Epothilone E

Details

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Internal ID b1c4f8ce-5a31-40e6-973f-24a638f1fa59
Taxonomy Phenylpropanoids and polyketides > Macrolides and analogues > Epothilones and analogues
IUPAC Name (1S,3S,7S,10R,11S,12S,16R)-7,11-dihydroxy-3-[(E)-1-[2-(hydroxymethyl)-1,3-thiazol-4-yl]prop-1-en-2-yl]-8,8,10,12-tetramethyl-4,17-dioxabicyclo[14.1.0]heptadecane-5,9-dione
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C26H39NO7S/c1-14-7-6-8-18-20(33-18)10-19(15(2)9-17-13-35-22(12-28)27-17)34-23(30)11-21(29)26(4,5)25(32)16(3)24(14)31/h9,13-14,16,18-21,24,28-29,31H,6-8,10-12H2,1-5H3/b15-9+/t14-,16+,18+,19-,20-,21-,24-/m0/s1
InChI Key FCCNKYGSMOSYPV-OKOHHBBGSA-N
Popularity 7 references in papers

Physical and Chemical Properties

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Molecular Formula C26H39NO7S
Molecular Weight 509.70 g/mol
Exact Mass 509.24472376 g/mol
Topological Polar Surface Area (TPSA) 158.00 Ų
XlogP 2.80

Synonyms

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201049-37-8
(-)-Epothilone E
UK5H6YZZ8A
(1S,3S,7S,10R,11S,12S,16R)-7,11-dihydroxy-3-[(E)-1-[2-(hydroxymethyl)-1,3-thiazol-4-yl]prop-1-en-2-yl]-8,8,10,12-tetramethyl-4,17-dioxabicyclo[14.1.0]heptadecane-5,9-dione
(1S,3S,7S,10R,11S,12S,16R)-7,11-Dihydroxy-3-((1E)-2-(2-(hydroxymethyl)-4-thiazolyl)-1-methylethenyl)-8,8,10,12-tetramethyl-4,17-dioxabicyclo(14.1.0)heptadecane-5,9-dione
4,17-Dioxabicyclo(14.1.0)heptadecane-5,9-dione, 7,11-dihydroxy-3-((1E)-2-(2-(hydroxymethyl)-4-thiazolyl)-1-methylethenyl)-8,8,10,12-tetramethyl-, (1S,3S,7S,10R,11S,12S,16R)-
Epothilon E
UNII-UK5H6YZZ8A
SCHEMBL4126
CHEMBL470478
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

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2D Structure of Epothilone E

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.33% 96.09%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 94.91% 85.14%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 93.65% 99.23%
CHEMBL1293249 Q13887 Kruppel-like factor 5 92.33% 86.33%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 90.94% 91.11%
CHEMBL2581 P07339 Cathepsin D 90.66% 98.95%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 90.60% 95.56%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 86.56% 94.45%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 85.98% 93.00%
CHEMBL241 Q14432 Phosphodiesterase 3A 84.63% 92.94%
CHEMBL1994 P08235 Mineralocorticoid receptor 83.79% 100.00%
CHEMBL2095226 P05556 Integrin alpha-5/beta-1 82.75% 96.39%
CHEMBL3401 O75469 Pregnane X receptor 81.93% 94.73%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 81.88% 96.90%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 81.74% 93.10%
CHEMBL1293294 P51151 Ras-related protein Rab-9A 80.82% 87.67%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 9806341
LOTUS LTS0212888
wikiData Q75052974