Disorazole H

Details

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Internal ID 1e05fb08-6953-4e60-9e79-7302962569da
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Dicarboxylic acids and derivatives
IUPAC Name (12E,14Z,24Z,26Z)-4,22-bis[(E)-3-hydroxy-2-methylhex-4-en-2-yl]-30-methoxy-3,7,10,17,21,33-hexaoxa-35,36-diazapentacyclo[30.2.1.116,19.06,8.09,11]hexatriaconta-1(34),12,14,16(36),18,24,26,28,32(35)-nonaene-2,20-dione
SMILES (Canonical) CC=CC(C(C)(C)C1CC=CC=CC=CC(CC2=NC(=CO2)C(=O)OC(CC3C(O3)C4C(O4)C=CC=CC5=NC(=CO5)C(=O)O1)C(C)(C)C(C=CC)O)OC)O
SMILES (Isomeric) C/C=C/C(C(C)(C)C1C/C=C\C=C/C=CC(CC2=NC(=CO2)C(=O)OC(CC3C(O3)C4C(O4)/C=C/C=C\C5=NC(=CO5)C(=O)O1)C(C)(C)C(/C=C/C)O)OC)O
InChI InChI=1S/C43H54N2O11/c1-8-17-32(46)42(3,4)34-21-14-12-10-11-13-19-27(50-7)23-37-45-29(26-52-37)41(49)56-35(43(5,6)33(47)18-9-2)24-31-39(54-31)38-30(53-38)20-15-16-22-36-44-28(25-51-36)40(48)55-34/h8-20,22,25-27,30-35,38-39,46-47H,21,23-24H2,1-7H3/b11-10-,14-12-,17-8+,18-9+,19-13?,20-15+,22-16-
InChI Key QBKIVBASHDDBID-CLXWHGGYSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C43H54N2O11
Molecular Weight 774.90 g/mol
Exact Mass 774.37276054 g/mol
Topological Polar Surface Area (TPSA) 179.00 Ų
XlogP 7.50

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Disorazole H

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL1293249 Q13887 Kruppel-like factor 5 95.60% 86.33%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 95.02% 94.45%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 94.96% 85.14%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 93.59% 91.11%
CHEMBL3401 O75469 Pregnane X receptor 92.26% 94.73%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 91.60% 96.09%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 89.23% 94.00%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 88.92% 95.56%
CHEMBL253 P34972 Cannabinoid CB2 receptor 87.16% 97.25%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 87.06% 100.00%
CHEMBL2373 P21730 C5a anaphylatoxin chemotactic receptor 86.79% 92.62%
CHEMBL3060 Q9Y345 Glycine transporter 2 86.63% 99.17%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 85.13% 97.33%
CHEMBL3137262 O60341 LSD1/CoREST complex 84.94% 97.09%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 84.17% 97.14%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 83.75% 93.03%
CHEMBL2581 P07339 Cathepsin D 82.76% 98.95%
CHEMBL4662 P28074 Proteasome Macropain subunit MB1 82.52% 93.85%
CHEMBL230 P35354 Cyclooxygenase-2 81.28% 89.63%
CHEMBL3976 Q9UHL4 Dipeptidyl peptidase II 80.99% 92.29%
CHEMBL2094135 Q96BI3 Gamma-secretase 80.96% 98.05%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 80.79% 99.23%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139586839
LOTUS LTS0177988
wikiData Q77515683