Hormaomycin C

Details

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Internal ID 4a3a434d-1cb1-4bff-ba9d-cb3a7391f898
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name N-[(2S)-1-[[(3S,6S,9R,12S,15R,16R,19S,21R)-6-benzyl-3-[(2S)-butan-2-yl]-16-methyl-9-[[(1R,2R)-2-nitrocyclopropyl]methyl]-2,5,8,11,14,18-hexaoxo-12-[(1R)-1-phenylethyl]-21-[(Z)-prop-1-enyl]-17-oxa-1,4,7,10,13-pentazabicyclo[17.3.0]docosan-15-yl]amino]-3-[(1S,2S)-2-nitrocyclopropyl]-1-oxopropan-2-yl]-5-chloro-1-hydroxypyrrole-2-carboxamide
SMILES (Canonical) CCC(C)C1C(=O)N2CC(CC2C(=O)OC(C(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N1)CC3=CC=CC=C3)CC4CC4[N+](=O)[O-])C(C)C5=CC=CC=C5)NC(=O)C(CC6CC6[N+](=O)[O-])NC(=O)C7=CC=C(N7O)Cl)C)C=CC
SMILES (Isomeric) CC[C@H](C)[C@H]1C(=O)N2C[C@H](C[C@H]2C(=O)O[C@@H]([C@H](C(=O)N[C@H](C(=O)N[C@@H](C(=O)N[C@H](C(=O)N1)CC3=CC=CC=C3)C[C@@H]4C[C@H]4[N+](=O)[O-])[C@H](C)C5=CC=CC=C5)NC(=O)[C@H](C[C@H]6C[C@@H]6[N+](=O)[O-])NC(=O)C7=CC=C(N7O)Cl)C)/C=C\C
InChI InChI=1S/C54H67ClN10O14/c1-6-14-32-22-42-54(73)79-30(5)46(61-49(68)38(24-35-26-41(35)65(77)78)57-50(69)39-19-20-43(55)63(39)74)52(71)60-45(29(4)33-17-12-9-13-18-33)51(70)58-37(23-34-25-40(34)64(75)76)47(66)56-36(21-31-15-10-8-11-16-31)48(67)59-44(28(3)7-2)53(72)62(42)27-32/h6,8-20,28-30,32,34-38,40-42,44-46,74H,7,21-27H2,1-5H3,(H,56,66)(H,57,69)(H,58,70)(H,59,67)(H,60,71)(H,61,68)/b14-6-/t28-,29+,30+,32-,34+,35-,36-,37+,38-,40+,41-,42-,44-,45-,46+/m0/s1
InChI Key CCONVECKWRPBMJ-ARSFXBAVSA-N
Popularity 14 references in papers

Physical and Chemical Properties

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Molecular Formula C54H67ClN10O14
Molecular Weight 1115.60 g/mol
Exact Mass 1114.4526745 g/mol
Topological Polar Surface Area (TPSA) 338.00 Ų
XlogP 6.80

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Hormaomycin C

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL221 P23219 Cyclooxygenase-1 99.82% 90.17%
CHEMBL2581 P07339 Cathepsin D 99.71% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.76% 96.09%
CHEMBL3837 P07711 Cathepsin L 95.94% 96.61%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 95.51% 94.45%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 94.38% 97.14%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 93.65% 97.64%
CHEMBL4072 P07858 Cathepsin B 93.39% 93.67%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 92.03% 95.56%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 91.08% 95.00%
CHEMBL3401 O75469 Pregnane X receptor 90.28% 94.73%
CHEMBL1293249 Q13887 Kruppel-like factor 5 89.50% 86.33%
CHEMBL3060 Q9Y345 Glycine transporter 2 89.18% 99.17%
CHEMBL4578 Q14680 Maternal embryonic leucine zipper kinase 89.01% 81.58%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 88.80% 98.33%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 88.75% 93.03%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 88.19% 93.00%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 88.17% 100.00%
CHEMBL3359 P21462 Formyl peptide receptor 1 87.62% 93.56%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 86.18% 95.89%
CHEMBL1163125 O60885 Bromodomain-containing protein 4 86.08% 97.31%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 85.70% 96.47%
CHEMBL5939 Q9NZ08 Endoplasmic reticulum aminopeptidase 1 85.36% 100.00%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 85.12% 92.88%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 84.86% 95.50%
CHEMBL3137262 O60341 LSD1/CoREST complex 84.33% 97.09%
CHEMBL4523377 Q86WV6 Stimulator of interferon genes protein 83.75% 95.48%
CHEMBL340 P08684 Cytochrome P450 3A4 83.02% 91.19%
CHEMBL2413 P32246 C-C chemokine receptor type 1 82.48% 89.50%
CHEMBL5608 Q16288 NT-3 growth factor receptor 82.29% 95.89%
CHEMBL4016 P42262 Glutamate receptor ionotropic, AMPA 2 82.10% 86.92%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 81.54% 91.11%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 81.42% 96.90%
CHEMBL5103 Q969S8 Histone deacetylase 10 80.87% 90.08%
CHEMBL1937 Q92769 Histone deacetylase 2 80.29% 94.75%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139585326
LOTUS LTS0196602
wikiData Q77420203