H-bAla(2-OH,3-pentyl)-DL-Val-DL-N(Me)xiIle-DL-N(Me)Tyr-DL-Tyr-OH

Details

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Internal ID 1806a996-73d6-41ba-ae88-169a6a11f7b4
Taxonomy Organic acids and derivatives > Peptidomimetics > Hybrid peptides
IUPAC Name 2-[[2-[[2-[[2-[(3-amino-2-hydroxyoctanoyl)amino]-3-methylbutanoyl]-methylamino]-3-methylpentanoyl]-methylamino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoic acid
SMILES (Canonical) CCCCCC(C(C(=O)NC(C(C)C)C(=O)N(C)C(C(C)CC)C(=O)N(C)C(CC1=CC=C(C=C1)O)C(=O)NC(CC2=CC=C(C=C2)O)C(=O)O)O)N
SMILES (Isomeric) CCCCCC(C(C(=O)NC(C(C)C)C(=O)N(C)C(C(C)CC)C(=O)N(C)C(CC1=CC=C(C=C1)O)C(=O)NC(CC2=CC=C(C=C2)O)C(=O)O)O)N
InChI InChI=1S/C39H59N5O9/c1-8-10-11-12-29(40)34(47)36(49)42-32(23(3)4)37(50)44(7)33(24(5)9-2)38(51)43(6)31(22-26-15-19-28(46)20-16-26)35(48)41-30(39(52)53)21-25-13-17-27(45)18-14-25/h13-20,23-24,29-34,45-47H,8-12,21-22,40H2,1-7H3,(H,41,48)(H,42,49)(H,52,53)
InChI Key LMTZMDMYSIVNCR-UHFFFAOYSA-N
Popularity 0 references in papers

Physical and Chemical Properties

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Molecular Formula C39H59N5O9
Molecular Weight 741.90 g/mol
Exact Mass 741.43127848 g/mol
Topological Polar Surface Area (TPSA) 223.00 Ų
XlogP 2.50

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of H-bAla(2-OH,3-pentyl)-DL-Val-DL-N(Me)xiIle-DL-N(Me)Tyr-DL-Tyr-OH

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.89% 98.95%
CHEMBL3060 Q9Y345 Glycine transporter 2 98.40% 99.17%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.43% 96.09%
CHEMBL2514 O95665 Neurotensin receptor 2 96.55% 100.00%
CHEMBL3837 P07711 Cathepsin L 96.30% 96.61%
CHEMBL3359 P21462 Formyl peptide receptor 1 95.62% 93.56%
CHEMBL4040 P28482 MAP kinase ERK2 95.49% 83.82%
CHEMBL1255126 O15151 Protein Mdm4 94.16% 90.20%
CHEMBL4072 P07858 Cathepsin B 93.42% 93.67%
CHEMBL3892 Q99500 Sphingosine 1-phosphate receptor Edg-3 92.67% 97.29%
CHEMBL1907591 P30926 Neuronal acetylcholine receptor; alpha4/beta4 91.82% 100.00%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 90.46% 95.56%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 90.26% 90.71%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 88.17% 100.00%
CHEMBL4227 P25090 Lipoxin A4 receptor 88.14% 100.00%
CHEMBL236 P41143 Delta opioid receptor 87.80% 99.35%
CHEMBL3004 P33527 Multidrug resistance-associated protein 1 87.62% 96.37%
CHEMBL268 P43235 Cathepsin K 86.91% 96.85%
CHEMBL3401 O75469 Pregnane X receptor 86.31% 94.73%
CHEMBL2955 O95136 Sphingosine 1-phosphate receptor Edg-5 86.11% 92.86%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 86.01% 95.89%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 85.77% 94.45%
CHEMBL3976 Q9UHL4 Dipeptidyl peptidase II 85.41% 92.29%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 85.29% 95.50%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 84.52% 93.00%
CHEMBL3308 P55212 Caspase-6 82.50% 97.56%
CHEMBL3891 P07384 Calpain 1 82.39% 93.04%
CHEMBL2345 P51812 Ribosomal protein S6 kinase alpha 3 82.04% 95.64%
CHEMBL1907 P15144 Aminopeptidase N 80.30% 93.31%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 80.13% 93.10%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 73837482
LOTUS LTS0075951
wikiData Q104171106