Cyclosporin E

Details

Top
Internal ID ff6d6ce9-420f-4cbb-b2b3-ab8a798f91b3
Taxonomy Organic acids and derivatives > Peptidomimetics > Peptoid-peptide hybrids > Cyclosporins
IUPAC Name (3S,6R,9S,12S,15S,18S,24S,27S,30S,33S)-24-ethyl-27-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,6,9,13,19,22,28-octamethyl-3,12,18,33-tetrakis(2-methylpropyl)-15,30-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undecone
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C61H109N11O12/c1-24-26-27-39(15)51(74)50-56(79)64-42(25-2)58(81)67(18)32-47(73)68(19)43(28-33(3)4)54(77)65-48(37(11)12)60(83)70(21)44(29-34(5)6)53(76)62-40(16)52(75)63-41(17)57(80)71(22)46(31-36(9)10)59(82)69(20)45(30-35(7)8)55(78)66-49(38(13)14)61(84)72(50)23/h24,26,33-46,48-51,74H,25,27-32H2,1-23H3,(H,62,76)(H,63,75)(H,64,79)(H,65,77)(H,66,78)/b26-24+/t39-,40+,41-,42+,43+,44+,45+,46+,48+,49+,50+,51-/m1/s1
InChI Key SYXYUKMELXLDBD-WKHWYDSQSA-N
Popularity 4 references in papers

Physical and Chemical Properties

Top
Molecular Formula C61H109N11O12
Molecular Weight 1188.60 g/mol
Exact Mass 1187.82571795 g/mol
Topological Polar Surface Area (TPSA) 288.00 Ų
XlogP 7.30

Synonyms

Top
63798-73-2
Cyclosporin A, 5-L-valine-
Cyclosporin E, (-)-
UNII-26496N541O
26496N541O
Cyclo(L-alanyl-D-alanyl-N-methyl-L-leucyl-N-methyl-L-leucyl-L-valyl-(3R,4R,6E)-6,7-didehydro-3-hydroxy-N,4-dimethyl-L-2-aminooctanoyl-L-2-aminobutanoyl-N-methylglycyl-N-methyl-L-leucyl-L-valyl-N-methyl-L-leucyl
DTXSID10904565
(3S,6R,9S,12S,15S,18S,24S,27S,30S,33S)-24-ethyl-27-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,6,9,13,19,22,28-octamethyl-3,12,18,33-tetrakis(2-methylpropyl)-15,30-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undecone
(3S,6R,9S,12S,15S,18S,24S,27S,30S,33S)-24-ethyl-27-((E,1R,2R)-1-hydroxy-2-methylhex-4-enyl)-1,4,6,9,13,19,22,28-octamethyl-3,12,18,33-tetrakis(2-methylpropyl)-15,30-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undecone
RefChem:129980
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

Top
2D Structure of Cyclosporin E

3D Structure

Top

ADMET Properties (via admetSAR 2)

Top
Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

Top

Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL1949 P62937 Cyclophilin A 99.46% 98.57%
CHEMBL2581 P07339 Cathepsin D 98.46% 98.95%
CHEMBL253 P34972 Cannabinoid CB2 receptor 98.06% 97.25%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.31% 96.09%
CHEMBL321 P14780 Matrix metalloproteinase 9 91.31% 92.12%
CHEMBL1937 Q92769 Histone deacetylase 2 91.25% 94.75%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 90.40% 95.56%
CHEMBL5103 Q969S8 Histone deacetylase 10 90.32% 90.08%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 89.42% 85.14%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 88.94% 90.71%
CHEMBL218 P21554 Cannabinoid CB1 receptor 88.47% 96.61%
CHEMBL3137262 O60341 LSD1/CoREST complex 88.34% 97.09%
CHEMBL333 P08253 Matrix metalloproteinase-2 86.05% 96.31%
CHEMBL3267 P48736 PI3-kinase p110-gamma subunit 85.45% 95.71%
CHEMBL255 P29275 Adenosine A2b receptor 85.01% 98.59%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 84.01% 90.93%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 83.32% 99.23%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 83.10% 96.47%
CHEMBL1806 P11388 DNA topoisomerase II alpha 82.33% 89.00%
CHEMBL226 P30542 Adenosine A1 receptor 82.14% 95.93%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 82.01% 91.11%
CHEMBL4208 P20618 Proteasome component C5 81.21% 90.00%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 81.10% 94.45%
CHEMBL4588 P22894 Matrix metalloproteinase 8 80.07% 94.66%
CHEMBL2413 P32246 C-C chemokine receptor type 1 80.06% 89.50%

Plants that contains it

Top
Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

Top
PubChem 90478790
LOTUS LTS0078963
wikiData Q27254040