Desmethylisaridin C2

Details

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Internal ID 9cb9c746-c062-436f-b93c-b7282708760b
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name (3S,10S,13S,16S,19S,20S)-16-benzyl-11,20-dimethyl-3-(2-methylpropyl)-10,13-di(propan-2-yl)-4-oxa-1,8,11,14,17-pentazabicyclo[17.3.0]docosane-2,5,9,12,15,18-hexone
SMILES (Canonical) CC1CCN2C1C(=O)NC(C(=O)NC(C(=O)N(C(C(=O)NCCC(=O)OC(C2=O)CC(C)C)C(C)C)C)C(C)C)CC3=CC=CC=C3
SMILES (Isomeric) C[C@H]1CCN2[C@@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N([C@H](C(=O)NCCC(=O)O[C@H](C2=O)CC(C)C)C(C)C)C)C(C)C)CC3=CC=CC=C3
InChI InChI=1S/C35H53N5O7/c1-20(2)18-26-34(45)40-17-15-23(7)30(40)33(44)37-25(19-24-12-10-9-11-13-24)31(42)38-28(21(3)4)35(46)39(8)29(22(5)6)32(43)36-16-14-27(41)47-26/h9-13,20-23,25-26,28-30H,14-19H2,1-8H3,(H,36,43)(H,37,44)(H,38,42)/t23-,25-,26-,28-,29-,30-/m0/s1
InChI Key YCGVVPXVWFYGHR-QUODLWGASA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C35H53N5O7
Molecular Weight 655.80 g/mol
Exact Mass 655.39449905 g/mol
Topological Polar Surface Area (TPSA) 154.00 Ų
XlogP 4.30

Synonyms

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CHEMBL2407690

2D Structure

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2D Structure of Desmethylisaridin C2

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.73% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.37% 96.09%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.31% 95.56%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 93.90% 97.64%
CHEMBL3837 P07711 Cathepsin L 92.47% 96.61%
CHEMBL228 P31645 Serotonin transporter 91.56% 95.51%
CHEMBL333 P08253 Matrix metalloproteinase-2 90.63% 96.31%
CHEMBL5103 Q969S8 Histone deacetylase 10 88.99% 90.08%
CHEMBL253 P34972 Cannabinoid CB2 receptor 88.89% 97.25%
CHEMBL4588 P22894 Matrix metalloproteinase 8 87.91% 94.66%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 87.85% 91.11%
CHEMBL5608 Q16288 NT-3 growth factor receptor 87.53% 95.89%
CHEMBL226 P30542 Adenosine A1 receptor 87.48% 95.93%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 87.08% 97.14%
CHEMBL1293249 Q13887 Kruppel-like factor 5 86.82% 86.33%
CHEMBL4616 Q92847 Ghrelin receptor 86.05% 92.00%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 85.65% 90.93%
CHEMBL3137262 O60341 LSD1/CoREST complex 85.41% 97.09%
CHEMBL4072 P07858 Cathepsin B 84.49% 93.67%
CHEMBL255 P29275 Adenosine A2b receptor 84.42% 98.59%
CHEMBL1949 P62937 Cyclophilin A 84.38% 98.57%
CHEMBL5805 Q9NR97 Toll-like receptor 8 82.95% 96.25%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 82.85% 96.47%
CHEMBL2189110 Q15910 Histone-lysine N-methyltransferase EZH2 82.65% 97.50%
CHEMBL3359 P21462 Formyl peptide receptor 1 80.96% 93.56%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 80.41% 90.71%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 80.25% 95.89%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 80.18% 93.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 71745527
LOTUS LTS0124612
wikiData Q77567522