Chlorajapolide B, (rel)-

Details

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Internal ID 19eddc34-b0fb-4182-a9f8-20e7098fb777
Taxonomy Lipids and lipid-like molecules > Prenol lipids > Terpene lactones > Sesquiterpene lactones > Eudesmanolides, secoeudesmanolides, and derivatives
IUPAC Name (1S,2R,4S,6S,8R,13S)-6-hydroxy-1,10-dimethyl-7,12-dioxapentacyclo[6.6.1.02,4.05,15.09,13]pentadeca-5(15),9-dien-11-one
SMILES (Canonical) CC1=C2C(CC3(C4CC4C5=C3C2OC5O)C)OC1=O
SMILES (Isomeric) CC1=C2[C@H](C[C@]3([C@@H]4C[C@@H]4C5=C3[C@H]2O[C@@H]5O)C)OC1=O
InChI InChI=1S/C15H16O4/c1-5-9-8(18-13(5)16)4-15(2)7-3-6(7)10-11(15)12(9)19-14(10)17/h6-8,12,14,17H,3-4H2,1-2H3/t6-,7+,8-,12-,14-,15-/m0/s1
InChI Key IIFNVNIPMCRQPC-YIEVAYSQSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C15H16O4
Molecular Weight 260.28 g/mol
Exact Mass 260.10485899 g/mol
Topological Polar Surface Area (TPSA) 55.80 Ų
XlogP -0.10

Synonyms

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CHEBI:70172
Chlorajapolide B
CHEMBL1668790
SCHEMBL30190141
Q27138513

2D Structure

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2D Structure of Chlorajapolide B, (rel)-

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 91.72% 95.56%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 91.59% 85.14%
CHEMBL3137262 O60341 LSD1/CoREST complex 91.08% 97.09%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 90.53% 99.23%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 89.60% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 88.53% 96.09%
CHEMBL253 P34972 Cannabinoid CB2 receptor 86.96% 97.25%
CHEMBL1994 P08235 Mineralocorticoid receptor 83.92% 100.00%
CHEMBL1293249 Q13887 Kruppel-like factor 5 83.47% 86.33%
CHEMBL1806 P11388 DNA topoisomerase II alpha 82.47% 89.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Chloranthus serratus

Cross-Links

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PubChem 50993898
NPASS NPC319861
ChEMBL CHEMBL1668790
LOTUS LTS0094472
wikiData Q27138513