L-Tyrosine, N-(1-(N-(4-((3-hydroxy-4-((N-(N-(1-(2-hydroxy-1-oxopropyl)-L-prolyl)-N-methyl-L-leucyl)-L-threonyl)amino)-6-methyl-1-oxoheptyl)oxy)-2,5-dimethyl-1,3-dioxohexyl)-L-leucyl)-L-prolyl)-N,O-dimethyl-, phi-lactone

Details

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Internal ID 1e38d177-744d-497b-966d-4e873f2c8c06
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name N-[1-[[13-butan-2-yl-12-hydroxy-20-[(4-methoxyphenyl)methyl]-6,17,21-trimethyl-3-(2-methylpropyl)-2,5,7,10,15,19,22-heptaoxo-8-propan-2-yl-9,18-dioxa-1,4,14,21-tetrazabicyclo[21.3.0]hexacosan-16-yl]amino]-4-methyl-1-oxopentan-2-yl]-1-(2-hydroxypropanoyl)-N-methylpyrrolidine-2-carboxamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C57H89N7O15/c1-15-33(8)46-44(66)29-45(67)79-49(32(6)7)48(68)34(9)50(69)58-39(26-30(2)3)54(73)64-25-17-19-41(64)56(75)62(13)43(28-37-20-22-38(77-14)23-21-37)57(76)78-36(11)47(52(71)59-46)60-51(70)42(27-31(4)5)61(12)55(74)40-18-16-24-63(40)53(72)35(10)65/h20-23,30-36,39-44,46-47,49,65-66H,15-19,24-29H2,1-14H3,(H,58,69)(H,59,71)(H,60,70)
InChI Key KYHUYMLIVQFXRI-UHFFFAOYSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C57H89N7O15
Molecular Weight 1112.40 g/mol
Exact Mass 1111.64166516 g/mol
Topological Polar Surface Area (TPSA) 288.00 Ų
XlogP 5.50

Synonyms

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C57H89N7O15
Neuro_000164
KYHUYMLIVQFXRI-UHFFFAOYSA-N
CDA32705
MFCD01677226
N-[1-[[13-butan-2-yl-12-hydroxy-20-[(4-methoxyphenyl)methyl]-6,17,21-trimethyl-3-(2-methylpropyl)-2,5,7,10,15,19,22-heptaoxo-8-propan-2-yl-9,18-dioxa-1,4,14,21-tetrazabicyclo[21.3.0]hexacosan-16-yl]amino]-4-methyl-1-oxopentan-2-yl]-1-(2-hydroxypropanoyl)-N-methylpyrrolidine-2-carboxamide
L-Tyrosine,5-dimethyl-1,3-dioxohexyl]-L-leucyl]-1-prolyl]-N,O-dimethyl-, .phi.-lactone
L-Tyrosine, N-(1-(N-(4-((3-hydroxy-4-((N-(N-(1-(2-hydroxy-1-oxopropyl) -L-propyl)-N-methyl-L-leucyl)-L-threonyl)amino)-6-methyl-1- oxoheptyl)oxy)-2,5-dimethyl-1,3-dioxohexyl)-L-leucyl)-1- prolyl)-N,O-dimethyl-, phi-lactone
N-[1-(([10-Sec-butyl-11-hydroxy-20-isobutyl-15-isopropyl-3-(4-methoxybenzyl)-2,6,17-trimethyl-1,4,8,13,16,18,21-heptaoxodocosahydro-15H-pyrrolo[2,1-f][1,15,4,7,10,20]dioxatetraazacyclotricosin-7-yl]am #
N-[1-[[12-hydroxy-3-isobutyl-8-isopropyl-20-[(4-methoxyphenyl)methyl]-6,17,21-trimethyl-2,5,7,10,15,19,22-heptaoxo-13-sec-butyl-9,18-dioxa-1,4,14,21-tetrazabicyclo[21.3.0]hexacosan-16-yl]carbamoyl]-3-methyl-butyl]-1-(2-hydroxypropanoyl)-N-methyl-pyrrolidine-2-carboxamide

2D Structure

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2D Structure of L-Tyrosine, N-(1-(N-(4-((3-hydroxy-4-((N-(N-(1-(2-hydroxy-1-oxopropyl)-L-prolyl)-N-methyl-L-leucyl)-L-threonyl)amino)-6-methyl-1-oxoheptyl)oxy)-2,5-dimethyl-1,3-dioxohexyl)-L-leucyl)-L-prolyl)-N,O-dimethyl-, phi-lactone

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.90% 98.95%
CHEMBL3837 P07711 Cathepsin L 99.87% 96.61%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.64% 96.09%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 98.69% 85.14%
CHEMBL333 P08253 Matrix metalloproteinase-2 96.95% 96.31%
CHEMBL332 P03956 Matrix metalloproteinase-1 96.94% 94.50%
CHEMBL221 P23219 Cyclooxygenase-1 95.32% 90.17%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 94.54% 95.56%
CHEMBL4208 P20618 Proteasome component C5 94.51% 90.00%
CHEMBL253 P34972 Cannabinoid CB2 receptor 94.34% 97.25%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 94.32% 97.14%
CHEMBL5608 Q16288 NT-3 growth factor receptor 93.97% 95.89%
CHEMBL321 P14780 Matrix metalloproteinase 9 93.57% 92.12%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 93.45% 82.38%
CHEMBL4588 P22894 Matrix metalloproteinase 8 92.97% 94.66%
CHEMBL5103 Q969S8 Histone deacetylase 10 92.75% 90.08%
CHEMBL3060 Q9Y345 Glycine transporter 2 92.15% 99.17%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 91.21% 93.00%
CHEMBL3137262 O60341 LSD1/CoREST complex 91.09% 97.09%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 89.99% 90.71%
CHEMBL340 P08684 Cytochrome P450 3A4 89.97% 91.19%
CHEMBL283 P08254 Matrix metalloproteinase 3 89.88% 97.29%
CHEMBL3492 P49721 Proteasome Macropain subunit 89.82% 90.24%
CHEMBL3359 P21462 Formyl peptide receptor 1 89.77% 93.56%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 89.42% 97.64%
CHEMBL4073 P09237 Matrix metalloproteinase 7 88.96% 97.56%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 88.88% 95.89%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 87.87% 95.00%
CHEMBL1902 P62942 FK506-binding protein 1A 87.59% 97.05%
CHEMBL261 P00915 Carbonic anhydrase I 87.00% 96.76%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 85.87% 92.88%
CHEMBL2443 P49862 Kallikrein 7 85.68% 94.00%
CHEMBL205 P00918 Carbonic anhydrase II 85.51% 98.44%
CHEMBL2514 O95665 Neurotensin receptor 2 85.48% 100.00%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 85.25% 94.00%
CHEMBL235 P37231 Peroxisome proliferator-activated receptor gamma 85.09% 95.39%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 84.90% 100.00%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 84.77% 98.33%
CHEMBL4051 P13569 Cystic fibrosis transmembrane conductance regulator 84.75% 95.71%
CHEMBL4618 P09960 Leukotriene A4 hydrolase 84.47% 97.86%
CHEMBL5203 P33316 dUTP pyrophosphatase 84.43% 99.18%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 83.92% 94.45%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 83.80% 91.11%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 83.70% 94.33%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 83.09% 96.00%
CHEMBL6175 Q9H3R0 Lysine-specific demethylase 4C 82.90% 96.69%
CHEMBL3691 Q13822 Autotaxin 82.84% 96.39%
CHEMBL255 P29275 Adenosine A2b receptor 82.42% 98.59%
CHEMBL3430907 Q96GD4 Aurora kinase B/Inner centromere protein 81.92% 97.50%
CHEMBL1075317 P61964 WD repeat-containing protein 5 81.61% 96.33%
CHEMBL2535 P11166 Glucose transporter 81.36% 98.75%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 80.84% 96.90%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 80.58% 96.38%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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Cross-Links

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PubChem 550898
LOTUS LTS0054973
wikiData Q105147733