Hapalosin

Details

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Internal ID 1d82450a-8885-4a32-a56f-0703f11d8f38
Taxonomy Phenylpropanoids and polyketides > Macrolide lactams
IUPAC Name (2S,5S,6R,10R,11S)-5-benzyl-10-heptyl-6-hydroxy-4,11-dimethyl-2-propan-2-yl-1,9-dioxa-4-azacyclododecane-3,8,12-trione
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C28H43NO6/c1-6-7-8-9-13-16-24-20(4)28(33)35-26(19(2)3)27(32)29(5)22(23(30)18-25(31)34-24)17-21-14-11-10-12-15-21/h10-12,14-15,19-20,22-24,26,30H,6-9,13,16-18H2,1-5H3/t20-,22-,23+,24+,26-/m0/s1
InChI Key NJNAHFYVTBZQHU-LFFUDGMSSA-N
Popularity 18 references in papers

Physical and Chemical Properties

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Molecular Formula C28H43NO6
Molecular Weight 489.60 g/mol
Exact Mass 489.30903809 g/mol
Topological Polar Surface Area (TPSA) 93.10 Ų
XlogP 6.00

Synonyms

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159542-04-8
(2S,5S,6R,10R,11S)-5-benzyl-10-heptyl-6-hydroxy-4,11-dimethyl-2-propan-2-yl-1,9-dioxa-4-azacyclododecane-3,8,12-trione
CHEMBL269137
BDBM50403688
1,9-Dioxa-4-azacyclododecane-3,8,12-trione, 10-heptyl-6-hydroxy-4,11-dimethyl-2-(1-methylethyl)-5-(phenylmethyl)-, (2S-(2R*,5R*,6S*,10S*,11R*))-

2D Structure

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2D Structure of Hapalosin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.74% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.41% 96.09%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.59% 95.56%
CHEMBL221 P23219 Cyclooxygenase-1 93.84% 90.17%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 90.51% 85.14%
CHEMBL253 P34972 Cannabinoid CB2 receptor 90.28% 97.25%
CHEMBL2265 P23141 Acyl coenzyme A:cholesterol acyltransferase 89.00% 85.94%
CHEMBL3359 P21462 Formyl peptide receptor 1 88.97% 93.56%
CHEMBL4769 O95749 Geranylgeranyl pyrophosphate synthetase 86.39% 92.08%
CHEMBL1951 P21397 Monoamine oxidase A 86.21% 91.49%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 85.18% 90.71%
CHEMBL1293249 Q13887 Kruppel-like factor 5 84.20% 86.33%
CHEMBL3401 O75469 Pregnane X receptor 83.47% 94.73%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 83.33% 97.64%
CHEMBL3060 Q9Y345 Glycine transporter 2 83.16% 99.17%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 82.99% 100.00%
CHEMBL5103 Q969S8 Histone deacetylase 10 82.08% 90.08%
CHEMBL5608 Q16288 NT-3 growth factor receptor 81.69% 95.89%
CHEMBL3891 P07384 Calpain 1 81.02% 93.04%
CHEMBL3892 Q99500 Sphingosine 1-phosphate receptor Edg-3 80.99% 97.29%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 80.60% 95.89%
CHEMBL3004 P33527 Multidrug resistance-associated protein 1 80.25% 96.37%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 133055
LOTUS LTS0225334
wikiData Q83035888