Cortistatin J

Details

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Internal ID d9aec44a-bfbb-4933-ad94-6720eb9168bd
Taxonomy Organoheterocyclic compounds > Isoquinolines and derivatives
IUPAC Name (1S,2R,5S,6R,14S,16R)-5-isoquinolin-7-yl-N,N,6-trimethyl-19-oxapentacyclo[14.2.1.01,9.02,6.011,16]nonadeca-8,10,12-trien-14-amine
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C30H34N2O/c1-28-12-10-24-17-23-6-7-25(32(2)3)18-29(23)13-14-30(24,33-29)27(28)9-8-26(28)21-5-4-20-11-15-31-19-22(20)16-21/h4-7,10-11,15-17,19,25-27H,8-9,12-14,18H2,1-3H3/t25-,26-,27-,28-,29-,30-/m1/s1
InChI Key FJXAOLJCOASQTL-VHNXJUCRSA-N
Popularity 9 references in papers

Physical and Chemical Properties

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Molecular Formula C30H34N2O
Molecular Weight 438.60 g/mol
Exact Mass 438.267113712 g/mol
Topological Polar Surface Area (TPSA) 25.40 Ų
XlogP 4.70

Synonyms

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Cortistatine J
(-)-Cortistatin J
F69CWM0JQX
944804-62-0
DTXSID901336421
(3S,3aR,9S,10aR,12aS,12bR)-1,2,3,3a,4,9,10,11,12,12b-Decahydro-3-(7-isoquinolinyl)-N,N,3a-trimethyl-10a,12a-epoxybenzo(4,5)cyclohept(1,2-E)inden-9-amine
10a,12a-Epoxybenzo(4,5)cyclohept(1,2-E)inden-9-amine, 1,2,3,3a,4,9,10,11,12,12b-decahydro-3-(7-isoquinolinyl)-N,N,3a-trimethyl-, (3S,3aR,9S,10aR,12aS,12bR)-
RefChem:128107
DTXCID201766617
(1S,2R,5S,6R,14S,16R)-5-isoquinolin-7-yl-N,N,6-trimethyl-19-oxapentacyclo(14.2.1.01,9.02,6.011,16)nonadeca-8,10,12-trien-14-amine
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

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2D Structure of Cortistatin J

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2039 P27338 Monoamine oxidase B 98.06% 92.51%
CHEMBL4145 Q9UKV0 Histone deacetylase 9 95.51% 85.49%
CHEMBL4224 P49759 Dual specificty protein kinase CLK1 94.22% 85.30%
CHEMBL1951 P21397 Monoamine oxidase A 93.95% 91.49%
CHEMBL3524 P56524 Histone deacetylase 4 93.18% 92.97%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 91.49% 96.09%
CHEMBL2553 Q15418 Ribosomal protein S6 kinase alpha 1 91.26% 85.11%
CHEMBL226 P30542 Adenosine A1 receptor 90.65% 95.93%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 90.65% 91.11%
CHEMBL3137262 O60341 LSD1/CoREST complex 90.58% 97.09%
CHEMBL5608 Q16288 NT-3 growth factor receptor 90.10% 95.89%
CHEMBL253 P34972 Cannabinoid CB2 receptor 89.71% 97.25%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 86.65% 94.45%
CHEMBL2716 Q8WUI4 Histone deacetylase 7 86.55% 89.44%
CHEMBL1293249 Q13887 Kruppel-like factor 5 86.46% 86.33%
CHEMBL1907601 P11802 Cyclin-dependent kinase 4/cyclin D1 85.67% 98.99%
CHEMBL2000 P03952 Plasma kallikrein 85.15% 93.92%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 84.62% 97.33%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 84.60% 100.00%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 84.35% 94.00%
CHEMBL4105838 Q96GG9 DCN1-like protein 1 84.04% 95.00%
CHEMBL2581 P07339 Cathepsin D 83.84% 98.95%
CHEMBL4225 P49760 Dual specificity protein kinase CLK2 83.43% 80.96%
CHEMBL6175 Q9H3R0 Lysine-specific demethylase 4C 82.31% 96.69%
CHEMBL3192 Q9BY41 Histone deacetylase 8 82.30% 93.99%
CHEMBL4158 P49327 Fatty acid synthase 81.99% 82.50%
CHEMBL344 Q99705 Melanin-concentrating hormone receptor 1 81.59% 92.50%
CHEMBL221 P23219 Cyclooxygenase-1 81.29% 90.17%
CHEMBL4444 P04070 Vitamin K-dependent protein C 81.22% 93.89%
CHEMBL1907599 P05556 Integrin alpha-4/beta-1 80.87% 92.86%
CHEMBL2378 P30307 Dual specificity phosphatase Cdc25C 80.72% 96.67%
CHEMBL2094127 P06493 Cyclin-dependent kinase 1/cyclin B 80.69% 96.00%
CHEMBL5103 Q969S8 Histone deacetylase 10 80.12% 90.08%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 16737543
LOTUS LTS0083901
wikiData Q27277712