Destruxin-E diol

Details

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Internal ID 58cdb912-c49e-4c04-9b8d-75db9a456eac
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name 16-butan-2-yl-3-(2,3-dihydroxypropyl)-10,11,14-trimethyl-13-propan-2-yl-4-oxa-1,8,11,14,17-pentazabicyclo[17.3.0]docosane-2,5,9,12,15,18-hexone
SMILES (Canonical) CCC(C)C1C(=O)N(C(C(=O)N(C(C(=O)NCCC(=O)OC(C(=O)N2CCCC2C(=O)N1)CC(CO)O)C)C)C(C)C)C
SMILES (Isomeric) CCC(C)C1C(=O)N(C(C(=O)N(C(C(=O)NCCC(=O)OC(C(=O)N2CCCC2C(=O)N1)CC(CO)O)C)C)C(C)C)C
InChI InChI=1S/C29H49N5O9/c1-8-17(4)23-28(41)33(7)24(16(2)3)29(42)32(6)18(5)25(38)30-12-11-22(37)43-21(14-19(36)15-35)27(40)34-13-9-10-20(34)26(39)31-23/h16-21,23-24,35-36H,8-15H2,1-7H3,(H,30,38)(H,31,39)
InChI Key DJYDCIUMNXZSBH-UHFFFAOYSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C29H49N5O9
Molecular Weight 611.70 g/mol
Exact Mass 611.35302816 g/mol
Topological Polar Surface Area (TPSA) 186.00 Ų
XlogP 0.20

Synonyms

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AKOS040739497
NCGC00381220-02
NCGC00381220-01!16-butan-2-yl-3-(2,3-dihydroxypropyl)-10,11,14-trimethyl-13-propan-2-yl-4-oxa-1,8,11,14,17-pentazabicyclo[17.3.0]docosane-2,5,9,12,15,18-hexone

2D Structure

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2D Structure of Destruxin-E diol

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.25% 98.95%
CHEMBL253 P34972 Cannabinoid CB2 receptor 98.72% 97.25%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.67% 96.09%
CHEMBL5103 Q969S8 Histone deacetylase 10 96.69% 90.08%
CHEMBL4588 P22894 Matrix metalloproteinase 8 95.50% 94.66%
CHEMBL333 P08253 Matrix metalloproteinase-2 94.48% 96.31%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 94.39% 85.14%
CHEMBL3137262 O60341 LSD1/CoREST complex 93.58% 97.09%
CHEMBL5608 Q16288 NT-3 growth factor receptor 90.57% 95.89%
CHEMBL1902 P62942 FK506-binding protein 1A 90.02% 97.05%
CHEMBL332 P03956 Matrix metalloproteinase-1 89.35% 94.50%
CHEMBL2189110 Q15910 Histone-lysine N-methyltransferase EZH2 88.39% 97.50%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 87.91% 90.71%
CHEMBL1937 Q92769 Histone deacetylase 2 87.79% 94.75%
CHEMBL3524 P56524 Histone deacetylase 4 87.44% 92.97%
CHEMBL4616 Q92847 Ghrelin receptor 87.29% 92.00%
CHEMBL255 P29275 Adenosine A2b receptor 87.19% 98.59%
CHEMBL228 P31645 Serotonin transporter 86.22% 95.51%
CHEMBL3837 P07711 Cathepsin L 85.68% 96.61%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 85.40% 82.38%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 85.38% 93.00%
CHEMBL1806 P11388 DNA topoisomerase II alpha 85.23% 89.00%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 84.71% 95.56%
CHEMBL217 P14416 Dopamine D2 receptor 84.11% 95.62%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 83.95% 95.00%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 83.64% 91.11%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 83.21% 96.47%
CHEMBL3691 Q13822 Autotaxin 83.19% 96.39%
CHEMBL3310 Q96DB2 Histone deacetylase 11 82.90% 88.56%
CHEMBL4005 P42336 PI3-kinase p110-alpha subunit 82.65% 97.47%
CHEMBL5203 P33316 dUTP pyrophosphatase 81.80% 99.18%
CHEMBL325 Q13547 Histone deacetylase 1 81.73% 95.92%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 81.48% 100.00%
CHEMBL299 P17252 Protein kinase C alpha 81.31% 98.03%
CHEMBL5469 Q14289 Protein tyrosine kinase 2 beta 81.27% 91.03%
CHEMBL3359 P21462 Formyl peptide receptor 1 81.09% 93.56%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 81.01% 94.45%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 81.00% 95.50%
CHEMBL2443 P49862 Kallikrein 7 80.92% 94.00%
CHEMBL2781 P19634 Sodium/hydrogen exchanger 1 80.69% 90.24%
CHEMBL1293249 Q13887 Kruppel-like factor 5 80.64% 86.33%
CHEMBL1994 P08235 Mineralocorticoid receptor 80.55% 100.00%
CHEMBL321 P14780 Matrix metalloproteinase 9 80.49% 92.12%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 80.46% 99.23%
CHEMBL1949 P62937 Cyclophilin A 80.46% 98.57%
CHEMBL4208 P20618 Proteasome component C5 80.36% 90.00%
CHEMBL2996 Q05655 Protein kinase C delta 80.13% 97.79%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 3804245
LOTUS LTS0069492
wikiData Q103818455