Concanamycin E

Details

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Internal ID e51fe5ac-3890-4618-9a32-2e93d88facbf
Taxonomy Phenylpropanoids and polyketides > Macrolides and analogues
IUPAC Name [6-[2-[4-[(4E,6E,14E,16Z)-10,12-dihydroxy-3,17-dimethoxy-7,9,13,15-tetramethyl-18-oxo-1-oxacyclooctadeca-4,6,14,16-tetraen-2-yl]-3-hydroxypentan-2-yl]-2-hydroxy-5-methyl-6-[(E)-prop-1-enyl]oxan-4-yl]oxy-4-hydroxy-2-methyloxan-3-yl] carbamate
SMILES (Canonical) CC=CC1C(C(CC(O1)(C(C)C(C(C)C2C(C=CC=C(CC(C(CC(C(C=C(C=C(C(=O)O2)OC)C)C)O)O)C)C)OC)O)O)OC3CC(C(C(O3)C)OC(=O)N)O)C
SMILES (Isomeric) C/C=C/C1C(C(CC(O1)(C(C)C(C(C)C2C(/C=C/C=C(/CC(C(CC(C(/C=C(/C=C(/C(=O)O2)\OC)\C)C)O)O)C)\C)OC)O)O)OC3CC(C(C(O3)C)OC(=O)N)O)C
InChI InChI=1S/C44H71NO14/c1-12-14-34-27(6)37(56-38-21-33(48)41(30(9)55-38)58-43(45)51)22-44(52,59-34)29(8)39(49)28(7)40-35(53-10)16-13-15-23(2)17-25(4)31(46)20-32(47)26(5)18-24(3)19-36(54-11)42(50)57-40/h12-16,18-19,25-35,37-41,46-49,52H,17,20-22H2,1-11H3,(H2,45,51)/b14-12+,16-13+,23-15+,24-18+,36-19-
InChI Key NNJUTDASDBXCIX-KYPZQYTFSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C44H71NO14
Molecular Weight 838.00 g/mol
Exact Mass 837.48745594 g/mol
Topological Polar Surface Area (TPSA) 226.00 Ų
XlogP 5.20

Synonyms

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Concanamycin A, 8-deethyl-
SCHEMBL29884597

2D Structure

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2D Structure of Concanamycin E

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 99.80% 85.14%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.56% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.67% 96.09%
CHEMBL3137262 O60341 LSD1/CoREST complex 94.87% 97.09%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 93.43% 95.56%
CHEMBL3880 P07900 Heat shock protein HSP 90-alpha 92.53% 96.21%
CHEMBL1293249 Q13887 Kruppel-like factor 5 91.24% 86.33%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 89.19% 94.45%
CHEMBL5608 Q16288 NT-3 growth factor receptor 89.10% 95.89%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 88.76% 99.23%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 88.58% 97.14%
CHEMBL1806 P11388 DNA topoisomerase II alpha 88.05% 89.00%
CHEMBL2007 P16234 Platelet-derived growth factor receptor alpha 87.84% 91.07%
CHEMBL1902 P62942 FK506-binding protein 1A 86.99% 97.05%
CHEMBL253 P34972 Cannabinoid CB2 receptor 86.74% 97.25%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 86.57% 96.47%
CHEMBL5028 O14672 ADAM10 85.65% 97.50%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 84.99% 97.33%
CHEMBL4303 P08238 Heat shock protein HSP 90-beta 84.90% 96.77%
CHEMBL1163125 O60885 Bromodomain-containing protein 4 84.44% 97.31%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 83.88% 95.89%
CHEMBL3359 P21462 Formyl peptide receptor 1 83.83% 93.56%
CHEMBL2535 P11166 Glucose transporter 83.67% 98.75%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 83.60% 96.00%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 83.51% 95.50%
CHEMBL3714130 P46095 G-protein coupled receptor 6 82.86% 97.36%
CHEMBL3267 P48736 PI3-kinase p110-gamma subunit 82.86% 95.71%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 82.84% 100.00%
CHEMBL1293255 P15428 15-hydroxyprostaglandin dehydrogenase [NAD+] 82.60% 83.57%
CHEMBL2581 P07339 Cathepsin D 82.18% 98.95%
CHEMBL340 P08684 Cytochrome P450 3A4 81.96% 91.19%
CHEMBL4208 P20618 Proteasome component C5 81.42% 90.00%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 80.86% 93.00%
CHEMBL4793 Q86TI2 Dipeptidyl peptidase IX 80.62% 96.95%
CHEMBL4481 P35228 Nitric oxide synthase, inducible 80.62% 94.80%
CHEMBL4657 Q6V1X1 Dipeptidyl peptidase VIII 80.39% 97.21%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 6438773
LOTUS LTS0057026
wikiData Q105182178