Isaridin E

Details

Top
Internal ID 9ebdea85-1eea-45f3-848e-be8635faa974
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name (10S,13S,16S,19S)-16-benzyl-11,14-dimethyl-3-(2-methylpropyl)-10,13-di(propan-2-yl)-4-oxa-1,8,11,14,17-pentazabicyclo[17.3.0]docosane-2,5,9,12,15,18-hexone
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C35H53N5O7/c1-21(2)19-27-34(45)40-18-12-15-26(40)31(42)37-25(20-24-13-10-9-11-14-24)33(44)39(8)30(23(5)6)35(46)38(7)29(22(3)4)32(43)36-17-16-28(41)47-27/h9-11,13-14,21-23,25-27,29-30H,12,15-20H2,1-8H3,(H,36,43)(H,37,42)/t25-,26-,27?,29-,30-/m0/s1
InChI Key RTZWJENDDHDLIV-UTKDJJAFSA-N
Popularity 7 references in papers

Physical and Chemical Properties

Top
Molecular Formula C35H53N5O7
Molecular Weight 655.80 g/mol
Exact Mass 655.39449905 g/mol
Topological Polar Surface Area (TPSA) 145.00 Ų
XlogP 4.10

Synonyms

Top
RefChem:148891
(10S,13S,16S,19S)-16-benzyl-11,14-dimethyl-3-(2-methylpropyl)-10,13-di(propan-2-yl)-4-oxa-1,8,11,14,17-pentazabicyclo(17.3.0)docosane-2,5,9,12,15,18-hexone
CHEMBL227907
SCHEMBL29384850

2D Structure

Top
2D Structure of Isaridin E

3D Structure

Top

ADMET Properties (via admetSAR 2)

Top
Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

Top

Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.82% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 96.89% 96.09%
CHEMBL3524 P56524 Histone deacetylase 4 95.12% 92.97%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 95.04% 97.64%
CHEMBL333 P08253 Matrix metalloproteinase-2 94.97% 96.31%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 94.36% 95.56%
CHEMBL5103 Q969S8 Histone deacetylase 10 91.71% 90.08%
CHEMBL5608 Q16288 NT-3 growth factor receptor 91.26% 95.89%
CHEMBL253 P34972 Cannabinoid CB2 receptor 90.85% 97.25%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 90.72% 82.38%
CHEMBL226 P30542 Adenosine A1 receptor 88.57% 95.93%
CHEMBL1902 P62942 FK506-binding protein 1A 88.49% 97.05%
CHEMBL3137262 O60341 LSD1/CoREST complex 88.38% 97.09%
CHEMBL204 P00734 Thrombin 86.99% 96.01%
CHEMBL228 P31645 Serotonin transporter 86.97% 95.51%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 86.47% 93.00%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 86.19% 90.93%
CHEMBL1293249 Q13887 Kruppel-like factor 5 86.05% 86.33%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 85.87% 85.14%
CHEMBL3837 P07711 Cathepsin L 85.12% 96.61%
CHEMBL255 P29275 Adenosine A2b receptor 84.79% 98.59%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 84.68% 97.14%
CHEMBL4588 P22894 Matrix metalloproteinase 8 84.45% 94.66%
CHEMBL4616 Q92847 Ghrelin receptor 84.31% 92.00%
CHEMBL5805 Q9NR97 Toll-like receptor 8 82.80% 96.25%
CHEMBL5203 P33316 dUTP pyrophosphatase 82.68% 99.18%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 82.22% 91.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 81.42% 94.45%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 81.19% 93.03%

Plants that contains it

Top
Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

Top
PubChem 16680915
LOTUS LTS0082692
wikiData Q105245521