEMBL4979 P13866 Sodium/glucose cotransporter 1 83.94% 98.24%
CHEMBL2413 P32246 C-C chemokine receptor type 1 83.40% 89.50%
CHEMBL3310 Q96DB2 Histone deacetylase 11 83.40% 88.56%
CHEMBL3137262 O60341 LSD1/CoREST complex 83.11% 97.09%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 83.05% 97.14%
CHEMBL1808 P12821 Angiotensin-converting enzyme 82.74% 93.39%
CHEMBL259 P32245 Melanocortin receptor 4 82.45% 95.38%
CHEMBL2095172 P14867 GABA-A receptor; alpha-1/beta-2/gamma-2 82.19% 92.67%
CHEMBL216 P11229 Muscarinic acetylcholine receptor M1 82.18% 94.23%
CHEMBL3384 Q16512 Protein kinase N1 81.58% 80.71%
CHEMBL3359 P21462 Formyl peptide receptor 1 81.48% 93.56%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 81.40% 97.23%
CHEMBL5608 Q16288 NT-3 growth factor receptor 81.39% 95.89%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 81.33% 96.90%
CHEMBL1806 P11388 DNA topoisomerase II alpha 80.68% 89.00%
CHEMBL3192 Q9BY41 Histone deacetylase 8 80.41% 93.99%
CHEMBL3430907 Q96GD4 Aurora kinase B/Inner centromere protein 80.40% 97.50%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 80.06% 100.00%
CHEMBL1075317 P61964 WD repeat-containing protein 5 80.05% 96.33%

Plants that contains it

Top
Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

Top
PubChem 72744759
LOTUS LTS0073668
wikiData Q105189461