Destruxin B

Details

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Internal ID 0b644b1b-d6a0-4529-8704-17c17f8223f9
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name 16-butan-2-yl-10,11,14-trimethyl-3-(2-methylpropyl)-13-propan-2-yl-4-oxa-1,8,11,14,17-pentazabicyclo[17.3.0]docosane-2,5,9,12,15,18-hexone
SMILES (Canonical) CCC(C)C1C(=O)N(C(C(=O)N(C(C(=O)NCCC(=O)OC(C(=O)N2CCCC2C(=O)N1)CC(C)C)C)C)C(C)C)C
SMILES (Isomeric) CCC(C)C1C(=O)N(C(C(=O)N(C(C(=O)NCCC(=O)OC(C(=O)N2CCCC2C(=O)N1)CC(C)C)C)C)C(C)C)C
InChI InChI=1S/C30H51N5O7/c1-10-19(6)24-29(40)34(9)25(18(4)5)30(41)33(8)20(7)26(37)31-14-13-23(36)42-22(16-17(2)3)28(39)35-15-11-12-21(35)27(38)32-24/h17-22,24-25H,10-16H2,1-9H3,(H,31,37)(H,32,38)
InChI Key GNBHVMBELHWUIF-UHFFFAOYSA-N
Popularity 50 references in papers

Physical and Chemical Properties

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Molecular Formula C30H51N5O7
Molecular Weight 593.80 g/mol
Exact Mass 593.37884898 g/mol
Topological Polar Surface Area (TPSA) 145.00 Ų
XlogP 2.80

Synonyms

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UNII-7R6CR62KFE
NSC236580
MEGxm0_000393
.beta.-Alanine, .rho.-lactone
CHEMBL1736621
SCHEMBL22163465
ACon1_002320
DTXSID10947891
CHEBI:181259
NCGC00169957-01
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

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2D Structure of Destruxin B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.13% 98.95%
CHEMBL253 P34972 Cannabinoid CB2 receptor 98.55% 97.25%
CHEMBL333 P08253 Matrix metalloproteinase-2 98.22% 96.31%
CHEMBL5103 Q969S8 Histone deacetylase 10 97.09% 90.08%
CHEMBL4588 P22894 Matrix metalloproteinase 8 96.94% 94.66%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 96.40% 96.09%
CHEMBL3837 P07711 Cathepsin L 95.90% 96.61%
CHEMBL332 P03956 Matrix metalloproteinase-1 95.85% 94.50%
CHEMBL255 P29275 Adenosine A2b receptor 93.63% 98.59%
CHEMBL1902 P62942 FK506-binding protein 1A 93.53% 97.05%
CHEMBL3137262 O60341 LSD1/CoREST complex 93.41% 97.09%
CHEMBL4616 Q92847 Ghrelin receptor 90.96% 92.00%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 90.88% 82.38%
CHEMBL3524 P56524 Histone deacetylase 4 90.49% 92.97%
CHEMBL5203 P33316 dUTP pyrophosphatase 90.40% 99.18%
CHEMBL2996 Q05655 Protein kinase C delta 90.16% 97.79%
CHEMBL226 P30542 Adenosine A1 receptor 90.10% 95.93%
CHEMBL2189110 Q15910 Histone-lysine N-methyltransferase EZH2 90.01% 97.50%
CHEMBL321 P14780 Matrix metalloproteinase 9 90.00% 92.12%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 89.32% 90.71%
CHEMBL228 P31645 Serotonin transporter 89.25% 95.51%
CHEMBL5608 Q16288 NT-3 growth factor receptor 89.19% 95.89%
CHEMBL1937 Q92769 Histone deacetylase 2 87.55% 94.75%
CHEMBL325 Q13547 Histone deacetylase 1 87.26% 95.92%
CHEMBL217 P14416 Dopamine D2 receptor 86.40% 95.62%
CHEMBL3691 Q13822 Autotaxin 85.78% 96.39%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 85.13% 95.56%
CHEMBL4072 P07858 Cathepsin B 85.08% 93.67%
CHEMBL2781 P19634 Sodium/hydrogen exchanger 1 84.92% 90.24%
CHEMBL3310 Q96DB2 Histone deacetylase 11 84.58% 88.56%
CHEMBL4835 P00338 L-lactate dehydrogenase A chain 84.53% 95.34%
CHEMBL299 P17252 Protein kinase C alpha 84.23% 98.03%
CHEMBL1949 P62937 Cyclophilin A 83.83% 98.57%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 83.45% 93.00%
CHEMBL2443 P49862 Kallikrein 7 82.71% 94.00%
CHEMBL1806 P11388 DNA topoisomerase II alpha 82.59% 89.00%
CHEMBL5697 Q9GZT9 Egl nine homolog 1 82.33% 93.40%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 82.27% 96.47%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 81.38% 98.33%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 81.07% 90.93%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 80.61% 99.23%
CHEMBL3359 P21462 Formyl peptide receptor 1 80.61% 93.56%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 80.44% 96.38%
CHEMBL4005 P42336 PI3-kinase p110-alpha subunit 80.28% 97.47%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 80.25% 97.64%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 428373
LOTUS LTS0079247
wikiData Q105012275