hapalindole H

Details

Top
Internal ID e564be1a-108d-4ea2-bd7a-78fd76a14931
IUPAC Name (2R,3R,4R,7R)-4-ethenyl-3-isocyano-4,8,8-trimethyl-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(15),9(16),10,12-tetraene
SMILES (Canonical) CC1(C2CCC(C(C2C3=CNC4=CC=CC1=C43)[N+]#[C-])(C)C=C)C
SMILES (Isomeric) C[C@@]1(CC[C@@H]2[C@@H]([C@H]1[N+]#[C-])C3=CNC4=CC=CC(=C43)C2(C)C)C=C
InChI InChI=1S/C21H24N2/c1-6-21(4)11-10-15-18(19(21)22-5)13-12-23-16-9-7-8-14(17(13)16)20(15,2)3/h6-9,12,15,18-19,23H,1,10-11H2,2-4H3/t15-,18+,19-,21+/m1/s1
InChI Key SLUFHMQYBPOTFZ-LKRGOLFISA-N
Popularity 4 references in papers

Physical and Chemical Properties

Top
Molecular Formula C21H24N2
Molecular Weight 304.40 g/mol
Exact Mass 304.193948774 g/mol
Topological Polar Surface Area (TPSA) 20.20 Ų
XlogP 5.10

Synonyms

Top
101968-75-6
CHEBI:140440
(2R,3R,4R,7R)-4-ethenyl-3-isocyano-4,8,8-trimethyl-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(15),9(16),10,12-tetraene
(6aR,9R,10R,10aR)-9-ethenyl-10-isocyano-6,6,9-trimethyl-2,2a,6,6a,7,8,9,10,10a,10c-decahydronaphtho[1,2,3-cd]indole
(2R,3R,4R,7R)-4-ethenyl-3-isocyano-4,8,8-trimethyl-14-azatetracyclo(7.6.1.02,7.013,16)hexadeca-1(15),9(16),10,12-tetraene
(6aR,9R,10R,10aR)-9-ethenyl-10-isocyano-6,6,9-trimethyl-2,2a,6,6a,7,8,9,10,10a,10c-decahydronaphtho(1,2,3-cd)indole
RefChem:145220
(6aR,9R,10R,10aR)-10-isocyano-6,6,9-trimethyl-9-vinyl-2,6,6a,7,8,9,10,10a-octahydronaphtho[1,2,3-cd]indole
MLS004797563
CHEMBL562103
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

Top
2D Structure of hapalindole H

3D Structure

Top

ADMET Properties (via admetSAR 2)

Top
Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

Top

Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 97.33% 94.45%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 96.50% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 96.28% 96.09%
CHEMBL4224 P49759 Dual specificty protein kinase CLK1 94.69% 85.30%
CHEMBL2095226 P05556 Integrin alpha-5/beta-1 92.53% 96.39%
CHEMBL1994 P08235 Mineralocorticoid receptor 91.72% 100.00%
CHEMBL4225 P49760 Dual specificity protein kinase CLK2 91.71% 80.96%
CHEMBL3137262 O60341 LSD1/CoREST complex 90.98% 97.09%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 90.63% 95.56%
CHEMBL3310 Q96DB2 Histone deacetylase 11 88.61% 88.56%
CHEMBL5608 Q16288 NT-3 growth factor receptor 88.17% 95.89%
CHEMBL253 P34972 Cannabinoid CB2 receptor 85.82% 97.25%
CHEMBL4145 Q9UKV0 Histone deacetylase 9 85.81% 85.49%
CHEMBL1902 P62942 FK506-binding protein 1A 85.57% 97.05%
CHEMBL3192 Q9BY41 Histone deacetylase 8 84.04% 93.99%
CHEMBL2716 Q8WUI4 Histone deacetylase 7 83.37% 89.44%
CHEMBL3492 P49721 Proteasome Macropain subunit 83.29% 90.24%
CHEMBL1937 Q92769 Histone deacetylase 2 81.98% 94.75%
CHEMBL2581 P07339 Cathepsin D 80.94% 98.95%
CHEMBL5028 O14672 ADAM10 80.84% 97.50%
CHEMBL1806 P11388 DNA topoisomerase II alpha 80.32% 89.00%

Plants that contains it

Top
Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

Top
PubChem 21671525
LOTUS LTS0203221
wikiData Q74410841