Herbicolin B

Details

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Internal ID e0bfe20a-2c2e-4b8a-a17c-3e19cec79dea
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name N-[(Z)-1-[[12-(3-amino-3-oxopropyl)-3-[3-(diaminomethylideneamino)propyl]-6,21-bis(1-hydroxyethyl)-7,25-dimethyl-18-(2-methylpropyl)-2,5,8,11,14,17,20,23-octaoxo-1-oxa-4,7,10,13,16,19,22-heptazacyclopentacos-24-yl]amino]-1-oxobut-2-en-2-yl]-3-hydroxytetradecanamide
SMILES (Canonical) CCCCCCCCCCCC(CC(=O)NC(=CC)C(=O)NC1C(OC(=O)C(NC(=O)C(N(C(=O)CNC(=O)C(NC(=O)CNC(=O)C(NC(=O)C(NC1=O)C(C)O)CC(C)C)CCC(=O)N)C)C(C)O)CCCN=C(N)N)C)O
SMILES (Isomeric) CCCCCCCCCCCC(CC(=O)N/C(=C\C)/C(=O)NC1C(OC(=O)C(NC(=O)C(N(C(=O)CNC(=O)C(NC(=O)CNC(=O)C(NC(=O)C(NC1=O)C(C)O)CC(C)C)CCC(=O)N)C)C(C)O)CCCN=C(N)N)C)O
InChI InChI=1S/C52H91N13O15/c1-9-11-12-13-14-15-16-17-18-20-33(68)26-39(70)59-34(10-2)47(75)64-43-32(7)80-51(79)36(21-19-24-56-52(54)55)61-50(78)44(31(6)67)65(8)41(72)28-58-45(73)35(22-23-38(53)69)60-40(71)27-57-46(74)37(25-29(3)4)62-48(76)42(30(5)66)63-49(43)77/h10,29-33,35-37,42-44,66-68H,9,11-28H2,1-8H3,(H2,53,69)(H,57,74)(H,58,73)(H,59,70)(H,60,71)(H,61,78)(H,62,76)(H,63,77)(H,64,75)(H4,54,55,56)/b34-10-
InChI Key YFNLBROYERMWJP-FWBDCHAOSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C52H91N13O15
Molecular Weight 1138.40 g/mol
Exact Mass 1137.67575925 g/mol
Topological Polar Surface Area (TPSA) 448.00 Ų
XlogP 1.20

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Herbicolin B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL4040 P28482 MAP kinase ERK2 99.73% 83.82%
CHEMBL2581 P07339 Cathepsin D 99.51% 98.95%
CHEMBL3837 P07711 Cathepsin L 99.41% 96.61%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.51% 96.09%
CHEMBL230 P35354 Cyclooxygenase-2 98.00% 89.63%
CHEMBL4588 P22894 Matrix metalloproteinase 8 97.85% 94.66%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 96.45% 91.11%
CHEMBL3060 Q9Y345 Glycine transporter 2 96.44% 99.17%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 95.43% 96.47%
CHEMBL2094135 Q96BI3 Gamma-secretase 93.13% 98.05%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 92.92% 93.10%
CHEMBL255 P29275 Adenosine A2b receptor 92.69% 98.59%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 92.56% 96.90%
CHEMBL299 P17252 Protein kinase C alpha 92.50% 98.03%
CHEMBL3892 Q99500 Sphingosine 1-phosphate receptor Edg-3 91.97% 97.29%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 91.58% 90.71%
CHEMBL4462 Q8IXJ6 NAD-dependent deacetylase sirtuin 2 91.39% 90.24%
CHEMBL4071 P08311 Cathepsin G 91.24% 94.64%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 90.86% 96.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 90.74% 94.45%
CHEMBL3359 P21462 Formyl peptide receptor 1 90.49% 93.56%
CHEMBL2096618 P11274 Bcr/Abl fusion protein 89.99% 85.83%
CHEMBL4227 P25090 Lipoxin A4 receptor 89.86% 100.00%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 89.74% 95.50%
CHEMBL2955 O95136 Sphingosine 1-phosphate receptor Edg-5 89.64% 92.86%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 89.31% 100.00%
CHEMBL236 P41143 Delta opioid receptor 89.13% 99.35%
CHEMBL253 P34972 Cannabinoid CB2 receptor 88.73% 97.25%
CHEMBL1806 P11388 DNA topoisomerase II alpha 88.46% 89.00%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 88.44% 99.23%
CHEMBL4072 P07858 Cathepsin B 88.33% 93.67%
CHEMBL333 P08253 Matrix metalloproteinase-2 87.78% 96.31%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 86.98% 97.64%
CHEMBL3137262 O60341 LSD1/CoREST complex 86.48% 97.09%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 86.39% 91.81%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 86.25% 95.00%
CHEMBL4769 O95749 Geranylgeranyl pyrophosphate synthetase 86.23% 92.08%
CHEMBL2514 O95665 Neurotensin receptor 2 85.90% 100.00%
CHEMBL5103 Q969S8 Histone deacetylase 10 85.77% 90.08%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 85.61% 92.88%
CHEMBL321 P14780 Matrix metalloproteinase 9 85.54% 92.12%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 84.99% 95.56%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 84.84% 88.42%
CHEMBL3145 P42338 PI3-kinase p110-beta subunit 84.19% 98.75%
CHEMBL2413 P32246 C-C chemokine receptor type 1 82.70% 89.50%
CHEMBL3401 O75469 Pregnane X receptor 82.55% 94.73%
CHEMBL2996 Q05655 Protein kinase C delta 82.26% 97.79%
CHEMBL3038469 P24941 CDK2/Cyclin A 80.65% 91.38%
CHEMBL332 P03956 Matrix metalloproteinase-1 80.57% 94.50%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 80.32% 93.00%
CHEMBL1907602 P06493 Cyclin-dependent kinase 1/cyclin B1 80.26% 91.24%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 6443862
LOTUS LTS0080378
wikiData Q105347692