Disporoside A

Details

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Internal ID 1c12f8b6-0fba-41a3-b719-df8b534568e1
Taxonomy Lipids and lipid-like molecules > Steroids and steroid derivatives > Steroidal glycosides > Steroidal saponins
IUPAC Name (2R,3R,4S,5S,6R)-2-[[(2R,3S,4S,5R,6R)-3,4-dihydroxy-6-[(1R,2S,4S,5'R,6R,7S,8R,9S,12S,13S,16S,18R)-5',7,9,13-tetramethylspiro[5-oxapentacyclo[10.8.0.02,9.04,8.013,18]icosane-6,2'-oxane]-16-yl]oxy-5-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]methoxy]-6-(hydroxymethyl)oxane-3,4,5-triol
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C45H74O18/c1-19-7-12-45(57-17-19)20(2)30-26(63-45)14-25-23-6-5-21-13-22(8-10-43(21,3)24(23)9-11-44(25,30)4)58-42-39(62-41-38(55)35(52)32(49)28(16-47)60-41)36(53)33(50)29(61-42)18-56-40-37(54)34(51)31(48)27(15-46)59-40/h19-42,46-55H,5-18H2,1-4H3/t19-,20+,21-,22+,23-,24+,25+,26+,27-,28-,29-,30+,31-,32-,33-,34+,35+,36+,37-,38-,39-,40-,41+,42-,43+,44+,45-/m1/s1
InChI Key UTXFFSIHMAHBLN-YGNOLRTQSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C45H74O18
Molecular Weight 903.10 g/mol
Exact Mass 902.48751551 g/mol
Topological Polar Surface Area (TPSA) 276.00 Ų
XlogP 1.20

Synonyms

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(2R,3R,4S,5S,6R)-2-(((2R,3S,4S,5R,6R)-3,4-dihydroxy-6-((1R,2S,4S,5'R,6R,7S,8R,9S,12S,13S,16S,18R)-5',7,9,13-tetramethylspiro(5-oxapentacyclo(10.8.0.02,9.04,8.013,18)icosane-6,2'-oxane)-16-yl)oxy-5-((2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl)oxyoxan-2-yl)methoxy)-6-(hydroxymethyl)oxane-3,4,5-triol
(2R,3R,4S,5S,6R)-2-[[(2R,3S,4S,5R,6R)-3,4-dihydroxy-6-[(1R,2S,4S,5'R,6R,7S,8R,9S,12S,13S,16S,18R)-5',7,9,13-tetramethylspiro[5-oxapentacyclo[10.8.0.02,9.04,8.013,18]icosane-6,2'-oxane]-16-yl]oxy-5-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]methoxy]-6-(hydroxymethyl)oxane-3,4,5-triol
RefChem:135116
770721-94-3
CHEMBL505982
SCHEMBL31345829

2D Structure

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2D Structure of Disporoside A

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.10% 96.09%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.03% 91.11%
CHEMBL3137262 O60341 LSD1/CoREST complex 96.17% 97.09%
CHEMBL233 P35372 Mu opioid receptor 94.63% 97.93%
CHEMBL237 P41145 Kappa opioid receptor 93.52% 98.10%
CHEMBL218 P21554 Cannabinoid CB1 receptor 93.03% 96.61%
CHEMBL253 P34972 Cannabinoid CB2 receptor 92.69% 97.25%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 92.12% 95.50%
CHEMBL4681 P42330 Aldo-keto-reductase family 1 member C3 91.95% 89.05%
CHEMBL1994 P08235 Mineralocorticoid receptor 91.69% 100.00%
CHEMBL226 P30542 Adenosine A1 receptor 91.21% 95.93%
CHEMBL5255 O00206 Toll-like receptor 4 90.48% 92.50%
CHEMBL3880 P07900 Heat shock protein HSP 90-alpha 90.13% 96.21%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 89.80% 94.45%
CHEMBL2955 O95136 Sphingosine 1-phosphate receptor Edg-5 89.17% 92.86%
CHEMBL4618 P09960 Leukotriene A4 hydrolase 87.29% 97.86%
CHEMBL4793 Q86TI2 Dipeptidyl peptidase IX 86.75% 96.95%
CHEMBL6136 O60341 Lysine-specific histone demethylase 1 86.20% 95.58%
CHEMBL241 Q14432 Phosphodiesterase 3A 85.04% 92.94%
CHEMBL3430907 Q96GD4 Aurora kinase B/Inner centromere protein 84.76% 97.50%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 84.64% 100.00%
CHEMBL5608 Q16288 NT-3 growth factor receptor 83.70% 95.89%
CHEMBL4303 P08238 Heat shock protein HSP 90-beta 83.60% 96.77%
CHEMBL5888 Q99558 Mitogen-activated protein kinase kinase kinase 14 83.33% 100.00%
CHEMBL1871 P10275 Androgen Receptor 83.16% 96.43%
CHEMBL2996 Q05655 Protein kinase C delta 83.00% 97.79%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 82.91% 95.89%
CHEMBL1806 P11388 DNA topoisomerase II alpha 81.96% 89.00%
CHEMBL2072 P35499 Sodium channel protein type IV alpha subunit 81.67% 92.32%
CHEMBL4016 P42262 Glutamate receptor ionotropic, AMPA 2 81.62% 86.92%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 81.44% 93.10%
CHEMBL3351 Q13085 Acetyl-CoA carboxylase 1 80.89% 93.04%
CHEMBL1163125 O60885 Bromodomain-containing protein 4 80.85% 97.31%
CHEMBL2094128 P24941 Cyclin-dependent kinase 2/cyclin A 80.69% 97.25%
CHEMBL206 P03372 Estrogen receptor alpha 80.17% 97.64%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 80.00% 96.38%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Disporopsis pernyi
Smilax aristolochiifolia

Cross-Links

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PubChem 11600450
LOTUS LTS0073495
wikiData Q105279156