Comazaphilone B

Details

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Internal ID 0ce1018a-6b62-432b-a5c3-861ddb5c760c
Taxonomy Organoheterocyclic compounds > Azaphilones
IUPAC Name [(6R,7R)-6-hydroxy-7-methyl-8-oxo-3-propyl-5,6-dihydro-1H-isochromen-7-yl] 3,4-dihydroxy-2-methoxy-6-methylbenzoate
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C22H26O8/c1-5-6-13-8-12-9-16(24)22(3,20(26)14(12)10-29-13)30-21(27)17-11(2)7-15(23)18(25)19(17)28-4/h7-8,16,23-25H,5-6,9-10H2,1-4H3/t16-,22-/m1/s1
InChI Key UIYAMSRXSZRILG-OPAMFIHVSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C22H26O8
Molecular Weight 418.40 g/mol
Exact Mass 418.16276778 g/mol
Topological Polar Surface Area (TPSA) 123.00 Ų
XlogP 2.20

Synonyms

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CHEBI:70011
CHEMBL1689196
Q27138352
(6R,7R)-6-Hydroxy-7-methyl-8-oxo-3-propyl-5,6,7,8-tetrahydro-1H-isochromen-7-yl 3,4-dihydroxy-2-methoxy-6-methylbenzoate
[(6R,7R)-6-hydroxy-7-methyl-8-oxo-3-propyl-5,6-dihydro-1H-isochromen-7-yl] 3,4-dihydroxy-2-methoxy-6-methyl-benzoate
rel-(6R,7R)-6-hydroxy-7-methyl-8-oxo-3-propyl-5,6,7,8-tetrahydro-1H-isochromen-7-yl 3,4-dihydroxy-2-methoxy-6-methylbenzoate

2D Structure

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2D Structure of Comazaphilone B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.44% 91.11%
CHEMBL1293249 Q13887 Kruppel-like factor 5 97.13% 86.33%
CHEMBL2581 P07339 Cathepsin D 96.08% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 95.45% 96.09%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 94.77% 85.14%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 94.36% 94.45%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 90.96% 94.00%
CHEMBL215 P09917 Arachidonate 5-lipoxygenase 90.43% 92.68%
CHEMBL1806 P11388 DNA topoisomerase II alpha 89.95% 89.00%
CHEMBL4793 Q86TI2 Dipeptidyl peptidase IX 88.63% 96.95%
CHEMBL4657 Q6V1X1 Dipeptidyl peptidase VIII 88.43% 97.21%
CHEMBL3401 O75469 Pregnane X receptor 87.93% 94.73%
CHEMBL4208 P20618 Proteasome component C5 87.40% 90.00%
CHEMBL226 P30542 Adenosine A1 receptor 87.25% 95.93%
CHEMBL241 Q14432 Phosphodiesterase 3A 87.10% 92.94%
CHEMBL1994 P08235 Mineralocorticoid receptor 86.84% 100.00%
CHEMBL1871 P10275 Androgen Receptor 86.18% 96.43%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 85.88% 82.38%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 85.46% 90.71%
CHEMBL2781 P19634 Sodium/hydrogen exchanger 1 85.40% 90.24%
CHEMBL3137262 O60341 LSD1/CoREST complex 85.14% 97.09%
CHEMBL2007 P16234 Platelet-derived growth factor receptor alpha 83.50% 91.07%
CHEMBL3922 P50579 Methionine aminopeptidase 2 83.04% 97.28%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 82.03% 94.33%
CHEMBL255 P29275 Adenosine A2b receptor 81.39% 98.59%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 80.98% 95.56%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 80.35% 99.23%
CHEMBL2345 P51812 Ribosomal protein S6 kinase alpha 3 80.27% 95.64%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 51041530
LOTUS LTS0082763
wikiData Q27138352