Fabclavine Ib

Details

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Internal ID fe27e8d5-0be8-40a2-9db9-a34609a2ba82
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Cyclic peptides
IUPAC Name 2-amino-4-[[(2S)-1-[[6-(2-amino-2-oxoethyl)-3-[2-[1-hydroxy-3-oxo-3-[(11,19,27,35-tetraamino-3-hydroxyhexatriacontyl)amino]propyl]pyrrolidine-1-carbonyl]-2-methyl-5,8,11-trioxo-1,4,7-triazacycloundec-9-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-4-oxobutanoic acid
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C68H121N13O12/c1-46(69)27-16-7-3-8-19-30-49(70)31-20-9-4-10-21-32-50(71)33-22-11-5-12-23-34-51(72)35-24-13-6-14-25-36-52(82)38-39-75-60(85)45-58(83)57-37-26-40-81(57)67(91)63-47(2)76-62(87)44-56(65(89)78-55(43-59(74)84)66(90)80-63)79-64(88)54(41-48-28-17-15-18-29-48)77-61(86)42-53(73)68(92)93/h15,17-18,28-29,46-47,49-58,63,82-83H,3-14,16,19-27,30-45,69-73H2,1-2H3,(H2,74,84)(H,75,85)(H,76,87)(H,77,86)(H,78,89)(H,79,88)(H,80,90)(H,92,93)/t46?,47?,49?,50?,51?,52?,53?,54-,55?,56?,57?,58?,63?/m0/s1
InChI Key IZSKWNSKICNTCU-KBXWAUECSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C68H121N13O12
Molecular Weight 1312.80 g/mol
Exact Mass 1311.92576635 g/mol
Topological Polar Surface Area (TPSA) 446.00 Ų
XlogP 1.90

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Fabclavine Ib

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.96% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.41% 96.09%
CHEMBL4040 P28482 MAP kinase ERK2 99.17% 83.82%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 97.57% 98.33%
CHEMBL236 P41143 Delta opioid receptor 96.81% 99.35%
CHEMBL4801 P29466 Caspase-1 96.54% 96.85%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 95.97% 96.47%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 95.91% 91.11%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 95.86% 97.64%
CHEMBL233 P35372 Mu opioid receptor 95.16% 97.93%
CHEMBL4979 P13866 Sodium/glucose cotransporter 1 94.71% 98.24%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 94.69% 94.45%
CHEMBL221 P23219 Cyclooxygenase-1 93.91% 90.17%
CHEMBL3837 P07711 Cathepsin L 93.90% 96.61%
CHEMBL5103 Q969S8 Histone deacetylase 10 93.72% 90.08%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 93.59% 95.00%
CHEMBL4588 P22894 Matrix metalloproteinase 8 93.12% 94.66%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 92.31% 88.42%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 91.88% 90.71%
CHEMBL3060 Q9Y345 Glycine transporter 2 91.61% 99.17%
CHEMBL3137262 O60341 LSD1/CoREST complex 91.57% 97.09%
CHEMBL2514 O95665 Neurotensin receptor 2 91.44% 100.00%
CHEMBL1744525 P43490 Nicotinamide phosphoribosyltransferase 91.02% 96.25%
CHEMBL2327 P21452 Neurokinin 2 receptor 90.63% 98.89%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 90.51% 97.23%
CHEMBL1255126 O15151 Protein Mdm4 90.35% 90.20%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 89.86% 97.14%
CHEMBL5608 Q16288 NT-3 growth factor receptor 88.55% 95.89%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 88.45% 95.56%
CHEMBL3359 P21462 Formyl peptide receptor 1 88.24% 93.56%
CHEMBL5028 O14672 ADAM10 88.10% 97.50%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 88.09% 93.00%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 87.59% 93.03%
CHEMBL3976 Q9UHL4 Dipeptidyl peptidase II 87.34% 92.29%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 86.36% 82.69%
CHEMBL4227 P25090 Lipoxin A4 receptor 83.92% 100.00%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 82.96% 95.89%
CHEMBL340 P08684 Cytochrome P450 3A4 82.73% 91.19%
CHEMBL1806 P11388 DNA topoisomerase II alpha 81.81% 89.00%
CHEMBL4302 P08183 P-glycoprotein 1 80.36% 92.98%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 145720648
LOTUS LTS0150460
wikiData Q105123442