Cyanopeptolin CP978

Details

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Internal ID 1596c01a-e480-440c-8473-66e69de153aa
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name 4-[[15-(5-amino-5-iminopentyl)-2-benzyl-21-hydroxy-5-[(4-hydroxyphenyl)methyl]-4,11-dimethyl-3,6,9,13,16,22-hexaoxo-8-propan-2-yl-10-oxa-1,4,7,14,17-pentazabicyclo[16.3.1]docosan-12-yl]amino]-3-(butanoylamino)-4-oxobutanoic acid
SMILES (Canonical) CCCC(=O)NC(CC(=O)O)C(=O)NC1C(OC(=O)C(NC(=O)C(N(C(=O)C(N2C(CCC(C2=O)NC(=O)C(NC1=O)CCCCC(=N)N)O)CC3=CC=CC=C3)C)CC4=CC=C(C=C4)O)C(C)C)C
SMILES (Isomeric) CCCC(=O)NC(CC(=O)O)C(=O)NC1C(OC(=O)C(NC(=O)C(N(C(=O)C(N2C(CCC(C2=O)NC(=O)C(NC1=O)CCCCC(=N)N)O)CC3=CC=CC=C3)C)CC4=CC=C(C=C4)O)C(C)C)C
InChI InChI=1S/C48H67N9O13/c1-6-12-37(59)51-33(25-39(61)62)43(64)55-41-27(4)70-48(69)40(26(2)3)54-44(65)34(23-29-17-19-30(58)20-18-29)56(5)47(68)35(24-28-13-8-7-9-14-28)57-38(60)22-21-32(46(57)67)53-42(63)31(52-45(41)66)15-10-11-16-36(49)50/h7-9,13-14,17-20,26-27,31-35,38,40-41,58,60H,6,10-12,15-16,21-25H2,1-5H3,(H3,49,50)(H,51,59)(H,52,66)(H,53,63)(H,54,65)(H,55,64)(H,61,62)
InChI Key URCPMPQTYGGFBQ-UHFFFAOYSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C48H67N9O13
Molecular Weight 978.10 g/mol
Exact Mass 977.48583323 g/mol
Topological Polar Surface Area (TPSA) 340.00 Ų
XlogP 1.50

Synonyms

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DTXSID101334071

2D Structure

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2D Structure of Cyanopeptolin CP978

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.94% 98.95%
CHEMBL4040 P28482 MAP kinase ERK2 99.65% 83.82%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.89% 96.09%
CHEMBL3060 Q9Y345 Glycine transporter 2 98.50% 99.17%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.95% 91.11%
CHEMBL221 P23219 Cyclooxygenase-1 96.78% 90.17%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.24% 95.56%
CHEMBL5103 Q969S8 Histone deacetylase 10 93.78% 90.08%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 92.81% 94.45%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 91.84% 95.89%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 90.71% 97.64%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 90.36% 93.00%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 89.71% 99.23%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 89.58% 90.93%
CHEMBL5608 Q16288 NT-3 growth factor receptor 89.48% 95.89%
CHEMBL3137262 O60341 LSD1/CoREST complex 89.25% 97.09%
CHEMBL1949 P62937 Cyclophilin A 88.94% 98.57%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 88.49% 97.14%
CHEMBL1806 P11388 DNA topoisomerase II alpha 88.42% 89.00%
CHEMBL3891 P07384 Calpain 1 86.80% 93.04%
CHEMBL4072 P07858 Cathepsin B 86.51% 93.67%
CHEMBL4769 O95749 Geranylgeranyl pyrophosphate synthetase 85.77% 92.08%
CHEMBL1293249 Q13887 Kruppel-like factor 5 85.36% 86.33%
CHEMBL3468 P55210 Caspase-7 84.76% 95.68%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 84.55% 90.71%
CHEMBL3776 Q14790 Caspase-8 84.46% 97.06%
CHEMBL3359 P21462 Formyl peptide receptor 1 83.88% 93.56%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 82.82% 97.33%
CHEMBL226 P30542 Adenosine A1 receptor 82.66% 95.93%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 82.32% 82.38%
CHEMBL340 P08684 Cytochrome P450 3A4 82.03% 91.19%
CHEMBL2413 P32246 C-C chemokine receptor type 1 81.58% 89.50%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 81.47% 96.47%
CHEMBL2535 P11166 Glucose transporter 81.42% 98.75%
CHEMBL4394 Q9NYA1 Sphingosine kinase 1 80.40% 96.03%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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Cross-Links

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PubChem 146682047
LOTUS LTS0128465
wikiData Q105277668