H-DL-Pyr-DL-xiIle-DL-Pro-DL-Trp-DL-Phe-DL-His-DL-Arg-NH2

Details

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Internal ID 30ba2a4e-643a-4513-bc19-5e8d3a981af9
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides
IUPAC Name N-[1-[2-[[1-[[1-[[1-[[1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxopentan-2-yl]-5-oxopyrrolidine-2-carboxamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C48H64N14O8/c1-3-27(2)40(61-42(65)34-17-18-39(63)56-34)47(70)62-20-10-16-38(62)46(69)60-36(22-29-24-54-32-14-8-7-13-31(29)32)44(67)58-35(21-28-11-5-4-6-12-28)43(66)59-37(23-30-25-52-26-55-30)45(68)57-33(41(49)64)15-9-19-53-48(50)51/h4-8,11-14,24-27,33-38,40,54H,3,9-10,15-23H2,1-2H3,(H2,49,64)(H,52,55)(H,56,63)(H,57,68)(H,58,67)(H,59,66)(H,60,69)(H,61,65)(H4,50,51,53)
InChI Key BSBFUZUALMLLAA-UHFFFAOYSA-N
Popularity 0 references in papers

Physical and Chemical Properties

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Molecular Formula C48H64N14O8
Molecular Weight 965.10 g/mol
Exact Mass 964.50315506 g/mol
Topological Polar Surface Area (TPSA) 347.00 Ų
XlogP 0.60

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of H-DL-Pyr-DL-xiIle-DL-Pro-DL-Trp-DL-Phe-DL-His-DL-Arg-NH2

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 99.90% 97.64%
CHEMBL2581 P07339 Cathepsin D 99.88% 98.95%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 99.56% 91.81%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 99.48% 98.33%
CHEMBL3837 P07711 Cathepsin L 99.40% 96.61%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.34% 96.09%
CHEMBL4644 P41968 Melanocortin receptor 3 98.63% 99.52%
CHEMBL259 P32245 Melanocortin receptor 4 98.08% 95.38%
CHEMBL3310 Q96DB2 Histone deacetylase 11 97.95% 88.56%
CHEMBL333 P08253 Matrix metalloproteinase-2 97.72% 96.31%
CHEMBL230 P35354 Cyclooxygenase-2 97.29% 89.63%
CHEMBL4588 P22894 Matrix metalloproteinase 8 97.11% 94.66%
CHEMBL1255126 O15151 Protein Mdm4 96.87% 90.20%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 96.46% 95.56%
CHEMBL2514 O95665 Neurotensin receptor 2 95.83% 100.00%
CHEMBL4361 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 95.73% 95.52%
CHEMBL4123 P30989 Neurotensin receptor 1 95.57% 96.67%
CHEMBL5939 Q9NZ08 Endoplasmic reticulum aminopeptidase 1 95.28% 100.00%
CHEMBL261 P00915 Carbonic anhydrase I 95.05% 96.76%
CHEMBL5608 Q16288 NT-3 growth factor receptor 94.84% 95.89%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 94.72% 91.11%
CHEMBL255 P29275 Adenosine A2b receptor 94.57% 98.59%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 94.20% 94.45%
CHEMBL2535 P11166 Glucose transporter 94.08% 98.75%
CHEMBL4393 P39900 Matrix metalloproteinase 12 93.65% 92.22%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 93.60% 88.42%
CHEMBL4979 P13866 Sodium/glucose cotransporter 1 93.34% 98.24%
CHEMBL5103 Q969S8 Histone deacetylase 10 93.24% 90.08%
CHEMBL3137262 O60341 LSD1/CoREST complex 91.26% 97.09%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 91.24% 99.23%
CHEMBL3202 P48147 Prolyl endopeptidase 90.82% 90.65%
CHEMBL5028 O14672 ADAM10 90.72% 97.50%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 88.49% 97.23%
CHEMBL1744525 P43490 Nicotinamide phosphoribosyltransferase 88.30% 96.25%
CHEMBL1907591 P30926 Neuronal acetylcholine receptor; alpha4/beta4 87.26% 100.00%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 87.00% 95.00%
CHEMBL213 P08588 Beta-1 adrenergic receptor 86.93% 95.56%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 86.77% 93.03%
CHEMBL4777 P25929 Neuropeptide Y receptor type 1 86.73% 96.67%
CHEMBL4462 Q8IXJ6 NAD-dependent deacetylase sirtuin 2 86.03% 90.24%
CHEMBL2327 P21452 Neurokinin 2 receptor 85.96% 98.89%
CHEMBL3060 Q9Y345 Glycine transporter 2 85.91% 99.17%
CHEMBL321 P14780 Matrix metalloproteinase 9 85.48% 92.12%
CHEMBL3192 Q9BY41 Histone deacetylase 8 85.24% 93.99%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 85.17% 90.71%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 84.29% 96.47%
CHEMBL221 P23219 Cyclooxygenase-1 83.74% 90.17%
CHEMBL3729 P22748 Carbonic anhydrase IV 82.97% 99.23%
CHEMBL5203 P33316 dUTP pyrophosphatase 82.91% 99.18%
CHEMBL4227 P25090 Lipoxin A4 receptor 82.85% 100.00%
CHEMBL4073 P09237 Matrix metalloproteinase 7 82.52% 97.56%
CHEMBL204 P00734 Thrombin 81.35% 96.01%
CHEMBL4608 P33032 Melanocortin receptor 5 81.00% 97.00%
CHEMBL3880 P07900 Heat shock protein HSP 90-alpha 80.55% 96.21%
CHEMBL1944495 P28065 Proteasome subunit beta type-9 80.47% 97.50%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 80.45% 96.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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Cross-Links

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PubChem 163044468
LOTUS LTS0183201
wikiData Q104945145